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Michelle R. Arkin

University of California

57H指数
311论文数
1.5W被引数
收录论文 96
发表时间
A Molecular Mechanistic Deep Dive into 14–3–3 Molecular Glue Cooperativity14–3–3分子胶合协同作用的分子机制深度解析
err2026-09-01
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PREAI
errMarloes A. M. Pennings; Edmee M. F. Vandenboorn-Bönner; Lisa Nooren; Markella Konstantinidou; Chad Altobelli; Christian Ottmann; Albert J. Markvoort; Galen P. Miley; Michelle R. Arkin; Luc Brunsveld
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FOXM1 inhibition primes terminal differentiation of human iPSC-derived hepatocytesFOXM1抑制促进人iPSC来源肝细胞的终末分化
err2026-07-08
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errOAAI
errKayque Alves Telles-Silva; Lara Pacheco; Sabrina Komatsu; Fernanda Chianca; Gustavo Chagas; Gabrielly Cristine Martins; Maria Gridina; Daria Panchenko; Valdemir Melechco Carvalho; Elia G. Caldini; Veniamin S. Fishman; Michelle Arkin; Ernesto Goulart; Mayana Zatz
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Modulation of the 14-3-3σ/C-RAF “Auto”inhibited Complex by Molecular Glues分子胶对14-3-3σ/c-raf “自动” 抑制复合物的调制
err2026-01-30
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errOAAI
errMarkella Konstantinidou; Holly R. Vickery; Marloes A. M. Pennings; Johanna M. Virta; Shu Yue Luo; Emira J. Visser; Sean D. Bannier; Mrudula Srikanth; Sabine Z. Cismoski; Lucy C. Young; Maxime C. M. van den Oetelaar; Frank McCormick; Christian Ottmann; Luc Brunsveld; Michelle R. Arkin
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Fragment-to-Lead Medicinal Chemistry Publications in 2024: A Tenth Annual Perspective (vol 68, pg 24830, 2025)2024年片段到先导药物化学出版物:第十年度展望(卷 68,第 24830 页,2025年)
err2026-01-01
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PREAI
errTwigg, David G.; Arai, Kenta; Arkin, Michelle R.; Erlanson, Daniel A.; de Esch, Iwan J. P.; Farkas, Barbara; Fesik, Stephen W.; Jahnke, Wolfgang; Johnson, Christopher N.; Schroeder, Martin
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Fragment-to-Lead Medicinal Chemistry Publications in 2024: A Tenth Annual Perspective2024年片段到先导化合物的药物化学出版物:第十年度展望
err2025-11-25
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PREAI
errDavid G. Twigg; Kenta Arai; Michelle R. Arkin; Daniel A. Erlanson; Iwan J. P. de Esch; Barbara Farkaš; Stephen W. Fesik; Wolfgang Jahnke; Christopher N. Johnson; Martin Schroeder
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Scaffold-hopping for molecular glues targeting the 14-3-3/ERα complex针对14-3-3/ERα复合物的骨架跳跃分子胶开发
err2025-07-14
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errOAAI
errMarkella Konstantinidou; Marios Zingiridis; Marloes A. M. Pennings; Michael Fragkiadakis; Johanna M. Virta; Jezrael L. Revalde; Emira J. Visser; Christian Ottmann; Luc Brunsveld; Constantinos G. Neochoritis; Michelle R. Arkin
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Blocking C-terminal processing of KRAS4b via a direct covalent attack on the CaaX-box cysteine通过直接共价攻击CaaX盒半胱氨酸来阻断KRAS4b的C末端加工
err2025-05-09
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errOAAI
errMaciag, Anna E.; Yang, Yue; Sharma, Alok K.; Turner, David M.; Dehart, Caroline J.; Abdelkarim, Hazem; Fan, Lixin; Smith, Brian P.; Kumari, Vandana; Dyba, Marcin; Rigby, Megan; Badillo, Jean A. Castillo; Adams, Lauren; Fornelli, Luca; Fox, Stephen; Brafman, Alla; Turbyville, Thomas; Gillette, William; Messing, Simon; Agamasu, Constance; Wolfe, Andrew L.; Gysin, Stephan; Chan, Albert H.; Simanshu, Dhirendra K.; Esposito, Dominic; Chertov, Oleg; Stephen, Andrew G.; Arkin, Michelle; Renslo, Adam; Kelleher, Neil L.; Gaponenko, Vadim; Lightstone, Felice C.; Nissley, Dwight, V; McCormick, Frank
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Structure-based discovery of highly bioavailable, covalent, broad-spectrum coronavirus MPro inhibitors with potent in vivo efficacy基于结构的具有高生物利用度、共价键、广谱冠状病毒MPro抑制剂的发现,并具有强体内效力
err2025-04-25
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errOAAI
errDetomasi, Tyler C.; Degotte, Gilles; Huang, Sijie; Suryawanshi, Rahul K.; Diallo, Amy; Lizzadro, Luca; Zaptero-Belinchon, Francisco J.; Taha, Taha Y.; Li, Jiapeng; Richards, Alicia L.; Hantz, Eric R.; Alam, Zain; Montano, Mauricio; McCavitt-Malvido, Maria; Gumpena, Rajesh; Partridge, James R.; Correy, Galen J.; Matsui, Yusuke; Charvat, Annemarie F.; Glenn, Isabella S.; Rosecrans, Julia; Revalde, Jezrael L.; Anderson, Dashiell; Hultquist, Judd F.; Arkin, Michelle R.; Neitz, R. Jeffrey; Swaney, Danielle L.; Krogan, Nevan J.; Shoichet, Brian K.; Verba, Kliment A.; Ott, Melanie; Renslo, Adam R.; Craik, Charles S.
