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Design, synthesis, and structure-activity relationship studies of 6H-benzo[b]indeno[1,2-d]thiophen-6-one derivatives as DYRK1A/CLK1/CLK4/haspin inhibitors Faouzi, Abdelfattah; Arnaud, Alexandre; Halle, Francois; Roussel, Jean; Aymard, Mandy; Denavit, Vincent; Do, Cong Viet; Mularoni, Angelique; Salah, Mohamed; ElHady, Ahmed; Pham, Thanh-Nhat; Bancet, Alexandre; Le Borgne, Marc; Terreux, Raphael; Barret, Roland; Engel, Matthias; Lomberget, Thierry 分享 收藏
Efficient synthesis, crystallographic study, antimicrobial activity and in silico studies of novel bioactive α-aminophosphonates based on pyridine moiety Grib, Ismahene; Berredjem, Malika; Djouad, Seif-Eddine; Benzaid, Chahrazed; Rachedi, Khadidja Otmane; Bahadi, Rania; Djendi, Lina Manel; Ibrahim-Ouali, Malika; Bouacida, Sofiane; Bachari, Khaldoun; Laichi, Yacine; Marminon, Christelle; Borgne, Marc L. E.; Bouasla, Radia 分享 收藏
New 2,4-bis[(substituted-aminomethyl)phenyl]phenylquinazoline and 2,4-bis[(substituted-aminomethyl)phenyl]phenylquinoline Derivatives: Synthesis and Biological Evaluation as Novel Anticancer Agents by Targeting G-Quadruplex 新的2，4-双 [(取代的氨基甲基) 苯基] 苯基喹唑啉和2，4-双 [(取代的氨基甲基) 苯基] 苯基喹啉衍生物: 通过靶向G-四链体作为新型抗癌剂的合成和生物学评估 Guillon, Jean; Le Borgne, Marc; Milano, Vittoria; Guedin-Beaurepaire, Aurore; Moreau, Stephane; Pinaud, Noel; Ronga, Luisa; Savrimoutou, Solene; Albenque-Rubio, Sandra; Marchivie, Mathieu; Kalout, Haouraa; Walker, Charley; Chevallier, Louise; Bure, Corinne; Largy, Eric; Gabelica, Valerie; Mergny, Jean-Louis; Baylot, Virginie; Ferrer, Jacky; Idrissi, Yamina; Chevret, Edith; Cappellen, David; Desplat, Vanessa; Schelz, Zsuzsanna; Zupko, Istvan 分享 收藏
Formulation and Investigation of CK2 Inhibitor-Loaded Alginate Microbeads with Different Excipients Papp, Boglarka; Le Borgne, Marc; Perret, Florent; Marminon, Christelle; Jozsa, Liza; Peto, Agota; Kosa, Dora; Nagy, Lajos; Keki, Sandor; Ujhelyi, Zoltan; Paller, Adam; Budai, Istvan; Bacskay, Ildiko; Feher, Palma 分享 收藏
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Inhibitors of ABCG2-mediated multidrug resistance: Lead generation through computer-aided drug design Goracci, Laura; Nurisso, Alessandra; Roussel, Emile; Peres, Basile; Chaptal, Vincent; Falson, Pierre; Marminon, Christelle; Jose, Joachim; Le Borgne, Marc; Boumendjel, Ahcene 分享 收藏
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Synthesis, in silico study (DFT, ADMET) and crystal structure of novel sulfamoyloxy-oxazolidinones: Interaction with SARS-CoV-2 Bouzina, Abdeslem; Berredjem, Malika; Bouacida, Sofiane; Bachari, Khaldoun; Marminon, Christelle; Le Borgne, Marc; Bouaziz, Zouhair; Bouone, Yousra Ouafa 分享 收藏
Broad-Spectrum Anticancer Activity and Pharmacokinetic Properties of a Prenyloxy-Substituted Indeno[1,2-b]indole Derivative, Discovered as CK2 Inhibitor El-Awaad, Ehab; Birus, Robin; Marminon, Christelle; Bouaziz, Zouhair; Ballentin, Laurens; Aichele, Dagmar; Le Borgne, Marc; Jose, Joachim 分享 收藏
Solubility enhancement of mefenamic acid by inclusion complex with β-cyclodextrin: in silico modelling, formulation, characterisation, and in vitro studies 通过与 β-环糊精的包合物提高甲芬那酸的溶解度: 计算机模拟，配方，表征和体外研究 Sid, Dounia; Baitiche, Milad; Elbahri, Zineb; Djerboua, Ferhat; Boutahala, Mokhtar; Bouaziz, Zouhair; Le Borgne, Marc 分享 收藏
Uncompetitive nanomolar dimeric indenoindole inhibitors of the human breast cancer resistance pump ABCG2 Guragossian, Nathalie; Belhani, Billel; Moreno, Alexis; Nunes, Magda Teixeira; Gonzalez-Lobato, Lucia; Marminon, Christelle; Berthier, Laurent; Pires, Amanda Do Rocio Andrade; Ozvegy-Laczka, Csilla; Sarkadi, Balazs; Terreux, Raphael; Bouaziz, Zouhair; Berredjem, Malika; Jose, Joachim; Di Pietro, Attilio; Falson, Pierre; Le Borgne, Marc 分享 收藏
Mechanistic basis of breast cancer resistance protein inhibition by new indeno[1,2-b]indoles Kita, Diogo Henrique; Guragossian, Nathalie; Zattoni, Ingrid Fatima; Moure, Vivian Rotuno; Rego, Fabiane Gomes de Moraes; Lusvarghi, Sabrina; Moulenat, Thomas; Belhani, Billel; Picheth, Geraldo; Bouacida, Sofiane; Bouaziz, Zouhair; Marminon, Christelle; Berredjem, Malika; Jose, Joachim; Goncalves, Marcos Brown; Ambudkar, Suresh V.; Valdameri, Glaucio; Le Borgne, Marc 分享 收藏
Ninhydrins inhibit carbonic anhydrases directly binding to the metal ion Bouzina, Abdeslem; Berredjem, Malika; Nocentini, Alessio; Bua, Silvia; Bouaziz, Zouhair; Jose, Joachim; Le Borgne, Marc; Marminon, Christelle; Gratteri, Paola; Supuran, Claudiu T. 分享 收藏
Synthesis, Optimization, Antifungal Activity, Selectivity, and CYP51 Binding of New 2-Aryl-3-azolyl-1-indolyl-propan-2-ols Lebouvier, Nicolas; Pagniez, Fabrice; Na, Young Min; Shi, Da; Pinson, Patricia; Marchivie, Mathieu; Guillon, Jean; Hakki, Tarek; Bernhardt, Rita; Yee, Sook Wah; Simons, Claire; Leze, Marie-Pierre; Hartmann, Rolf W.; Mularoni, Angelique; Le Baut, Guillaume; Krimm, Isabelle; Abagyan, Ruben; Le Pape, Patrice; Le Borgne, Marc 分享 收藏
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