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Synthesis and Evaluation of Fluorinated Piperazine-Hydroxyethylamine Analogues as Potential Antiplasmodial Candidates Upadhyay, Charu; Bhattacharya, Shreya; Kumar, Sumit; Vashisht, Kapil; Zhang, Xujie; Gagnon, Dominic; Singh, Pooja; Zhan, Peng; Richard, Dave; Rathi, Brijesh; Singh, Agam Prasad; Singh, Priyamvada 分享 收藏
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Discovery of low-molecular-weight phenylalanine derivatives as novel HIV capsid modulators with improved antiretroviral activity and metabolic stability Jiang, Xiangyi; Gao, Zhen; Sharma, Prem Prakash; Kumar, Sumit; Rathi, Brijesh; Ji, Xiangkai; Dai, Jiaojiao; Xie, Minghui; Dong, Guanyu; Xu, Shujing; De Clercq, Erik; Pannecouque, Christophe; Dick, Alexej; Zhan, Peng; Liu, Xinyong 分享 收藏
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Biological activity of 1,2,3-triazole-2-amino-1,4-naphthoquinone derivatives and their evaluation as therapeutic strategy for malaria control Souza, Renata Maria Costa; Pimentel, Lilian Maria Lapa Montenegro; Ferreira, Laryssa Kathleen Mendonca; Pereira, Valeria Rego Alves; Santos, Aline Caroline Da Silva; Dantas, Willyenne Marilia; Silva, Carla Jasmine Oliveira; Brito, Ramayana Morais De Medeiros; Andrade, Jose Lucas; De Andrade-Neto, Valter Ferreira; Fujiwara, Ricardo Toshio; Bueno, Lilian Lacerda; Silva Junior, Valdemiro Amaro; Pena, Lindomar; Camara, Celso Amorim; Rathi, Brijesh; De Oliveira, Ronaldo Nascimento 分享 收藏
Escaping from Flatland: Multiparameter Optimization Leads to the Discovery of Novel Tetrahydropyrido[4,3-d]pyrimidine Derivatives as Human Immunodeficiency Virus-1 Non-nucleoside Reverse Transcriptase Inhibitors with Superior Antiviral Activities against Non-nucleoside Reverse Transcriptase Inhibitor-Resistant Variants and Favorable Drug-like Profiles 逃离Flatland: 多参数优化导致发现新型四氢吡啶并 [4,3-d] 嘧啶衍生物作为人类免疫缺陷病毒-1非核苷类逆转录酶抑制剂,对非核苷类逆转录酶抑制剂耐药变体具有优异的抗病毒活性和良好的药物样概况 Wang, Zhao; Sharma, Prem Prakash; Rathi, Brijesh; Xie, Minghui; De Clercq, Erik; Pannecouque, Christophe; Kang, Dongwei; Zhan, Peng; Liu, Xinyong 分享 收藏
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