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Identification of constrained peptidomimetics carrying a Michael acceptor warhead as antitrypanosomal agents Previti, Santo; Calcaterra, Elsa; Di Chio, Carla; Natale, Benito; Waqas, Muhammad; Bogacz, Marta; Schirmeister, Tanja; Cavelier, Florine; Calabro, Maria Luisa; Cosconati, Sandro; Ettari, Roberta; Zappala, Maria 分享 收藏
Synthesis of α-fluorocinnamate derivatives as novel cathepsin S inhibitors with in vitro antiproliferative activity against pancreatic cancer cells Citarella, Andrea; Petrella, Serena; Moi, Davide; Dimasi, Alessandro; Braga, Tommaso; Ruberto, Lorenzo; Pieraccini, Stefano; Sironi, Maurizio; Micale, Nicola; Schirmeister, Tanja; Damia, Giovanna; Fasano, Valerio; Silvani, Alessandra; Giannini, Clelia; Passarella, Daniele 分享 收藏
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Inhibitory Effects of Mangifera indica Secondary Metabolites and Their Synthetic Derivatives against SARS-CoV-2 Mpro and NS2B/NS3 (ZIKV and DENV-2) Souza, Gabriella B.; Pontes, Carime L. M.; de Costa, Geovanna O.; de Sousa, Natalia F.; Tizziani, Tiago; Pollo, Luiz Antonio E.; Dambros, Bibiana P.; Scotti, Marcus T.; Steindel, Mario; Braga, Antonio L.; Schirmeister, Tanja; de Assis, Francisco F.; Sandjo, Louis P. 分享 收藏
Bacteria from the Amycolatopsis genus associated with a toxic bird secrete protective secondary metabolites Seibel, Elena; Um, Soohyun; Bodawatta, Kasun H.; Komor, Anna J.; Decker, Tanya; Fricke, Janis; Murphy, Robert; Maiah, Gibson; Iova, Bulisa; Maus, Hannah; Schirmeister, Tanja; Jonsson, Knud Andreas; Poulsen, Michael; Beemelmanns, Christine 分享 收藏
Structure-Based Design and Synthesis of Covalent Inhibitors for Deubiquitinase and Acetyltransferase ChlaDUB1 of Chlamydia trachomatis Zimmermann, Thomas; Feng, Jiachen; de Campos, Luana Janaina; Knight, Lindsey A.; Schloetzer, Jan; Ramirez, Yesid A.; Schwickert, Kevin; Zehe, Markus; Adler, Thomas B.; Schirmeister, Tanja; Kisker, Caroline; Sotriffer, Christoph; Conda-Sheridan, Martin; Decker, Michael 分享 收藏
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Dual Strategy to Design New Agents Targeting Schistosoma mansoni: Advancing Phenotypic and SmCB1 Inhibitors for Improved Efficacy Fuchs, Natalie; Zimmermann, Robert A.; Schwickert, Marvin; Gunkel, Annika; Zimmer, Collin; Meta, Mergim; Schwickert, Kevin; Keiser, Jennifer; Haeberli, Cecile; Kiefer, Werner; Schirmeister, Tanja 分享 收藏
Identification of Dual Inhibitors Targeting Main Protease (Mpro) and Cathepsin L as Potential Anti-SARS-CoV-2 Agents 鉴定靶向主要蛋白酶 (Mpro) 和组织蛋白酶L的双重抑制剂作为潜在的Anti-SARS-CoV-2剂 Previti, Santo; Ettari, Roberta; Calcaterra, Elsa; Roggia, Michele; Natale, Benito; Weldert, Annabelle C.; Mueller-Ruttloff, Christin; Salisch, Florian; Irto, Anna; Cigala, Rosalia Maria; Ziebuhr, John; Schirmeister, Tanja; Cosconati, Sandro; Zappala, Maria 分享 收藏
Peptidyl nitroalkene inhibitors of main protease rationalized by computational and crystallographic investigations as antivirals against SARS-CoV-2 Medrano, Francisco J.; de la Hoz-Rodriguez, Sergio; Marti, Sergio; Arafet, Kemel; Schirmeister, Tanja; Hammerschmidt, Stefan J.; Mueller, Christin; Gonzalez-Martinez, Agueda; Santillana, Elena; Ziebuhr, John; Romero, Antonio; Zimmer, Collin; Weldert, Annabelle; Zimmermann, Robert; Lodola, Alessio; Swiderek, Katarzyna; Moliner, Vicent; Gonzalez, Florenci V. 分享 收藏
Structural features and antiproliferative activity of Pd(ii) complexes with halogenated ligands: a comparative study between Schiff base and reduced Schiff base complexes Forooghi, Kimia; Amiri Rudbari, Hadi; Stagno, Claudio; Iraci, Nunzio; Cuevas-Vicario, Jose V.; Kordestani, Nazanin; Schirmeister, Tanja; Efferth, Thomas; Omer, Ejlal A.; Moini, Nakisa; Aryaeifar, Mahnaz; Blacque, Olivier; Azadbakht, Reza; Micale, Nicola 分享 收藏
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