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Carrie K. Jones

vanderbilt university

53H指数
271论文数
8.6K被引数
收录论文 107
发表时间
Drug Repurposing: Conversion of the Peripherally Restricted HIV Protease Inhibitor Amprenavir to Potent; Selective; and CNS-Penetrant Agonists for the Cannabinoid Receptor 2
err2026-02-05
err0
errOAAI
errDaniel H. Haymer; Renn A. Duncan; Alice L. Rodriguez; Allie Han; Richard J. Lindsay; N. Kithmini Wijesiri; Analisa Thompson Gray; Srinivasan Krishnan; Aidong Qi; Benjamin P. Brown; Olivier Boutaud; Darren W. Engers; Carrie K. Jones; Colleen M. Niswender; Craig W. Lindsley; Aaron M. Bender
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Discovery of VU6052254: A Novel; Potent M1 Positive Allosteric ModulatorVU6052254的发现:一种新型的强效M1正向别构调节剂
err2025-11-26
err0
errOAAI
errJulie L. Engers; Joseph D. Bungard; Christopher C. Presley; Irene Zagol-Ikapitte; Katherine J. Watson; Sichen Chang; Colin O’Carroll; P. Markus Dey; Ethan S. Burstein; Jonathan W. Dickerson; Analisa Thompson Gray; Michael Bubser; Jerri M. Rook; Hyekyung P. Cho; Valerie M. Kramlinger; Olivier Boutaud; Carrie K. Jones; P. Jeffrey Conn; Darren W. Engers; Craig W. Lindsley
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Optimization of Selective and CNS Penetrant Alkyne-Based TREK Inhibitors: The Discovery and Characterization of ONO-9517601 (VU6022856) and ONO-7927846 (VU6024391)
err2025-10-01
err0
PREAI
errTanaka, Motoyuki; Sekioka, Yoko; Hashimoto, Gakuji; Mori, Takahiro; Shono, Tomoyuki; Isaji, Yuuki; Hisaichi, Katsuya; Childress, Elizabeth S.; Bollinger, Sean; Schmitt, Joza A.; Chopko, Trevor C.; Garrison, Aaron T.; Perry, Charles K.; Chronister, Keagan; Kramer, Meghan; Chang, Sichen; Watson, Katherine J.; Dickerson, Jonathan W.; Bubser, Michael; Rook, Jerri M.; Jones, Carrie K.; Boutaud, Olivier; Bridges, Thomas M.; Denton, Jerod S.; Engers, Darren W.; Kurata, Haruto; Lindsley, Craig W.
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Shank3 modulates Rpl3 expression and protein synthesis via mGlu5: implications for Phelan McDermid syndromeShank3通过mGlu5调节Rpl3的表达和蛋白质合成:对Phelan McDermid综合征的启示
err2025-03-15
err0
errOAAI
errGiona, Federica; Beretta, Stefania; Zippo, Antonio; Stefanoni, Alessia; Tomasoni, Zaira; Vicidomini, Cinzia; Ponzoni, Luisa; Sala, Mariaelvina; Jones, Carrie K.; Conn, P. Jeffrey; Boeckers, Tobias M.; Sala, Carlo; Verpelli, Chiara
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Discovery of VU0467319: an M1 Positive Allosteric Modulator Candidate That Advanced into Clinical Trials
err2024-12-11
err0
errOAAI
errPoslunsey, Michael S.; Wood, Michael R.; Han, Changho; Stauffer, Shaun R.; Panarese, Joseph D.; Melancon, Bruce J.; Engers, Julie L.; Dickerson, Jonathan W.; Peng, Weimin; Noetzel, Meredith J.; Cho, Hyekyung P.; Rodriguez, Alice L.; Hopkins, Corey R.; Morrison, Ryan; Crouch, Rachel D.; Bridges, Thomas M.; Blobaum, Anna L.; Boutaud, Olivier; Daniels, J. Scott; Kates, Michael J.; Castelhano, Arlindo; Rook, Jerri M.; Niswender, Colleen M.; Jones, Carrie K.; Conn, P. Jeffrey; Lindsley, Craig W.
