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Yurii S. Moroz

enamine ltd.

34H指数
219论文数
7.5K被引数
收录论文 51
发表时间
Structure based discovery of antipsychotic-like TAAR1 agonists基于结构的抗精神病样TAAR1激动剂的发现
err2026-09-17
err0
errOAAI
errSijie Huang; Heng Liu; Yujin Wu; Joao M. Braz; Divya Kranthi; Brendan W. Hall; Xinyue Zhang; Dmytro S. Radchenko; Yurii S. Moroz; John J. Irwin; Allan I. Basbaum; H. Eric Xu; William C. Wetsel; Brian K. Shoichet
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Development of a random background to understand ligand optimization开发随机背景以理解配体优化
errNature
IF48.5
err2026-09-16
err0
errOAAI
errXinyu Xu; Olivier Mailhot; Galen J. Correy; Xi-Ping Huang; Joao M. Braz; Da Shi; Karthik Srinivasan; Kara Zielinski; Yuliia Holota; Yuliia Kuziv; Christos Iliopoulos-Tsoutsouvas; Nathan D. Levinzon; Yagmur U. Doruk; Moira M. Rachman; Morgan E. Diolaiti; Maisie G. V. Stevens; Fangyu Liu; Katie L. Holland; Harald Hübner; Jing Wang; Yujin Wu; Alan Ashworth; Alexandros Makriyannis; Yuqi Zhang; Yurii S. Moroz; Peter Gmeiner; Robert Abel; Aashish Manglik; Allan I. Basbaum; Bryan L. Roth; James S. Fraser; Brian K. Shoichet
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AI-enhanced adaptive virtual screening of large libraries for ligand discovery用于配体发现的大型文库的AI增强自适应虚拟筛选
err2026-09-01
err0
errOAAI
errDomiziana Cecchini; AkshatKumar Nigam; Ming Tang; Joana Reis; Matt Koop; Andrea Gottinger; Callum Robert Nicoll; Yao Wang; Abhilash Jayaraj; Süleyman Selim Çınaroglu˘; Ricarda Törner; Yehor Malets; Minko Gehev; Krishna M. Padmanabha Das; Kelly Churion; Jongwan Kim; Nidhin Thomas; Yong Li; Hyuk-Soo Seo; Sirano Dhe-Paganon; Christopher Secker; Mohammad Haddadnia; Alexander Hasson; Minkai Li; Abhishek Kumar; Roni Levin-Konigsberg; Eun-Bee Choi; Geoffrey I. Shapiro; Huel Cox; Luke Sebastian; Chelsea Braithwaite; Puspalata Bashyal; Dmytro S. Radchenko; Aditya Kumar; Lei Yang; Pierre-Yves Aquilanti; Henry Gabb; Amr Alhossary; Eric O’Neill; Gerhard Wagner; Alán Aspuru-Guzik; Yurii S. Moroz; Charalampos G. Kalodimos; Konstantin Fackeldey; John D. Schuetz; Andrea Mattevi; Haribabu Arthanari; Christoph Gorgulla
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First Structure–Activity-Relationship Study of Potent G2A Antagonists首次G2A拮抗剂构效关系研究
err2026-06-11
err0
errOAAI
errVictor Hernandez-Olmos; Jan Heering; Felix F. Lillich; Beatrice Marinescu; Sheila Nevermann; Johanna H. M. Ehrler; Dmytro S. Radchenko; Yurii S. Moroz; Astrid Kaiser; Andreas Krämer; Stefan Knapp; Manfred Schubert-Zsilavecz; Mohamad Wessam Alnouri; Stefan Offermanns; Dieter Steinhilber; Marco Sisignano; Ewgenij Proschak
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Ultra-large virtual screening unveils potent agonists of the neuromodulatory orphan receptor GPR139超大规模虚拟筛选揭示了神经调节孤核受体GPR139的强效激动剂
err2025-12-09
err0
errOAAI
