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Cathepsin B-Cleavable Doxorubicin Prodrug Nanoparticles for Eliciting Cancer-Specific Immunogenic Cell Death and Minimizing Systemic Toxicity 组织蛋白酶B可切割的阿霉素前药纳米颗粒,用于诱导癌症特异性免疫原性细胞死亡并减少全身毒性 Shim, Nayeon; Kim, Jinseong; Song, Sukyung; Yoo, Hyeonji; Kim, Yeonjin; Oh, Yoojeong; Hwang, Namcheol; Goo, Jagyeong; Hong, Seeun; Yu, Jinha; Cho, Hanhee; Kim, Kwangmeyung 分享 收藏
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Steric influence of 4′-position substituents and C2-Hexynyl group on A3AR antagonism in truncated 4′-Thioadenosine derivatives 4′位取代基和C2-己炔基对截短型4′-硫代腺苷衍生物中A3AR拮抗作用的空间影响 Kim, Minjae; Kim, Jina; Tripathi, Sushil K.; Aswar, Vikas R.; Gaikwad, Vidyasagar; Song, Jiyoon; Kim, Meehyein; Yu, Jinha; Chang, Tong-Shin; Jeong, Lak Shin 分享 收藏
Exploring C2 and N6 Substituent Effects on Truncated 4′-Thioadenosine Derivatives as Dual A2A and A3 Adenosine Receptor Ligands Naik, Siddhi D.; Kim, Minjae; Choi, Jiyoung; Kim, Gibae; Woo Kim, Seung; Aswar, Vikas R.; Tripathi, Sushil K.; Gaikwad, Vidyasagar; Yu, Jinha; Jeong, Lak Shin 分享 收藏
Structural Modification and Biological Evaluation of 2,8-Disubstituted Adenine and Its Nucleosides as A2A Adenosine Receptor Antagonists: Exploring the Roles of Ribose at Adenosine Receptors Kim, Gibae; Jarhad, Dnyandev B.; Lee, Grim; Kim, Gyudong; Hou, Xiyan; Yu, Jinha; Lee, Chang Soo; Warnick, Eugene; Gao, Zhan-Guo; Ahn, Sang Yeop; Kwak, Dongik; Park, Kichul; Lee, Summer Dabin; Park, Tae-uk; Jung, So-young; Lee, Jong Hyun; Choi, Jong-Ryoul; Kim, Myeongjoong; Kim, Donghyun; Kim, Bongtae; Jacobson, Kenneth A.; Jeong, Lak Shin 分享 收藏
Structure-Activity Relationship of Truncated 2,8-Disubstituted-Adenosine Derivatives as Dual A2A/A3 Adenosine Receptor Antagonists and Their Cancer Immunotherapeutic Activity (vol 66, pg 12249, 2023) Kim, Gibae; Hou, Xiyan; Byun, Woong Sub; Kim, Gyudong; Jarhad, Dnyandev B.; Lee, Grim; Hyun, Young Eum; Yu, Jinha; Lee, Chang Soo; Qu, Shuhao; Warnick, Eugene; Gao, Zhan-Guo; Kim, Ji Yong; Ji, Seunghee; Shin, Hyunwoo; Choi, Jong-Ryoul; Jacobson, Kenneth A.; Lee, Hyuk Woo; Lee, Sang Kook; Jeong, Lak Shin 分享 收藏
Structure-Activity Relationship of Truncated 2,8-Disubstituted-Adenosine Derivatives as Dual A2A/A3 Adenosine Receptor Antagonists and Their Cancer Immunotherapeutic Activity Kim, Gibae; Hou, Xiyan; Byun, Woong Sub; Kim, Gyudong; Jarhad, Dnyandev B.; Lee, Grim; Hyun, Young Eum; Yu, Jinha; Lee, Chang Soo; Qu, Shuhao; Warnick, Eugene; Gao, Zhan-Guo; Kim, Ji Yong; Ji, Seunghee; Shin, Hyunwoo; Choi, Jong-Ryoul; Jacobson, Kenneth A.; Lee, Hyuk Woo; Lee, Sang Kook; Jeong, Lak Shin 分享 收藏
GPCR Agonist-to-Antagonist Conversion: Enabling the Design of Nucleoside Functional Switches for the A2A Adenosine Receptor Shiriaeva, Anna; Park, Daejin; Kim, Gyudong; Lee, Yoonji; Hou, Xiyan; Jarhad, Dnyandev B.; Kim, Gibae; Yu, Jinha; Hyun, Young Eum; Kim, Woomi; Gao, Zhan-Guo; Jacobson, Kenneth A.; Han, Gye Won; Stevens, Raymond C.; Jeong, Lak Shin; Choi, Sun; Cherezov, Vadim 分享 收藏
Design, Synthesis and Biological Evaluation of 1,3,5-Triazine Derivatives Targeting hA1 and hA3 Adenosine Receptor Park, Sujin; Ahn, Yujin; Kim, Yongchan; Roh, Eun Joo; Lee, Yoonji; Han, Chaebin; Yoo, Hee Min; Yu, Jinha 分享 收藏
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Anticancer Effects of Propionic Acid Inducing Cell Death in Cervical Cancer Cells 丙酸诱导宫颈癌细胞死亡的抗癌作用 Pham, Chau Ha; Lee, Joo-Eun; Yu, Jinha; Lee, Sung Hoon; Yu, Kyung-Rok; Hong, Jaewoo; Cho, Namki; Kim, Seil; Kang, Dukjin; Lee, Soojin; Yoo, Hee Min 分享 收藏
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Discovery and Structure-Activity Relationships of Novel Template, Truncated 1′-Homologated Adenosine Derivatives as Pure Dual PPARγ/δ Modulators An, Seungchan; Kim, Gyudong; Kim, Hyun Jin; Ahn, Sungjin; Kim, Hyun Young; Ko, Hyejin; Hyun, Young Eum; Nguyen, Mai; Jeong, Juri; Liu, Zijing; Han, Jinhe; Choi, Hongseok; Yu, Jinha; Kim, Ji Won; Lee, Hyuk Woo; Jacobson, Kenneth A.; Cho, Won Jea; Kim, Young-Mi; Kang, Keon Wook; Noh, Minsoo; Jeong, Lak Shin 分享 收藏
Exploration of Alternative Scaffolds for P2Y14 Receptor Antagonists Containing a Biaryl Core Jung, Young-Hwan; Yu, Jinha; Wen, Zhiwei; Salmaso, Veronica; Karcz, Tadeusz P.; Phung, Ngan B.; Chen, Zhoumou; Duca, Sierra; Bennett, John M.; Dudas, Steven; Salvemini, Daniela; Gao, Zhan-Guo; Cook, Donald N.; Jacobson, Kenneth A. 分享 收藏
UBC12-mediatedSREBP-1 neddylation worsens metastatic tumor prognosis Heo, Mi Jeong; Kang, Sung Hyun; Kim, Yun Seok; Lee, Jung Min; Yu, Jinha; Kim, Hong-Rae; Lim, Hyesol; Kim, Kyoung Mee; Jung, Joohee; Jeong, Lak Shin; Moon, Aree; Kim, Sang Geon 分享 收藏
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