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Discovery of a new 1-(phenylsulfonyl)-1H-indole derivative targeting the EphA2 receptor with antiproliferative activity on U251 glioblastoma cell line 在U251胶质母细胞瘤细胞系上发现具有抗增殖活性的靶向EphA2受体的新1-(苯磺酰基)-1h-吲哚衍生物 Guidetti, Lorenzo; Castelli, Riccardo; Zappia, Alfonso; Ferrari, Francesca Romana; Giorgio, Carmine; Barocelli, Elisabetta; Pagliaro, Luca; Vento, Federica; Roti, Giovanni; Scalvini, Laura; Vacondio, Federica; Rivara, Silvia; Mor, Marco; Lodola, Alessio; Tognolini, Massimiliano 分享 收藏
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Pharmacological characterization of second generation FXR agonists as effective EphA2 antagonists: A successful application of target hopping approach Ferrari, Francesca Romana; Giorgio, Carmine; Zappia, Alfonso; Ballabeni, Vigilio; Bertoni, Simona; Barocelli, Elisabetta; Scalvini, Laura; Galvani, Francesca; Mor, Marco; Lodola, Alessio; Tognolini, Massimiliano 分享 收藏
Discovery of small-molecules targeting the CCL20/CCR6 axis as first-in-class inhibitors for inflammatory bowel diseases Martina, Maria Grazia; Giorgio, Carmine; Allodi, Marika; Palese, Simone; Barocelli, Elisabetta; Ballabeni, Vigilio; Szpakowska, Martyna; Chevigne, Andy; van Hamburg, Jan Piet; Davelaar, Nadine; Lubberts, Erik; Bertoni, Simona; Radi, Marco 分享 收藏
UniPR1331: Small Eph/Ephrin Antagonist Beneficial in Intestinal Inflammation by Interfering with Type-B Signaling UniPR1331: 小Eph/Ephrin拮抗剂通过干扰b型信号有益于肠道炎症 Giorgio, Carmine; Allodi, Marika; Palese, Simone; Grandi, Andrea; Tognolini, Massimiliano; Castelli, Riccardo; Lodola, Alessio; Flammini, Lisa; Cantoni, Anna Maria; Barocelli, Elisabetta; Bertoni, Simona 分享 收藏
Increased Mucosal Thrombin is Associated with Crohn's Disease and Causes Inflammatory Damage through Protease-activated Receptors Activation 粘膜凝血酶增加与克罗恩病相关,并通过蛋白酶激活受体激活引起炎症损伤 Motta, Jean-Paul; Palese, Simone; Giorgio, Carmine; Chapman, Kevin; Denadai-Souza, Alexandre; Rousset, Perrine; Sagnat, David; Guiraud, Laura; Edir, Anissa; Seguy, Carine; Alric, Laurent; Bonnet, Delphine; Bournet, Barbara; Buscail, Louis; Gilletta, Cyrielle; Buret, Andre G.; Wallace, John L.; Hollenberg, Morley D.; Oswald, Eric; Barocelli, Elisabetta; Le Grand, Sylvie; Le Grand, Bruno; Deraison, Celine; Vergnolle, Nathalie 分享 收藏
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Therapeutic Intervention Targeting Mucosal Thrombin Or Protease-Activated-Receptor 1 Are Protective Against Colitis Motta, Jean-Paul; Palese, Simone; Sagnat, David; Rousset, Perrine; Guiraud, Laura; Edir, Anissa; Seguy, Carine; Alric, Laurent; Bonnet, Delphine; Bournet, Barbara; Buscail, Louis; Gilletta, Cyrielle; Barocelli, Elisabetta; Le Grand, Sylvie; Le Grand, Bruno; Deraison, Celine; Vergnolle, Nathalie 分享 收藏
Evaluation of the Anti-Tumor Activity of Small Molecules Targeting Eph/Ephrins in APC min/J Mice Corrado, Miriam; Giorgio, Carmine; Barocelli, Elisabetta; Vittucci Marzetti, Giuseppe; Cantoni, Anna Maria; Di Lecce, Rosanna; Incerti, Matteo; Castelli, Riccardo; Lodola, Alessio; Tognolini, Massimiliano 分享 收藏
Third generation EGFR inhibitor osimertinib combined with pemetrexed or cisplatin exerts long-lasting anti-tumor effect in EGFR-mutated pre-clinical models of NSCLC La Monica, Silvia; Minari, Roberta; Cretella, Daniele; Flammini, Lisa; Fumarola, Claudia; Bonelli, Mara; Cavazzoni, Andrea; Digiacomo, Graziana; Galetti, Maricla; Madeddu, Denise; Falco, Angela; Lagrasta, Costanza Annamaria; Squadrilli, Anna; Barocelli, Elisabetta; Romanel, Alessandro; Quaini, Federico; Petronini, Pier Giorgio; Tiseo, Marcello; Alfieri, Roberta 分享 收藏
Inhibition of Eph/ephrin interaction with the small molecule UniPR500 improves glucose tolerance in healthy and insulin-resistant mice Giorgio, C.; Incerti, M.; Pala, D.; Russo, S.; Chiodelli, P.; Rusnati, M.; Cantoni, A. M.; Di Lecce, R.; Barocelli, E.; Bertoni, S.; Ravassard, P.; Manenti, F.; Piemonti, L.; Ferlenghi, F.; Lodola, A.; Tognolini, M. 分享 收藏
3D-printed chitosan-based scaffolds: An in vitro study of human skin cell growth and an in-vivo wound healing evaluation in experimental diabetes in rats Intini, Claudio; Elviri, Lisa; Cabral, Jaydee; Mros, Sonya; Bergonzi, Carlo; Bianchera, Annalisa; Flammini, Lisa; Govoni, Paolo; Barocelli, Elisabetta; Bettini, Ruggero; McConnell, Michelle 分享 收藏
Combined hyaluronate-based films loaded with pemetrexed and cisplatin for the treatment of malignant pleural mesothelioma: Preliminary evaluation in an orthotopic tumor recurrence model Sonvico, Fabio; Barbieri, Stefano; Colombo, Paolo; Barocelli, Elisabetta; Mucchino, Claudio; Cantoni, Anna Maria; Petronini, Pier Giorgio; Rusca, Michele; Carbognani, Paolo; Ampollini, Luca 分享 收藏
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