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Unique Interactions of Novel Rufomycin Click Chemistry Analogs with Mtb ClpC1 and Implications Ratia, Kiira; Jin, Shengnan; Abad-Zapatero, Celerino; Shetye, Gauri S.; Demissie, Robel; Qader, Mallique; Beautrait, Alexandre; Nikolic, Dejan S.; Wolf, Nina M.; Rubin, Eric J.; Krandor, Olga; Serbina, Natalya; Li, Guiying; Pauli, Guido F.; Klein, Larry L.; Cho, Sanghyun; Franzblau, Scott G.; Fotouhi, Nader; Kaneko, Takushi; Lee, Hyun 分享 收藏
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Characterization of Cyclic Peptides for Antituberculosis Drug Development Targeting ClpC1 用于靶向ClpC1的抗结核药物开发的环肽的表征 Demissie, Robel; Vaid, Tasneem M.; Kwon, Youngjin; Shetye, Gauri; Tran, Thao; Nomani, Fatema; Jin, Shengnan; Suh, Joo-Won; Lee, Hanki; Shin, Yern-Hyerk; Cui, Jinsheng; Oh, Dong-Chan; Franzblau, Scott G.; Cho, Sanghyun; Lee, Hyun 分享 收藏
Discovery of ultra short (3-peptoids with selective activity against drug-resistant Mycobacterium tuberculosis 发现具有选择性活性的超短(3-肽类)对耐药性结核分枝杆菌的作用 Kauffman, John; Cuevas, Jake; Feiner, Janaya; Metzger, Margaret; Shetye, Gauri; Wan, Baojie; Qader, Mallique; Nguyen, Duc; Nugent, Angela; Hossain, Akil; Franzblau, Scott; Umesiri, Francis E. 分享 收藏
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Nifuroxazide and 4-Hydroxybenzhydrazone Derivatives as New Antiparasitic (Trypanosoma cruzi and Leishmania mexicana) and Anti-Mycobacterium tuberculosis Agents 呋喃唑酮及其4-羟基苯肼盐衍生物作为新的抗寄生虫(克氏锥虫和墨西哥利什曼原虫)和抗分枝杆菌结核分枝杆菌剂 Delgado-Maldonado, Timoteo; Navarrete-Carriola, Diana V.; Vazquez-Jimenez, Lenci K.; Paz-Gonzalez, Alma D.; Wan, Baojie; Franzblau, Scott; Mohammed, Othman Mueen; Rodriguez-Paez, Lorena; Aguirre-Alvarado, Charmina; Alcantara-Farfan, Veronica; Cordero-Martinez, Joaquin; Bandyopadhyay, Debasish; Moreno-Rodriguez, Adriana; Rivera, Gildardo 分享 收藏
Structure-Based Analysis of Semisynthetic Anti-TB Rufomycin Analogues Zhou, Bin; Shetye, Gauri; Klein, Larry L.; Wolf, Nina M.; Lee, Hyun; Mcalpine, James B.; Harris, Guy; Chen, Shao-Nong; Suh, Joo Won; Cho, Sang-Hyun; Franzblau, Scott G.; Abad-Zapatero, Celerino; Pauli, Guido F. 分享 收藏
Expanding the Landscape of Dual Action Antifolate Antibacterials through 2,4-Diamino-1,6-dihydro-1,3,5-triazines Georgiades, John D.; Berkovich, Daniel A.; Mckee, Samuel R.; Smith, Angela R.; Sankaran, Banumathi; Flentie, Kelly N.; Castaneda, Carlos H.; Grohmann, Daniel G.; Rohatgi, Ram; Lasky, Carrie; Mason, Twila A.; Champine, James E.; Miller, Patricia A.; Moellmann, Ute; Moraski, Garrett C.; Franzblau, Scott G.; Miller, Marvin J.; Stallings, Christina L.; Jez, Joseph M.; Hathaway, Bruce A.; Wencewicz, Timothy A. 分享 收藏
Discovery of New Cyclic Lipodepsipeptide Orfamide N via Partnership with Middle School Students from the Boys and Girls Club Tan, Jin Yi; Augustinovic, Mario; Omar, Ashraf M.; Lourenzon, Vitor B.; Krull, Nyssa; Lopez, Xochitl; Khin, Manead; Shetye, Gauri; Nguyen, Duc; Qader, Mallique; Nugent, Angela C.; Mpofu, Enock; Williams, Camarria; Rodriguez, Jonathon; Burdette, Joanna E.; Cho, Sanghyun; Franzblau, Scott G.; Eustaquio, Alessandra S.; Zhang, Qibin; Murphy, Brian T. 分享 收藏
