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Andrzej J. Bojarski

polish academy of sciences

39H指数
389论文数
7.6K被引数
收录论文 184
发表时间
Synthesis and biological evaluation of C5-(1-substituted-1,2,3-triazol-4-yl)-uridines and their phosphoramidate prodrugsC5-(1-取代-1,2,3-三氮唑-4-基)-尿苷及其磷酰胺酯前药的合成与生物评价
err2026-06-10
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errEvan Saillard; Vincent Roy; Patrick Favetta; Dawid Warszycki; Andrzej J. Bojarski; Leentje Persoons; Dirk Daelemans; Steven De Jonghe; Luigi A. Agrofoglio
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Polyfunctionalized N-Arylsulfonyl Indoles: Identification of (E)-N-Hydroxy-3-{3-[(5-(3-(piperidin-1-yl)propoxy]-1H-indol-1-yl)sulfonyl]phenyl}acrylamide (MTP150) for the Epigenetic-based Therapy of Parkinson’s Disease多官能化N-芳基磺酰基吲哚:用于表观遗传学基础治疗帕金森病的(E)-N-羟基-3-{3-[(5-(3-(哌啶-1-基)丙氧基)-1H-吲哚-1-基)磺酰基]苯基}丙烯酰胺(MTP150)的鉴定
err2026-03-31
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errMireia Toledano-Pinedo; Alicia Porro-Pérez; Linda Schäker-Hübner; Daniel Diez-Iriepa; Isabel Iriepa; Agata Siwek; Małgorzata Wolak; Grzegorz Satała; Andrzej J. Bojarski; Agata Doroz-Płonka; Jadwiga Handzlik; Justyna Godyń; Patrick Dallemagne; Christophe Rochais; Audrey Davis; Marc Since; Belén Pérez; Aina Bellver-Sanchis; Alba Irisarri; Mercè Pallàs; Cristina Solana-Manrique; Francisco López-Muñoz; Lhassane Ismaili; Christian Griñán-Ferré; Nuria Paricio; Finn K. Hansen; Anna Więckowska; José Marco-Contelles
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Chronic 5-HT7R activation drives depressive phenotypes and synaptic dysfunction
err2026-02-03
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PREAI
errBartłomiej Pochwat; Julia Masternak; Bartosz Bobula; Krystian Bijata; Barbara Chruścicka-Smaga; Justyna Turek; Adam Hogendorf; Maria Walczak; Magdalena Smolik; Remigiusz Worch; Magdalena Kusek; Andrzej J. Bojarski; Krzysztof Tokarski; Bernadeta Szewczyk; Monika Bijata
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Fine-tuning 5-HT7 receptor selectivity, inverse agonism, and metabolic stability of new (aryloxy)ethyl-piperidines toward antidepressant and pro-cognitive properties优化新型(芳氧基)乙基哌啶类化合物的5-HT7受体选择性、反向激动作用和代谢稳定性,以增强其抗抑郁和促认知特性。
err2025-11-21
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PREAI
errVittorio Canale; Klaudia Blicharz-Futera; Monika Bijata; Natalie G. Cavalco; Anna Partyka; Matylda Stefaniak; Michał Kamiński; Grzegorz Satała; Dawid Warszycki; Janelle K. Lanham; Joanna Gołębiowska; Maciej Gawlik; Magdalena Smolik; Krystian Bijata; Magdalena Jastrzębska-Więsek; Rafał Kurczab; Andrzej J. Bojarski; Maria Walczak; John D. McCorvy; Jakub Włodarczyk
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The impact of secondary site interactions on the binding specificity of bitopic dopamine D2/D3 receptor ligands次级位点相互作用对双拓扑多巴胺D2/D3受体配体结合特异性的影响
err2025-10-20
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errAttila Egyed; Dóra Judit Kiss; Zsófia Pável; Keve Rajna; Supriya A. Gaitonde; Mariam Dubiel; María Isabel Loza; Edina Szűcs; Éva Borbély; Zsófia Hajna; Grzegorz Satala; Márton Vass; Pál Szabó; Katalin Jósvay; Andrzej J. Bojarski; Holger Stark; Zsuzsanna Helyes; Erika Pintér; Michel Bouvier; György M. Keserű
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Novel Dual 5-HT7 Antagonists and Sodium Channel Inhibitors as Potential Therapeutic Agents with Antidepressant and Anxiolytic Activities新型双5-HT7拮抗剂和钠通道抑制剂作为具有抗抑郁和抗焦虑活性的潜在治疗药物
err2025-10-02
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errAnna Czopek; Paulina Koczurkiewicz-Adamczyk; Katarzyna Wójcik-Pszczoła; Daria Kornas; Wojciech Sitko; Adam Bucki; Michał Sapa; Krzysztof Kamiński; Grzegorz Satała; Beata Duszyńska; Andrzej J. Bojarski; Gniewomir Latacz; Jacek Czopek; Joanna Szpor; Pola Dryja; Kinga Sałat