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Discovery of 4-(5-Membered)Heteroarylether-6-methylpicolinamide Negative Allosteric Modulators of Metabotropic Glutamate Receptor Subtype 5
err2024-11-18
err0
errOAAI
errChildress, Elizabeth S.; Capstick, Rory A.; Crocker, Katherine E.; Ledyard, Miranda L.; Bender, Aaron M.; Maurer, Mallory A.; Billard, Natasha B.; Cho, Hyekyung P.; Rodriguez, Alice L.; Niswender, Colleen M.; Peng, Weimin; Rook, Jerri M.; Chang, Sichen; Blobaum, Anna L.; Boutaud, Olivier; Thompson Gray, Analisa; Jones, Carrie K.; Conn, P. Jeffrey; Felts, Andrew S.; Lindsley, Craig W.; Temple, Kayla J.
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Discovery of VU6016235: A Highly Selective, Orally Bioavailable, and Structurally Distinct Tricyclic M4 Muscarinic Acetylcholine Receptor Positive Allosteric Modulator (PAM)
err2024-09-24
err0
errOAAI
errEngers, Julie L.; Baker, Logan A.; Chang, Sichen; Luscombe, Vincent B.; Rodriguez, Alice L.; Niswender, Colleen M.; Cho, Hyekyung P.; Bubser, Michael; Gray, Analisa Thompson; Jones, Carrie K.; Peng, Weimin; Rook, Jerri M.; Bridges, Thomas M.; Boutaud, Olivier; Conn, P. Jeffrey; Engers, Darren W.; Lindsley, Craig W.; Temple, Kayla J.
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Development of VU6036864: A Triazolopyridine-Based High-Quality Antagonist Tool Compound of the M5 Muscarinic Acetylcholine Receptor
err2024-08-06
err0
errOAAI
errLi, Jinming; Orsi, Douglas L.; Engers, Julie L.; Long, Madeline F.; Capstick, Rory A.; Maurer, Mallory A.; Presley, Christopher C.; Vinson, Paige N.; Rodriguez, Alice L.; Han, Allie; Cho, Hyekyung P.; Chang, Sichen; Jackson, Megan; Bubser, Michael; Blobaum, Anna L.; Boutaud, Olivier; Nader, Michael A.; Niswender, Colleen M.; Conn, P. Jeffrey; Jones, Carrie K.; Lindsley, Craig W.; Han, Changho
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Evaluation of the Indazole Analogs of 5-MeO-DMT and Related Tryptamines as Serotonin Receptor 2 Agonists
err2024-01-19
err1
errOAAI
errJayakodiarachchi, Navoda; Maurer, Mallory A.; Schultz, Daniel C.; Dodd, Cayden J.; Gray, Analisa Thompson; Cho, Hyekyung P.; Boutaud, Olivier; Jones, Carrie K.; Lindsley, Craig W.; Bender, Aaron M.
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M1/M4-Preferring Muscarinic Cholinergic Receptor Agonist Xanomeline Reverses Wake and Arousal Deficits in Nonpathologically Aged Mice
err2023-01-19
err7
errOAAI
errRussell, Jason K.; Ingram, Shalonda M.; Teal, Laura B.; Lindsley, Craig W.; Jones, Carrie K.
