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收藏Centriolar cap proteins CP110 and CPAP control slow elongation of microtubule plus ends中心粒帽蛋白CP110和CPAP调控微管正极的缓慢延长
Iyer, Saishree S.; Chen, Fangrui; Ogunmolu, Funso E.; Moradi, Shoeib; Volkov, Vladimir A.; van Grinsven, Emma J.; van Hoorn, Chris; Wu, Jingchao; Andrea, Nemo; Hua, Shasha; Jiang, Kai; Vakonakis, Ioannis; Potocnjak, Mia; Herzog, Franz; Gigant, Benoit; Gudimchuk, Nikita; Stecker, Kelly E.; Dogterom, Marileen; Steinmetz, Michel O.; Akhmanova, Anna
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收藏Engineering of brick and staple components for ordered assembly of synthetic repeat proteins
Miller, Jessalyn; Urvoas, Agathe; Gigant, Benoit; Ouldali, Malika; Arteni, Ana; Mesneau, Agnes; Valerio-Lepiniec, Marie; Artzner, Franck; Dujardin, Erik; Minard, Philippe
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收藏B-nor-methylene Colchicinoid PT-100 Selectively Induces Apoptosis in Multidrug-Resistant Human Cancer Cells via an Intrinsic Pathway in a Caspase-Independent Manner
Stein, Andreas; Thomopoulou, Persefoni Hilken Nee; Frias, Corazon; Hopff, Sina M.; Varela, Paloma; Wilke, Nicola; Mariappan, Arul; Neudoerfl, Jorg-Martin; Fedorov, Alexey Yu; Gopalakrishnan, Jay; Gigant, Benoit; Prokop, Aram; Schmalz, Hans-Gunther
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收藏GTP-dependent formation of straight tubulin oligomers leads to microtubule nucleation
Ayukawa, Rie; Iwata, Seigo; Imai, Hiroshi; Kamimura, Shinji; Hayashi, Masahito; Ngo, Kien Xuan; Minoura, Itsushi; Uchimura, Seiichi; Makino, Tsukasa; Shirouzu, Mikako; Shigematsu, Hideki; Sekimoto, Ken; Gigant, Benoit; Muto, Etsuko
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收藏Discovery of dihydrofuranoallocolchicinoids - Highly potent antimitotic agents with low acute toxicity
Shchegravina, Ekaterina S.; Svirshchevskaya, Elena, V; Combes, Sebastien; Allegro, Diane; Barbier, Pascale; Gigant, Benoit; Varela, Paloma F.; Gavryushin, Andrei E.; Kobanova, Daria A.; Shchekotikhin, Andrey E.; Fedorov, Alexey Yu
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收藏Insight into microtubule nucleation from tubulin-capping proteins从微管蛋白加帽蛋白洞察微管成核
Campanacci, Valerie; Urvoas, Agathe; Cantos-Fernandes, Soraya; Aumont-Nicaise, Magali; Arteni, Ana-Andreea; Velours, Christophe; Valerio-Lepiniec, Marie; Dreier, Birgit; Pluckthun, Andreas; Pilon, Antoine; Pous, Christian; Minard, Philippe; Gigant, Benoit
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收藏1,1-Diheterocyclic Ethylenes Derived from Quinaldine and Carbazole as New Tubulin-Polymerization Inhibitors: Synthesis, Metabolism, and Biological Evaluation
Naret, Timothee; Khelifi, Ilhem; Provot, Olivier; Bignon, Jerome; Levaique, Helene; Dubois, Joelle; Souce, Martin; Kasselouri, Athena; Deroussent, Alain; Paci, Angelo; Varela, Paloma F.; Gigant, Benoit; Alami, Mouad; Hamze, Abdallah
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收藏Mechanism of microtubule stabilization by taccalonolide AJ
Wang, Yuxi; Yu, Yamei; Li, Guo-Bo; Li, Shu-Ang; Wu, Chengyong; Gigant, Benoit; Qin, Wenming; Chen, Hao; Wu, Yangping; Chen, Qiang; Yang, Jinliang
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收藏Structures of a diverse set of colchicine binding site inhibitors in complex with tubulin provide a rationale for drug discovery与微管蛋白复合的秋水仙碱结合位点抑制剂的不同结构为药物发现提供了理论基础
Wang, Yuxi; Zhang, Hang; Gigant, Benoit; Yu, Yamei; Wu, Yangping; Chen, Xiangzheng; Lai, Qinhuai; Yang, Zhaoya; Chen, Qiang; Yang, Jinliang
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