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Intepirdine Derivatives Possessing Dual 5HT6 Antagonism / HDAC6 Inhibitory ActivityIntepirdine衍生物具有双重5HT6拮抗作用/HDAC6抑制活性
err2025-08-22
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errAndreas Gkanas; Maria Koutiva; Dr. Theodora Katsila; Vivi Bafiti; Prof.Dr. Minos-Timotheos Matsoukas; Vasilios Panagiotopoulos; Dr. Andrzej J. Bojarski; Theodoros Gkouvitsas; Dr. Georgios Moukas; Prof.Dr. Gerasimos Rassias
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Correction: Compound PZ-1262, a 4-isoquinoline-sulfonamide analog of Brexpiprazole, produces potential antidepressant, anxiolytic and procognitive effects in rodent models更正:化合物PZ-1262,一种Brexpiprazole的4-异喹啉磺酰胺类似物,在啮齿动物模型中产生潜在的抗抑郁、抗焦虑和促认知作用。
err2025-05-30
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PREAI
errAnna Partyka; Joanna Gołębiowska; Krzysztof Marciniec; Vittorio Canale; Wojciech Trybała; Grzegorza Satała; Katarzyna Grychowska; Magdalena Jastrzębska-Więsek; Andrzej J. Bojarski; Agnieszka Nikiforuk; Władysława A. Daniel; Anna Wesołowska; Paweł Zajdel; Piotr Popik
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Identification of Orthosteric GABAB Receptor Ligands by Virtual Screening and In Vitro Validation通过虚拟筛选和体外验证鉴定正构GABAB受体配体
err2025-05-16
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errEvenseth, LSM; Russotto, C; Wushur, I; Warszycki, D; Moldes-Anaya, AS; Bojarski, AJ; Gabrielsen, M; Sylte, I
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Compound PZ-1262, a 4-isoquinoline-sulfonamide analog of Brexpiprazole, produces potential antidepressant, anxiolytic and procognitive effects in rodent models
err2025-03-01
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PREAI
errPartyka, Anna; Golebiowska, Joanna; Marciniec, Krzysztof; Canale, Vittorio; Trybala, Wojciech; Satala, Grzegorza; Grychowska, Katarzyna; Jastrzebska-Wiesek, Magdalena; Bojarski, Andrzej J.; Nikiforuk, Agnieszka; Daniel, Wladyslawa A.; Wesolowska, Anna; Zajdel, Pawel; Popik, Piotr
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Simultaneous 5-HT1BR agonist/5-HT6R antagonist action as a potential treatment of Parkinson's disease and its comorbidities
err2025-02-01
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PREAI
errZajdel, Pawe l; Matloka, Mikolaj; Konieczny, Jolanta; Kos, Tomasz; Lammers, Josie C.; Cavalco, Natalie G.; Clark, Allison A.; Lenda, Tomasz; Satala, Grzegorz; Canale, Vittorio; Grychowska, Katarzyna; Krawczyk, Martyna; Nikiforuk, Agnieszka; Partyka, Anna; Jastrzebska-Wiesek, Magdalena; Berghauzen-Maciejewska, Klemencja; Biala, Dominika; Janicka, Monika; Janusz, Artur; Piast, Radoslaw; Mulewski, Krzysztof; Smuga, Damian; Pieczykolan, Jerzy; Wieczorek, Maciej; Moszczynski-Petkowski, Rafal; Dubiel, Krzysztof; Ossowska, Krystyna; Bojarski, Andrzej J.; Kaminski, Krzysztof; Mccorvy, John D.; Popik, Piotr
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Contilisant plus Tubastatin A Hybrids: Polyfunctionalized Indole Derivatives as New HDAC Inhibitor-Based Multitarget Small Molecules with In Vitro and In Vivo Activity in Neurodegenerative Diseases
err2024-09-10
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PREAI
errToledano-Pinedo, Mireia; Porro-Perez, Alicia; Schaeker-Huebner, Linda; Romero, Fernando; Dong, Min; Samadi, Abdelouahid; Almendros, Pedro; Iriepa, Isabel; Bautista-Aguilera, Oscar M.; Rodriguez-Fernandez, M. Mercedes; Solana-Manrique, Cristina; Sanchis, Inmaculada; Mora-Morell, Alba; Rodriguez, Ania Canseco; Sanchez-Perez, Ana M.; Knez, Damijan; Gobec, Stanislav; Bellver-Sanchis, Aina; Perez, Belen; Dobrydnev, Alexey V.; Artetxe-Zurutuza, Aizpea; Matheu, Ander; Siwek, Agata; Wolak, Malgorzata; Satala, Grzegorz; Bojarski, Andrzej J.; Doroz-Plonka, Agata; Handzlik, Jadwiga; Godyn, Justyna; Wieckowska, Anna; Paricio, Nuria; Grinan-Ferre, Christian; Hansen, Finn K.; Marco-Contelles, Jose