errIsrael Cabeza de Vaca; Boris Trapkov; Ling Shen; Duy Duc Vo; Xiaoqun Zhang; Yunting Yang; Mitra Pezeshki; Xuehan Zhang; Frida Bällgren; Aljona Saleh; Andrii V. Tarnovskiy; Dmytro S. Radchenko; Yurii S. Moroz; Hans Bräuner-Osborne; Per Svenningsson; Jan Kihlberg; Zhi-Jie Liu; Alexander Sebastian Hauser; Jens Carlsson
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Expanding Chemical Space of N-Acyl Sulfonamides for Carbonic Anhydrase Inhibitor Discovery扩展N-酰基磺酰胺的化学空间以发现碳酸酐酶抑制剂
err2025-10-23
err0
PREAI
errOleksii V. Gavrylenko; Bohdan V. Vashchenko; Vasyl Naumchyk; Oleksii Chuk; Olga Kuchuk; Alla Pogribna; Anzhelika I. Konovets; Volodymyr S. Brovarets; Sergey A. Zozulya; Dmytro S. Radchenko; Oleksandr O. Grygorenko; Yurii S. Moroz
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Freedom Space 3.0: ML-Assisted Selection of Synthetically Accessible Small MoleculesFreedom Space 3.0:机器学习辅助的可合成小分子筛选
err2025-09-26
err0
PREAI
errAnna Kapeliukha; Serhii Hlotov; Mykola Protopopov; Igor Dzyuba; Maryna Vasylchuk; Dmitriy M. Panov; Olga O. Tarkhanova; Yurii S. Moroz
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A generative deep learning approach to de novo antibiotic design一种用于全新抗生素设计的生成式深度学习方法
errCell
IF42.5
err2025-08-14
err0
PREAI
errAarti Krishnan; Melis N. Anahtar; Jacqueline A. Valeri; Wengong Jin; Nina M. Donghia; Leif Sieben; Andreas Luttens; Yu Zhang; Seyed Majed Modaresi; Andrew Hennes; Jenna Fromer; Parijat Bandyopadhyay; Jonathan C. Chen; Danyal Rehman; Ronak Desai; Paige Edwards; Ryan S. Lach; Marie-Stéphanie Aschtgen; Margaux Gaborieau; Massimiliano Gaetani; Samantha G. Palace; Satotaka Omori; Lutete Khonde; Yurii S. Moroz; Bruce Blough; Chunyang Jin; Edmund Loh; Yonatan H. Grad; Amir Ata Saei; Connor W. Coley; Felix Wong; James J. Collins
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A bottom-up approach to find lead compounds in expansive chemical spaces一种自下而上的方法,用于在广阔的化学空间中寻找先导化合物
err2025-08-01
err0
errOAAI
errÁlvaro Serrano-Morrás; Andrea Bertran-Mostazo; Marina Miñarro-Lleonar; Arnau Comajuncosa-Creus; Adrià Cabello; Carme Labranya; Carmen Escudero; Tian V. Tian; Inna Khutorianska; Dmytro S. Radchenko; Yurii S. Moroz; Lucas Defelipe; David Ruiz-Carrillo; Maria Garcia-Alai; Robert Schmidt; Matthias Rarey; Patrick Aloy; Carles Galdeano; Jordi Juárez-Jiménez; Xavier Barril
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CACHE Challenge #2: Targeting the RNA Site of the SARS-CoV-2 Helicase Nsp13CACHE挑战赛#2:靶向SARS-CoV-2解旋酶Nsp13的RNA位点
err2025-06-20
err0
PREAI
errOleksandra Herasymenko; Madhushika Silva; Abd Al-Aziz A. Abu-Saleh; Ayaz Ahmad; Jesus Alvarado-Huayhuaz; Oscar E. A. Arce; Roly J. Armstrong; Cheryl Arrowsmith; Kelly E. Bachta; Hartmut Beck; Denes Berta; Mateusz K. Bieniek; Vincent Blay; Albina Bolotokova; Philip E. Bourne; Marko Breznik; Peter J. Brown; Aaron D. G. Campbell; Emanuele Carosati; Irene Chau; Daniel J. Cole; Ben Cree; Wim Dehaen; Katrin Denzinger; Karina dos Santos Machado; Ian Dunn; Prasannavenkatesh