未登录
分享
收藏Functional and Structural Insights into the Human PPARa/d/? Targeting Preferences of Anti-NASH Investigational Drugs, Lanifibranor, Seladelpar, and Elafibranor
Kamata, Shotaro; Honda, Akihiro; Ishikawa, Ryo; Akahane, Makoto; Fujita, Ayane; Kaneko, Chihiro; Miyawaki, Saeka; Habu, Yuki; Shiiyama, Yui; Uchii, Kie; Machida, Yui; Oyama, Takuji; Ishii, Isao
分享
收藏
分享
收藏
分享
收藏
分享
收藏
分享
收藏Structural design and synthesis of arylalkynyl amide-type peroxisome proliferator-activated receptor γ (PPARγ)-selective antagonists based on the helix12-folding inhibition hypothesis
Ohashi, Masao; Gamo, Kanae; Tanaka, Yuta; Waki, Minoru; Beniyama, Yoko; Matsuno, Kenji; Wada, Jun; Tenta, Masafumi; Eguchi, Jun; Makishima, Makoto; Matsuura, Nobuyasu; Oyama, Takuji; Miyachi, Hiroyuki
分享
收藏
分享
收藏Design and synthesis of a series of α-benzyl phenylpropanoic acid-type peroxisome proliferator-activated receptor (PPAR) gamma partial agonists with improved aqueous solubility一系列水溶性提高的 α-苄基苯基丙酸型过氧化物酶体增殖物激活受体 (PPAR) γ 部分激动剂的设计与合成
Ohashi, Masao; Oyama, Takuji; Putranto, Endy Widya; Waku, Tsuyoshi; Nobusada, Hiromi; Kataoka, Ken; Matsuno, Kenji; Yashiro, Masakazu; Morikawa, Kosuke; Huh, Nam-ho; Miyachi, Hiroyuki
分享
收藏
分享
收藏
分享
收藏
分享
收藏
分享
收藏Design, Synthesis, and Structural Analysis of Phenylpropanoic Acid-Type PPARγ-Selective Agonists Discovery of Reversed Stereochemistry-Activity Relationship
Ohashi, Masao; Oyama, Takuji; Nakagome, Izumi; Satoh, Mayumi; Nishio, Yoshino; Nobusada, Hiromi; Hirono, Shuichi; Morikawa, Kosuke; Hashimoto, Yuichi; Miyachi, Hiroyuki
分享
收藏
分享
收藏
分享
收藏
分享
收藏
分享
收藏
分享
收藏
分享
收藏