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收藏Synthesis and Pharmacological Characterization of Nociceptin/Orphanin FQ Dimeric Ligands
Albanese, Valentina; Pola, Pietro; Argentieri, Michela; De Ventura, Tiziano; Frezza, Alessia; Illuminati, Davide; Malfacini, Davide; Marzola, Erika; Meneguzzo, Giulio; Morrone, Erika; Preti, Delia; Rizzo, Alessandra; Sturaro, Chiara; Calo, Girolamo; Guerrini, Remo; Pacifico, Salvatore; Ruzza, Chiara
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收藏Spiropiperidine-Based Oligomycin-Analog Ligands To Counteract the Ischemia-Reperfusion Injury in a Renal Cell Model
Turrin, Giulia; Lo Cascio, Ettore; Giacon, Noah; Fantinati, Anna; Cristofori, Virginia; Illuminati, Davide; Preti, Delia; Morciano, Giampaolo; Pinton, Paolo; Agyapong, Esther Densu; Trapella, Claudio; Arcovito, Alessandro
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收藏Novel Aryl Sulfonamide Derivatives as NLRP3 Inflammasome Inhibitors for the Potential Treatment of Cancer
Albanese, Valentina; Missiroli, Sonia; Perrone, Mariasole; Fabbri, Martina; Boncompagni, Caterina; Pacifico, Salvatore; De Ventura, Tiziano; Ciancetta, Antonella; Dondio, Giulio; Kricek, Franz; Pinton, Paolo; Guerrini, Remo; Preti, Delia; Giorgi, Carlotta
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收藏Non-neuronal TRPA1 encodes mechanical allodynia associated with neurogenic inflammation and partial nerve injury in rats
De Logu, Francesco; De Siena, Gaetano; Landini, Lorenzo; Marini, Matilde; de Araujo, Daniel Souza Monteiro; Albanese, Valentina; Preti, Delia; Romitelli, Antonia; Chieca, Martina; Titiz, Mustafa; Iannone, Luigi F.; Geppetti, Pierangelo; Nassini, Romina
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收藏Novel Mixed NOP/Opioid Receptor Peptide Agonists
Pacifico, Salvatore; Albanese, Valentina; Illuminati, Davide; Marzola, Erika; Fabbri, Martina; Ferrari, Federica; Holanda, Victor A. D.; Sturaro, Chiara; Malfacini, Davide; Ruzza, Chiara; Trapella, Claudio; Preti, Delia; Lo Cascio, Ettore; Arcovito, Alessandro; Della Longa, Stefano; Marangoni, Martina; Fattori, Davide; Nassini, Romina; Calo, Girolamo; Guerrini, Remo
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收藏Structure-Activity Relationship Studies on Oxazolo[3,4-a]pyrazine Derivatives Leading to the Discovery of a Novel Neuropeptide S Receptor Antagonist with Potent In Vivo Activity
Albanese, Valentina; Ruzza, Chiara; Marzola, Erika; Bernardi, Tatiana; Fabbri, Martina; Fantinati, Anna; Trapella, Claudio; Reinscheid, Rainer K.; Ferrari, Federica; Sturaro, Chiara; Calo, Girolamo; Amendola, Giorgio; Cosconati, Sandro; Pacifico, Salvatore; Guerrini, Remo; Preti, Delia
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收藏Role of TRPA1 receptors in skin inflammation induced by volatile chemical irritants in mice
Noroes, Maira Macedo; Santos, Larissa Gonzaga; Gavioli, Elaine Cristina; Soares Rachetti, Vanessa de Paula; Otuki, Michel Fleith; Cabrini, Daniela de Almeida; Prudente, Arthur da Silveira; Jentsch Matias Oliveira, Janiana Raiza; Goncalves, Muryel de Carvalho; Ferreira, Juliano; Preti, Delia; De Logu, Francesco; Nassini, Romina; Andre, Eunice
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收藏Tetrabranched Hetero-Conjugated Peptides as Bifunctional Agonists of the NOP and Mu Opioid Receptors
Pacifico, Salvatore; Albanese, Valentina; Illuminati, Davide; Fantinati, Anna; Marzola, Erika; Ferrari, Federica; Neto, Joaquim Azevedo; Sturaro, Chiara; Ruzza, Chiara; Cato, Girolamo; Preti, Delia; Guerrini, Remo
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收藏Synthesis and Biological Activity of Peptide α-Ketoamide Derivatives as Proteasome Inhibitors肽 α-酮酰胺类蛋白酶体抑制剂的合成及生物活性研究
Pacifico, Salvatore; Ferretti, Valeria; Albanese, Valentina; Fantinati, Anna; Gallerani, Eleonora; Nicoli, Francesco; Gavioli, Riccardo; Zamberlan, Francesco; Preti, Delia; Marastoni, Mauro
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收藏The acyl-glucuronide metabolite of ibuprofen has analgesic and anti-inflammatory effects via the TRPA1 channel
De Logu, Francesco; Puma, Simone Li; Landini, Lorenzo; Tuccinardi, Tiziano; Poli, Giulio; Preti, Delia; De Siena, Gaetano; Patacchini, Riccardo; Tsagareli, Merab G.; Geppetti, Pierangelo; Nassini, Romina
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收藏Design, synthesis, in vitro antiproliferative activity and apoptosis-inducing studies of 1-(3′,4′,5′-trimethoxyphenyl)-3-(2′-alkoxycarbonylindolyl)-2-propen-1-one derivatives obtained by a molecular hybridisation approach
Preti, Delia; Romagnoli, Romeo; Rondanin, Riccardo; Cacciari, Barbara; Hamel, Ernest; Balzarini, Jan; Liekens, Sandra; Schols, Dominique; Estevez-Sarmiento, Francisco; Quintana, Jose; Estevez, Francisco
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收藏Discovery of Novel 1,3,8-Triazaspiro[4.5]decane Derivatives That Target the c Subunit of F1/FO-Adenosine Triphosphate (ATP) Synthase for the Treatment of Reperfusion Damage in Myocardial Infarction发现靶向F1/FO-三磷酸腺苷 (ATP) 合酶c亚基的新型1,3,8-三唑螺 [4.5] 癸烷衍生物,用于治疗心肌梗塞的再灌注损伤
Morciano, Giampaolo; Preti, Delia; Pedriali, Gaia; Aquila, Giorgio; Missiroli, Sonia; Fantinati, Anna; Caroccia, Natascia; Pacifico, Salvatore; Bonora, Massimo; Talarico, Anna; Morganti, Claudia; Rizzo, Paola; Ferrari, Roberto; Wieckowski, Mariusz R.; Campo, Gianluca; Giorgi, Carlotta; Trapella, Claudio; Pinton, Paolo
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收藏Naphthoquinone amino acid derivatives, synthesis and biological activity as proteasome inhibitors
Marastoni, Mauro; Trapella, Claudio; Scotti, Alessandra; Fantinati, Anna; Ferretti, Valeria; Marzola, Erika; Eleonora, Gallerani; Gavioli, Riccardo; Preti, Delia
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