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Povl Krogsgaard-Larsen

University of Copenhagen

H指数:60

被引数:1.6万

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Probing the Orthosteric Binding Site of GABAA Receptors with Heterocyclic GABA Carboxylic Acid Bioisosteres

NEUROCHEMICAL RESEARCH

IF3.8

2013-12-2117

PREAI

The orthosteric GABAA receptor ligand Thio-4-PIOL displays distinctly different functional properties at synaptic and extrasynaptic receptors

BRITISH JOURNAL OF PHARMACOLOGY

IF7.7

2013-10-0116

OAAI

Selective mGAT2 (BGT-1) GABA Uptake Inhibitors: Design, Synthesis, and Pharmacological Characterization

JOURNAL OF MEDICINAL CHEMISTRY

IF6.8

2013-02-2737

PREAI

Design, Synthesis, and Pharmacological Characterization of N- and O-Substituted 5,6,7,8-Tetrahydro-4H-isoxazolo[4,5-d]azepin-3-ol Analogues: Novel 5-HT2A/5-HT2C Receptor Agonists with Pro-Cognitive Properties

JOURNAL OF MEDICINAL CHEMISTRY

IF6.8

2013-01-1752

PREAI

Scientific Social Responsibility: A Call to Arms

ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

IF16.9

2011-10-1010

OAAI

Selective GABA Transporter Inhibitors Tiagabine and EF1502 Exhibit Mechanistic Differences in Their Ability to Modulate the Ataxia and Anticonvulsant Action of the Extrasynaptic GABAA Receptor Agonist Gaboxadol

JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS

IF3.8

2011-07-0147

OAAI

Biostructural and Pharmacological Studies of Bicyclic Analogues of the 3-Isoxazolol Glutamate Receptor Agonist Ibotenic Acid

JOURNAL OF MEDICINAL CHEMISTRY

IF6.8

2010-11-1019

PREAI

The Glutamate Receptor GluR5 Agonist (S)-2-Amino-3-(3-hydroxy-7,8-dihydro-6H-cyclohepta[d]isoxazol-4-yl)propionic Acid and the 8-Methyl Analogue: Synthesis, Molecular Pharmacology, and Biostructural Characterization

JOURNAL OF MEDICINAL CHEMISTRY

IF6.8

2009-07-0923

PREAI

Detecting Protein-Protein Interactions in Living Cells: Development of a Bioluminescence Resonance Energy Transfer Assay to Evaluate the PSD-95/NMDA Receptor Interaction

检测活细胞中的蛋白质-蛋白质相互作用: 开发生物发光共振能量转移测定法以评估PSD-95/NMDA受体相互作用

NEUROCHEMICAL RESEARCH

IF3.8

2009-06-049

PREAI

Pharmacology of (S)-homoquisqualic acid and (S)-2-amino-5-phosphonopentanoic acid [(S)-AP5] at cloned metabotropic glutamate receptors

在克隆的代谢型谷氨酸受体上的 (S)-高奎尼酸和 (S)-2-氨基-5-膦酰基戊酸 [(S)-AP5] 的药理学

BRITISH JOURNAL OF PHARMACOLOGY

IF7.7

2009-02-0353

OAAI

Functional pharmacology of cloned heterodimeric GABAB receptors expressed in mammalian cells

BRITISH JOURNAL OF PHARMACOLOGY

IF7.7

2009-01-3039

OAAI

Subtype Selective Kainic Acid Receptor Agonists: Discovery and Approaches to Rational Design

MEDICINAL RESEARCH REVIEWS

IF11.6

2008-07-1153

PREAI

5-substituted imidazole-4-acetic acid analogues:: Synthesis, modeling, and pharmacological characterization of a series of novel γ-aminobutyric AcidC receptor agonists

JOURNAL OF MEDICINAL CHEMISTRY

IF6.8

2007-07-2653

PREAI

Novel 5-substituted 1-pyrazolol analogues of ibotenic acid:: Synthesis and pharmacology at glutamate receptors

BIOORGANIC & MEDICINAL CHEMISTRY

IF3

2007-05-0112

PRE

A tetrazolyl-substituted subtype-selective AMPA receptor agonist

JOURNAL OF MEDICINAL CHEMISTRY

IF6.8

2007-04-2527

PREAI

4-aryl-5-(4-piperidyl)-3-isoxazolol GABAA antagonists:: Synthesis, pharmacology, and structure-activity relationships

JOURNAL OF MEDICINAL CHEMISTRY

IF6.8

2007-03-2238

PREAI

A novel selective γ-aminobutyric acid transport inhibitor demonstrates a functional role for GABA transporter subtype GAT2/BGT-1 in the CNS

NEUROCHEMISTRY INTERNATIONAL

IF4

2006-05-0137

PREAI

Potent 4-arylalkyl-substituted 3-isothiazolol GABAA competitive/noncompetitive antagonists: Synthesis and pharmacology

JOURNAL OF MEDICINAL CHEMISTRY

IF6.8

2006-01-2132

PREAI

Medicinal chemistry education: What is needed and where is it going?

DRUG DEVELOPMENT RESEARCH

IF4.2

2006-01-0111

PREAI

Tetrazolyl isoxazole amino acids as ionotropic glutamate receptor antagonists:: Synthesis, modelling and molecular pharmacology

BIOORGANIC & MEDICINAL CHEMISTRY

IF3

2005-09-0111

PRE