Design, synthesis and biological evaluation of novel pyrido-[2,3-d]-pyrimidin-2-amine analogues as antimycobacterial agents Kumar, Boddupalli Venkata Siva; Khetmalis, Yogesh Mahadu; Chaitanya, Kosana Sai; Chandu, Ala; Shetye, Gauri; Ma, Rui; Murugesan, Sankaranarayanan; Franzblau, Scott G.; Sekhar, Kondapalli Venkata Gowri Chandra 分享 收藏
Cavomycins A-C, Linear Oligomer Depsipeptides from an Annelid-Associated Streptomyces cavourensis Cavomycins a-c,来自与链状链霉菌相关的链霉菌的线性低聚物缩肽 Wang, Weihong; Lee, Juni; Roh, Eun; Shetye, Gauri; Cao, Jin; Mcalpine, James; Pauli, Guido; Franzblau, Scott; Vu, Thi Hanh Nguyen; Quach, Ngoc Tung; Oh, Eunseok; Park, Kyu-Hyung; Park, Chanyoon; Cho, Youbin; Jang, Hyeseon; Han, Songjoo; Kim, Hiyoung; Cho, Sanghyun; Phi, Quyet-Tien; Kang, Heonjoong 分享 收藏
Expanding the chemical space of ester of quinoxaline-7-carboxylate 1,4-di-N-oxide derivatives as potential antitubercular agents 扩大quinoxaline-7-carboxylate 1,4-二-n-氧化物衍生物的酯作为潜在抗结核药的化学空间 Gonzalez-Gonzalez, Alonzo; Sanchez-Sanchez, Oscar; Wan, Baojie; Franzblau, Scott; Palos, Isidro; Espinoza-Hicks, Jose C.; Moreno-Rodriguez, Adriana; Martinez-Vazquez, Ana Veronica; Lara-Ramirez, Edgar E.; Ortiz-Perez, Eyra; Paz-Gonzalez, Alma D.; Rivera, Gildardo 分享 收藏
Discovery of a New Antibiotic Demethoxytetronasin Using a Dual-Sided Agar Plate Assay (DAPA) Lee, Jung-Ho; Ma, Rui; Nguyen, Linh; Kahn, Shahebraj; Qader, Mallique; Mpofu, Enock; Shetye, Gauri; Krull, Nyssa K.; Augustinovic, Mario; Omarsdottir, Sesselja; Cho, Sanghyun; Franzblau, Scott G.; Murphy, Brian T. 分享 收藏
Isolation and Characterization of Anti-Mycobacterial Natural Products from a Petrosia sp. Marine Sponge Chhetri, Bhuwan Khatri; Bhanushali, Riya; Liang, Yifan; Cepeda, Marisa R. .; Niradininoco, Adi Kula; Soapi, Katy; Wan, Baojie; Qader, Mallique; Franzblau, Scot t G.; Kubanek, Julia 分享 收藏
Design, synthesis and biological evaluation of phenanthridine amide and 1,2,3-triazole analogues against Mycobacterium tuberculosis Nandikolla, Adinarayana; Khetmalis, Yogesh Mahadu; Kumar, Boddupalli Venkata Siva; Chandu, Ala; Kumar, Banoth Karan; Shetye, Gauri; Ma, Rui; Murugesan, Sankaranarayanan; Franzblau, Scott G.; Sekhar, Kondapalli Venkata Gowri Chandra 分享 收藏
Anti-Microbial Activity of Aliphatic Alcohols from Chinese Black Cardamom (Amomum tsao-ko) against Mycobacterium tuberculosis H37Rv Lee, So Young; Shetye, Gauri S.; Son, So-Ri; Lee, Hyun; Klein, Larry L.; Yoshihara, Jeffrey K.; Ma, Rui; Franzblau, Scott G.; Cho, Sanghyun; Jang, Dae Sik 分享 收藏
New Rufomycins from Streptomyces atratus MJM3502 Expand Anti- Mycobacterium tuberculosis Structure-Activity Relationships Zhou, Bin; Shetye, Gauri; Wolf, Nina M.; Chen, Shao-Nong; Qader, Mallique; Ray, G. Joseph; Lankin, David C.; Cho, Sanghyun; Cheng, Jinhua; Suh, Joo-Won; Franzblau, Scott G.; McAlpine, James B.; Pauli, Guido F. 分享 收藏
Nitroimidazopyrazinones with Oral Activity against Tuberculosis and Chagas Disease in Mouse Models of Infection 在小鼠感染模型中具有口服抗结核和查加斯病活性的硝基咪唑并吡嗪酮 Ang, Chee Wei; Lee, Brendon M.; Jackson, Colin J.; Wang, Yuehong; Franzblau, Scott G.; Francisco, Amanda F.; Kelly, John M.; Bernhardt, Paul, V; Tan, Lendl; West, Nicholas P.; Sykes, Melissa L.; Hinton, Alexandra O.; Bolisetti, Raghu; Avery, Vicky M.; Cooper, Matthew A.; Blaskovich, Mark A. T. 分享 收藏