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Development of VU6019650: A Potent, Highly Selective, andSystemically Active Orthosteric Antagonist of the M5MuscarinicAcetylcholine Receptor for the Treatment of Opioid Use Disorder
err2022-04-13
err9
PREAI
errGarrison, Aaron T.; Orsi, Douglas L.; Capstick, Rory A.; Whomble, David; Li, Jinming; Carter, Trever R.; Felts, Andrew S.; Vinson, Paige N.; Rodriguez, Alice L.; Han, Allie; Hajari, Krishma; Cho, Hyekyung P.; Teal, Laura B.; Ragland, Madeline G.; Ghamari-Langroudi, Masoud; Bubser, Michael; Chang, Sichen; Schnetz-Boutaud, Nathalie C.; Boutaud, Olivier; Blobaum, Anna L.; Foster, Daniel J.; Niswender, Colleen M.; Conn, P. Jeffrey; Lindsley, Craig W.; Jones, Carrie K.; Han, Changho
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Partial mGlu5 Negative Allosteric Modulator M-5MPEP Demonstrates Antidepressant-Like Effects on Sleep Without Affecting Cognition or Quantitative EEG部分mGlu5负性变构调节剂M-5MPEP对睡眠表现出抗抑郁样作用,而不影响认知或定量脑电图
err2021-07-02
err8
errOAAI
errHolter, Kimberly M.; Lekander, Alex D.; LaValley, Christina M.; Bedingham, Elizabeth G.; Pierce, Bethany E.; Sands, L. Paul; Lindsley, Craig W.; Jones, Carrie K.; Gould, Robert W.
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Acetylcholine Muscarinic M4 Receptors as a Therapeutic Target for Alcohol Use Disorder: Converging Evidence From Humans and Rodents
err2020-12-01
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errOAAI
errWalker, Leigh C.; Berizzi, Alice E.; Chen, Nicola A.; Rueda, Patricia; Perreau, Victoria M.; Huckstep, Katherine; Srisontiyakul, Jirawoot; Govitrapong, Piyarat; Jia Xiaojian; Lindsley, Craig W.; Jones, Carrie K.; Riddy, Darren M.; Christopoulos, Arthur; Langmead, Christopher J.; Lawrence, Andrew J.
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Modulation of arousal and sleep/wake architecture by M1PAM VU0453595 across young and aged rodents and nonhuman primates
err2020-08-31
err17
errOAAI
errGould, Robert W.; Russell, Jason K.; Nedelcovych, Michael T.; Bubser, Michael; Blobaum, Anna L.; Bridges, Thomas M.; Newhouse, Paul A.; Lindsley, Craig W.; Conn, P. Jeffrey; Nader, Michael A.; Jones, Carrie K.
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The Effects of the M1 Muscarinic Acetylcholine Receptor Positive Allosteric Modulator VU0486846 on Cognitive Performance in Aged Nonhuman Primates
err2020-04-19
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PREAI
errNorman, Christina; Gould, Robert; Bragg, Chrystal; Lindsley, Craig; Jones, Carrie; Nader, Michael
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Acute Negative Allosteric Modulation of M5 Muscarinic Acetylcholine Receptors Inhibits Oxycodone Self-Administration and Cue-Induced Reactivity with No Effect on Antinociception
err2019-07-03
err26
errOAAI
errGould, Robert W.; Gunter, Barak W.; Bubser, Michael; Matthews, Robert T.; Teal, Laura B.; Ragland, Madeline G.; Bridges, Thomas M.; Garrison, Aaron T.; Winder, Danny G.; Lindsley, Craig W.; Jones, Carrie K.
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The Role of Estrogen in Brain and Cognitive Aging
err2019-07-01
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errOAAI
errRussell, Jason K.; Jones, Carrie K.; Newhouse, Paul A.
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Analgesic Effects of the GIRK Activator, VU0466551, Alone and in Combination with Morphine in Acute and Persistent Pain Models (vol 10, pg 1294, 2019)
err2019-03-26
err2
PREAI
errAbney, Kristopher K.; Bubser, Michael; Du, Yu; Kozek, Krystian A.; Bridges, Thomas M.; Lindsley, Craig W.; Daniels, J. Scott; Morrison, Ryan D.; Wickman, Kevin; Hopkins, Corey R.; Jones, Carrie K.; Weaver, C. David
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