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5-HT6 receptor neutral antagonists protect astrocytes: A lesson from 2-phenylpyrrole derivatives
err2024-09-01
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errDrop, Marcin; Koczurkiewicz-Adamczyk, Paulina; Bento, Ophelie; Pietrus, Wojciech; Satala, Grzegorz; Blicharz-Futera, Klaudia; Canale, Vittorio; Grychowska, Katarzyna; Bantreil, Xavier; Pekala, Elzbieta; Kurczab, Rafal; Bojarski, Andrzej J.; Chaumont-Dubel, Severine; Marin, Philippe; Lamaty, Frederic; Zajdel, Pawe l
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Unraveling psilocybin's therapeutic potential: behavioral and neuroplasticity insights in Wistar-Kyoto and Wistar male rat models of treatment-resistant depression (Jul, 10.1007/s00213-024-06644-3, 2024)
err2024-07-20
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errKolasa, Magdalena; Nikiforuk, Agnieszka; Korlatowicz, Agata; Solich, Joanna; Potasiewicz, Agnieszka; Dziedzicka-Wasylewska, Marta; Bugno, Ryszard; Hogendorf, Adam; Bojarski, Andrzej; Faron-Gorecka, Agata
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Unraveling psilocybin's therapeutic potential: behavioral and neuroplasticity insights in Wistar-Kyoto and Wistar male rat models of treatment-resistant depression
err2024-07-04
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errMagdalena, Kolasa; Agnieszka, Nikiforuk; Agata, Korlatowicz; Joanna, Solich; Agnieszka, Potasiewicz; Dziedzicka-Wasylewska, Marta; Ryszard, Bugno; Adam, Hogendorf; Andrzej, Bojarski; Agata, Faron-Gorecka
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Physicochemical, structural and biological characterisation of poly (3-hydroxyoctanoate) supplemented with diclofenac acid conjugates - Harnessing the potential in the construction of materials for skin regeneration processes
err2024-05-01
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errHarazna, Katarzyna; Fricker, Annabelle T.; Konefal, Rafal; Medaj, Aneta; Zimowska, Malgorzata; Leszczynski, Bartosz; Wrobel, Andrzej; Bojarski, Andrzej J.; Roy, Ipsita; Guzik, Maciej
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Structure-Activity Relationships and Therapeutic Potential of Purinergic P2X7 Receptor Antagonists
err2024-04-01
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PREAI
errEl Idrissi, Imane Ghafir; Podlewska, Sabina; Abate, Carmen; Bojarski, Andrzej J.; Lacivita, Enza; Leopoldo, Marcello
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Repeated low doses of psilocybin increase resilience to stress, lower compulsive actions, and strengthen cortical connections to the paraventricular thalamic nucleus in rats
err2023-10-02
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errKiilerich, Kat F.; Lorenz, Joe; Scharff, Malthe B.; Speth, Nikolaj; Brandt, Tobias G.; Czurylo, Julia; Xiong, Mengfei; Jessen, Naja S.; Casado-Sainz, Agata; Shalgunov, Vladimir; Kjaerby, Celia; Satala, Grzegorz; Bojarski, Andrzej J.; Jensen, Anders A.; Herth, Matthias M.; Cumming, Paul; Overgaard, Agnete; Palner, Mikael
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Novel object recognition test as an alternative approach to assessing the pharmacological profile of sigma-1 receptor ligands
err2023-08-12
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errSzczepanska, Katarzyna; Bojarski, Andrzej J. J.; Popik, Piotr; Malikowska-Racia, Natalia
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