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2024 VCP International Conference: Exploring multi-disciplinary approaches from basic science of valosin containing protein, an AAA plus ATPase protein, to the therapeutic advancement for VCP-associated multisystem proteinopathy
err2025-03-01
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errPeck, A.; Dadi, A.; Yavarow, Z.; Alfano, L. N.; Anderson, D.; Arkin, M. R.; Chou, T. F.; D'Ambrosio, E. S.; Diaz-Manera, J.; Dudley, J. P.; Elder, A. G.; Ghoshal, N.; Hart, C. E.; Hart, M. M.; Huryn, D. M.; Johnson, A. E.; Jones, K. B.; Kimonis, V.; Kiskinis, E.; Lee, E. B.; Lloyd, T. E.; Mapstone, M.; Martin, A.; Meyer, H.; Mozaffar, T.; Onyike, C. U.; Pfeffer, G.; Pindon, A.; Raman, M.; Richard, I.; Rubinsztein, D. C.; Schiava, M.; Schuetz, A. K.; Shen, P. S.; Southworth, D. R.; Staffaroni, A. M.; Taralio-Gravovac, M.; Weihl, C. C.; Yao, Q.; Ye, Y.; Peck, N.
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Deep phenotypic profiling of neuroactive drugs in larval zebrafish
err2024-11-17
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errOAAI
errGendelev, Leo; Taylor, Jack; Myers-Turnbull, Douglas; Chen, Steven; McCarroll, Matthew N.; Arkin, Michelle R.; Kokel, David; Keiser, Michael J.
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Haploinsufficiency underlies the neurodevelopmental consequences of SLC6A1 variants
err2024-06-01
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errOAAI
errSilva, Dina Buitrago; Trinidad, Marena; Ljungdahl, Alicia; Revalde, Jezrael L.; Berguig, Geoffrey Y.; Wallace, William; Patrick, Cory S.; Bomba, Lorenzo; Arkin, Michelle; Dong, Shan; Estrada, Karol; Hutchinson, Keino; Lebowitz, Jonathan H.; Schlessinger, Avner; Johannesen, Katrine M.; Moller, Rikke S.; Giacomini, Kathleen M.; Froelich, Steven; Sanders, Stephan J.; Wuster, Arthur
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A Top-Down Proteomic Assay to Evaluate KRAS4B-Compound Engagement
err2024-03-18
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errD'Ippolito, Robert A.; Rabara, Dana; Blanco, Maria Abreu; Alberico, Emily; Drew, Matthew R.; Ramakrishnan, Nitya; Sontan, Dara; Widmeyer, Stephanie R. T.; Scheidemantle, Grace M.; Messing, Simon; Turner, David; Arkin, Michelle; Maciag, Anna E.; Stephen, Andrew G.; Esposito, Dominic; Mccormick, Frank; Nissley, Dwight V.; Dehart, Caroline J.
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An in vivo screening platform identifies senolytic compounds that target p16 INK4a+fibroblasts in lung fibrosis
err2024-03-07
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errOAAI
errLee, Jin Young; Reyes, Nabora S.; Ravishankar, Supriya; Zhou, Minqi; Krasilnikov, Maria; Ringler, Christian; Pohan, Grace; Wilson, Chris; Ang, Kenny Kean-Hooi; Wolters, Paul J.; Tsukui, Tatsuya; Sheppard, Dean; Arkin, Michelle R.; Peng, Tien
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Synthetic autophagy receptor合成自噬受体
errAUTOPHAGY
IF14.3
err2024-02-14
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errOAAI
errJiang, Ziwen; Kuo, Yu-Hsuan; Arkin, Michelle R.
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Identifying ligands for the PHD1 finger of KDM5A through high-throughput screening
err2024-01-01
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errOAAI
errOrtiz, Gloria; Longbotham, James E.; Qin, Sophia L.; Zhang, Meng Yao; Lee, Gregory M.; Neitz, R. Jeffrey; Kelly, Mark J. S.; Arkin, Michelle R.; Fujimori, Danica Galonic
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The p97/VCP adaptor UBXD1 drives AAA plus remodeling and ring opening through multi-domain tethered interactions
err2023-11-09
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errOAAI
errBraxton, Julian R.; Altobelli, Chad R.; Tucker, Maxwell R.; Tse, Eric; Thwin, Aye C.; Arkin, Michelle R.; Southworth, Daniel R.
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Structure-Based Optimization of Covalent, Small-Molecule Stabilizers of the 14-3-3s/ERa Protein-Protein Interaction from Nonselective Fragments
err2023-09-07
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errOAAI
errKonstantinidou, Markella; Visser, Emira J.; Vandenboorn, Edmee; Chen, Sheng; Jaishankar, Priyadarshini; Overmans, Maurits; Dutta, Shubhankar; Neitz, R. Jeffrey; Renslo, Adam R.; Ottmann, Christian; Brunsveld, Luc; Arkin, Michelle R.
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