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György M. Keserű

Hun-ren Research Centre for Natural Sciences

50H指数
417论文数
1.3W被引数
收录论文 182
发表时间
Cannabinoid-Inspired Fluorescent Boroisoquinolines for CB1 Receptor Imaging大麻素启发荧光硼异喹啉用于CB1受体成像
err2026-09-16
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errDénes Szepesi Kovács; Csilla Nierner; Bettina Szepesi Kovács; Attila Lehotzky; Edina Szűcs; András Dávid Tóth; Dóra Judit Kiss; László Hunyady; György M. Keserű; Péter Ábrányi-Balogh
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The structure of the dopamine D3 receptor bound to cariprazine reveals principles for partial agonists with designed pharmacology多巴胺D3受体与卡利拉赞结合的结构揭示了具有设计药理学特性的部分激动剂的原则
err2026-08-28
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errEliane Hadas Yardeni; Dóra Judit Kiss; Julie Sanchez; Keshet Shavit; Dénes Szepesi Kovács; Attila Egyed; Caleb D. Vogt; Supriya A. Gaitonde; Jacqueline Glenn; Meritxell Canals; Michel Bouvier; Amy Hauck Newman; J. Robert Lane; György M. Keserű; Moran Shalev-Benami
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Probing 3-Amino-2H-Azaindazoles as Allosteric Inhibitors of the Protein Tyrosine Phosphatase SHP2探究3-氨基-2H-氮杂吲哚唑作为蛋白酪氨酸磷酸酶SHP2的别构抑制剂
err2026-06-14
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errMachoud Amoussa; Nina-Louisa Efrém; Feng Li; Ziqiong Guo; Yvette Roske; Katrin Jana Frank; Szymon Pach; Clemens Alexander Wolf; Feng Bo; Marina Lesina; Mika Kintzel; Rana Alsalim; Victoria Zeitz; Noémi Csorba; Silke Radetzki; György M. Keserű; Oliver Daumke; Hana Algül; Gerhard Wolber; Jia Li; Marc Nazaré
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Fragment-Based Design of Targeted Covalent Inhibitors: The Scope and Limitation of Linking Approaches靶向共价抑制剂的片段基设计:连接策略的适用范围与局限性
err2026-05-22
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errLevente Kollár; Levente M. Mihalovits; Dávid Bajusz; Damijan Knez; József Simon; Blake H. Balcomb; Daren Fearon; Stanislav Gobec; György M. Keserű
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α-Halothioamide warheads with enhanced cysteine reactivity and specificity for covalent protein labellingα-卤代硫酰胺基团作为具有增强半胱氨酸反应性和特异性的共价蛋白质标记物
err2026-05-14
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errLászló Petri; Ronen Gabizon; Nikolett Péczka; Péter Ábrányi-Balogh; József Simon; Tímea Imre; György G. Ferenczy; Nir London; György M. Keserű
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Merging Micellar Catalysis and C-H Activation: Silver-Free Direct Arylation of Fluoroarenes in Water将胶束催化与C-H活化相结合:水中无银直接芳基化氟代芳烃
err2026-05-14
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errBelnome, Federico; Garami, Kristof N.; Varga, Zoltan; Mihaly, Judith; Hauk, Pascal; Hergert, Tamas; Keseru, Gyorgy M.; Gallou, Fabrice; Wencel-Delord, Joanna; Abranyi-Balogh, Peter
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Mapping the SHP2 Allosteric Pocket With Target-Biased Covalent Fragments靶向偏倚共价片段绘制SHP2别构口袋
err2026-04-24
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errNina-Louisa Efrém; Noémi Csorba; Machoud Amoussa; Péter Ábrányi-Balogh; Ziqiong Guo; László Petri; Feng Bo; Vincenzo Di Lorenzo; Yvette Roske; Tibor Viktor Szalai; Levente Mihalovits; József Simon; Jia Li; Oliver Daumke; György M. Keserű; Marc Nazaré
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Efficiency landscape of bioorthogonal click reactions producing bispecific antibody conjugates生物正交点击反应生产双特异性抗体偶联物的效率景观
err2026-04-21
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errLászló Petri; Írisz K. Kovács; Boglárka Szabó; Tímea Imre; Anita Rácz; Vijay Chudasama; Peter A. Szijj; György M. Keserű
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The Discovery of RGH-706; a Highly Efficacious MCH1 Receptor Antagonist; for the Treatment of Obesity and Insatiable Hunger
err2026-01-22
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errGyula Beke; András Boros; György M. Keserű; Balázs Krámos; Krisztina Katalin Szalai; Anikó Gere; Mónika Vastag; Márta Thán; Balázs Varga; Ottilia Balázs; Sándor Farkas; Balázs Lendvai; István Greiner; János Éles
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Covalent Activation of the C-type Lectin DC-SIGNC型凝集素dc-sign的共价活化
err2025-11-24
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errJonathan Lefèbre; Maurice Besch; Noémi Csorba; Kristóf Garami; Zoltán Orgován; Gitta Schlosser; Iris Bermejo; Péter Ábrányi-Balogh; György M. Keserű; Prof. Dr. Christoph Rademacher
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The impact of secondary site interactions on the binding specificity of bitopic dopamine D2/D3 receptor ligands次级位点相互作用对双拓扑多巴胺D2/D3受体配体结合特异性的影响
err2025-10-20
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errAttila Egyed; Dóra Judit Kiss; Zsófia Pável; Keve Rajna; Supriya A. Gaitonde; Mariam Dubiel; María Isabel Loza; Edina Szűcs; Éva Borbély; Zsófia Hajna; Grzegorz Satala; Márton Vass; Pál Szabó; Katalin Jósvay; Andrzej J. Bojarski; Holger Stark; Zsuzsanna Helyes; Erika Pintér; Michel Bouvier; György M. Keserű
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Versatile Palladium-Catalyzed C-H Arylation of Fluoroarenes with 2-Chloropyridine Derivatives钯催化氟代芳烃与2-氯吡啶衍生物的多样性C-H芳基化反应
err2025-09-27
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errFederico Belnome; Péter P. Fehér; András Stirling; Csongor G. Németh; Tamás Hergert; György M. Keserű; Péter Ábrányi-Balogh
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Discovering Uncharted Binding Pockets on E3 Ligases Leads to the Identification of FBW7 Allosteric Modulators发现E3连接酶上未探索的结合口袋导致FBW7别构调节剂的鉴定
err2025-08-20
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errMíriam Martínez-Cartró; Álvaro Serrano-Morrás; Andrea Bertran-Mostazo; Roger Castaño-Muñiz; Salvatore Scaffidi; Varbina Ivanova; Noémi Csorba; József Simon; Péter Ábrányi-Balogh; Yunfeng Li; György M. Keserü; Bing Hao; Xavier Barril; Carles Galdeano
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Covalent ligand efficiency共价配体效率
err2025-08-13
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errGyörgy G. Ferenczy; György M. Keserű
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The changing landscape of medicinal chemistry optimization药物化学优化的变化格局
err2025-07-07
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PREAI
errAnita Rácz; Levente M. Mihalovits; Maximilian Beckers; Nikolas Fechner; Nikolaus Stiefl; Finton Sirockin; William McCoull; Emma Evertsson; Malin Lemurell; Gergely Makara; György M. Keserű
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