Hopkinson, Richard J.; Tumber, Anthony; Yapp, Clarence; Chowdhury, Rasheduzzaman; Aik, WeiShen; Che, Ka Hing; Li, Xuan Shirley; Kristensen, Jan B. L.; King, Oliver N. F.; Chan, Mun Chiang; Yeoh, Kar Kheng; Choi, Hwanho; Walport, Louise J.; Thinnes, Cyrille C.; Bush, Jacob T.; Lejeune, Clarisse; Rydzik, Anna M.; Rose, Nathan R.; Bagg, Eleanor A.; McDonough, Michael A.; Krojer, Tobias J.; Yue, Wyatt W.; Ng, Stanley S.; Olsen, Lars; Brennan, Paul E.; Oppermann, Udo; Mueller, Susanne; Klose, Robert J.; Ratcliffe, Peter J.; Schofield, Christopher J.; Kawamura, Akane

Plant Growth Regulator Daminozide Is a Selective Inhibitor of Human KDM2/7 Histone Demethylases

JOURNAL OF MEDICINAL CHEMISTRY

IF6.8

2012-07-11130

Rose, Nathan R.; Woon, Esther C. Y.; Tumber, Anthony; Walport, Louise J.; Chowdhury, Rasheduzzaman; Li, Xuan Shirley; King, Oliver N. F.; Lejeune, Clarisse; Ng, Stanley S.; Krojer, Tobias; Chan, Mun Chiang; Rydzik, Anna M.; Hopkinson, Richard J.; Che, Ka Hing; Daniel, Michelle; Strain-Damerell, Claire; Gileadi, Carina; Kochan, Grazyna; Leung, Ivanhoe K. H.; Dunford, James; Yeoh, Kar Kheng; Ratcliffe, Peter J.; Burgess-Brown, Nicola; von Delft, Frank; Muller, Susanne; Marsden, Brian; Brennan, Paul E.; McDonough, Michael A.; Oppermann, Udo; Klose, Robert J.; Schofield, Christopher J.; Kawamura, Akane

Dynamic Combinatorial Chemistry Employing Boronic Acids/Boronate Esters Leads to Potent Oxygenase Inhibitors

ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

IF16.9

2012-05-2582

PREAI

Dynamic Combinatorial Mass Spectrometry Leads to Inhibitors of a 2-Oxoglutarate-Dependent Nucleic Acid Demethylase

JOURNAL OF MEDICINAL CHEMISTRY

IF6.8

2012-02-2249

PREAI

Linking of 2-Oxoglutarate and Substrate Binding Sites Enables Potent and Highly Selective Inhibition of JmjC Histone Demethylases

ANGEWANDTE CHEMIE-INTERNATIONAL EDITION