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K

Karla Frydenvang

University of Copenhagen
H指数:28
被引数:2,683

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荣誉奖项

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Structure-guided optimization of 3-hydroxybenzoisoxazole derivatives as inhibitors of Aldo-keto reductase 1C3 (AKR1C3) to target prostate cancer

3-羟基苯并异恶唑衍生物作为醛酮还原酶1C3 (AKR1C3) 抑制剂靶向前列腺癌的结构指导优化

EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
IF5.9
2024-03-014
OAAI
Pippione, Agnese Chiara; Kovachka, Sandra; Vigato, Chiara; Bertarini, Laura; Mannella, Iole; Sainas, Stefano; Rolando, Barbara; Denasio, Enrica; Piercy-Mycock, Helen; Romalho, Linda; Salladini, Edoardo; Adinolfi, Salvatore; Zonari, Daniele; Peraldo-Neia, Caterina; Chiorino, Giovanna; Passoni, Alice; Mirza, Osman Asghar; Frydenvang, Karla; Pors, Klaus; Lolli, Marco Lucio; Spyrakis, Francesca; Oliaro-Bosso, Simonetta; Boschi, Donatella
Exploring thienothiadiazine dioxides as isosteric analogues of benzo- and pyridothiadiazine dioxides in the search of new AMPA and kainate receptor positive allosteric modulators
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
IF5.9
2024-01-010
OAAI
Francotte, Pierre; Bay, Yasmin; Goffin, Eric; Colson, Thomas; Lesenfants, Cindy; Dorosz, Jerzy; Laulumaa, Saara; Fraikin, Pierre; de Tullio, Pascal; Beaufour, Caroline; Botez, Iuliana; Pickering, Darryl S.; Frydenvang, Karla; Danober, Laurence; Kristensen, Anders Skov; Kastrup, Jette Sandholm; Pirotte, Bernard
N-(7-(1H-Imidazol-1-yl)-2,3-dioxo-6-(trifluoromethyl)-3,4-dihydroquinoxalin-1(2H)-yl)benzamide, a New Kainate Receptor Selective Antagonist and Analgesic: Synthesis, X-ray Crystallography, Structure-Affinity Relationships, and in Vitro and in Vivo Pharmacology
ACS CHEMICAL NEUROSCIENCE
IF3.9
2019-10-179
PREAI
Mollerud, Stine; Hansen, Rie B.; Pallesen, Jakob; Temperini, Piero; Pasini, Diletta; Bornholt, Jan; Nielsen, Birgitte; Mamedova, Esmira; Chalupnik, Paulina; Paternain, Ana V.; Lerma, Juan; Diaz-delCastillo, Marta; Andreasen, Jesper T.; Frydenvang, Karla; Kastrup, Jette S.; Johansen, Tommy N.; Pickering, Darryl S.
Five-Membered N-Heterocyclic Scaffolds as Novel Amino Bioisosteres at γ-Aminobutyric Acid (GABA) Type A Receptors and GABA Transporters
JOURNAL OF MEDICINAL CHEMISTRY
IF6.8
2019-05-2219
OAAI
Giraudo, Alessandro; Krall, Jacob; Bavo, Francesco; Nielsen, Birgitte; Kongstad, Kenneth T.; Rolando, Barbara; De Blasio, Rossella; Gloriam, David E.; Loftier, Rebekka; Thiesen, Louise; Harpsoe, Kasper; Frydenvang, Karla; Boschi, Donatella; Wellendorph, Petrine; Lolli, Marco L.; Jensen, Anders A.; Frolund, Bente
(S)-2-Amino-3-(5-methyl-3-hydroxyisoxazol-4-yl)propanoic Acid (AMPA) and Kainate Receptor Ligands: Further Exploration of Bioisosteric Replacements and Structural and Biological Investigation
JOURNAL OF MEDICINAL CHEMISTRY
IF6.8
2018-02-1620
OAAI
Brogi, Simone; Brindisi, Margherita; Butini, Stefania; Kshirsagar, Giridhar U.; Maramai, Samuele; Chemi, Giulia; Gemma, Sandra; Campiani, Giuseppe; Novellino, Ettore; Fiorenzani, Paolo; Pinassi, Jessica; Alois, Anna Maria; Gynther, Mikko; Venskutonyte, Raminta; Han, Liwei; Frydenvang, Karla; Kastrup, Jette Sandholm; Pickering, Darryl S.
7-Phenoxy-Substituted 3,4-Dihydro-2H-1,2,4-benzothiadiazine 1,1-Dioxides as Positive Allosteric Modulators of α-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid (AMPA) Receptors with Nanomolar Potency
JOURNAL OF MEDICINAL CHEMISTRY
IF6.8
2017-12-1941
OAAI
Goffin, Eric; Drapier, Thomas; Larsen, Anja Probst; Geubelle, Pierre; Ptak, Christopher P.; Laulumaa, Saara; Rovinskaja, Karoline; Gilissen, Julie; de Tullio, Pascal; Olsen, Lars; Frydenvang, Karla; Pirotte, Bernard; Hanson, Julien; Oswald, Robert E.; Kastrup, Jette Sandholm; Francotte, Pierre

研究方向

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J
J.S. Kastrup
H 指数:42论文数:253被引数:5,194
D
Darryl S. Pickering
H 指数:31论文数:166被引数:3,123
B
Birgitte Nielsen
H 指数:34论文数:257被引数:5,122
M
Michael Gajhede
H 指数:47论文数:317被引数:7,970
L
Lennart Bunch
H 指数:25论文数:117被引数:2,691
P
Povl Krogsgaard‐Larsen
H 指数:60论文数:758被引数:1.6万
B
Bernard Pirotte
H 指数:41论文数:708被引数:5,293
R
Raminta Venskutonytė
H 指数:14论文数:37被引数:525
T
Tommy N. Johansen
H 指数:24论文数:86被引数:1,455
P
Pierre Francotte
H 指数:19论文数:116被引数:934