Durai; Kristina Edfeldt; Aled Edwards; Darren Fayne; Daniel Felfoldi; Kallie Friston; Pegah Ghiabi; Elisa Gibson; Judith Günther; Anders Gunnarsson; Alexander Hillisch; Douglas R. Houston; Jan Halborg Jensen; Rachel J. Harding; Kate S. Harris; Laurent Hoffer; Anders Hogner; Joshua T. Horton; Scott Houliston; Judd F. Hultquist; Ashley Hutchinson; John J. Irwin; Marko Jukič; Shubhangi Kandwal; Andrea Karlova; Vittorio L. Katis; Ryan P. Kich; Dmitri Kireev; David Koes; Nicole L. Inniss; Uta Lessel; Sijie Liu; Peter Loppnau; Wei Lu; Sam Martino; Miles McGibbon; Jens Meiler; Akhila Mettu; Sam Money-Kyrle; Rocco Moretti; Yurii S. Moroz; Charuvaka Muvva; Joseph A. Newman; Leon Obendorf; Brooks Paige; Amit Pandit; Keunwan Park; Sumera Perveen; Rachael Pirie; Gennady Poda; Mykola Protopopov; Vera Pütter; Federico Ricci; Natalie J. Roper; Edina Rosta; Margarita Rzhetskaya; Yogesh Sabnis; Karla J. F. Satchell; Frederico Schmitt Kremer; Thomas Scott; Almagul Seitova; Casper Steinmann; Valerij Talagayev; Olga O. Tarkhanova; Natalie J. Tatum; Dakota Treleaven; Adriano Velasque Werhli; W. Patrick Walters; Xiaowen Wang; Jude Wells; Geoffrey Wells; Yvonne Westermaier; Gerhard Wolber; Lars Wortmann; Jixian Zhang; Zheng Zhao; Shuangjia Zheng; Matthieu Schapira
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A C-Degron Structure-Based Approach for the Development of Ligands Targeting the E3 Ligase TRIM7
err2024-06-27
err1
PREAI
errSosa, Christian J. Munoz; Lenz, Christopher; Hamann, Anton; Farges, Frederic; Dopfer, Johannes; Kraemer, Andreas; Cherkashyna, Veronika; Tarnovskiy, Andrey; Moroz, Yurii S.; Proschak, Ewgenij; Nemec, Vaclav; Mueller, Susanne; Saxena, Krishna; Knapp, Stefan
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Development of a Potent and Selective G2A (GPR132) Agonist
err2024-06-25
err0
PREAI
errHernandez-Olmos, Victor; Heering, Jan; Marinescu, Beatrice; Schermeng, Tina; Ivanov, Vladimir V.; Moroz, Yurii S.; Nevermann, Sheila; Mathes, Marius; Ehrler, Johanna H. M.; Alnouri, Mohamad Wessam; Wolf, Markus; Haydo, Alicia S.; Schmachtel, Tessa; Zaliani, Andrea; Ho''fner, Georg; Kaiser, Astrid; Schubert-Zsilavecz, Manfred; Beck-Sickinger, Annette G.; Offermanns, Stefan; Gribbon, Philipp; Rieger, Michael A.; Merk, Daniel; Sisignano, Marco; Steinhilber, Dieter; Proschak, Ewgenij
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Novel Fragment Inhibitors of PYCR1 from Docking-Guided X-ray Crystallography
err2024-02-27
err2
PREAI
errMeeks, Kaylen R.; Ji, Juan; Protopopov, Mykola V.; Tarkhanova, Olga O.; Moroz, Yurii S.; Tanner, John J.
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SNAr or Sulfonylation? Chemoselective Amination of Halo(het)arene Sulfonyl Halides for Synthetic Applications and Ultralarge Compound Library Design
err2024-02-21
err1
PREAI
errNaumchyk, Vasyl; Andriashvili, Vladyslav A.; Radchenko, Dmytro S.; Dudenko, Dmytro; Moroz, Yurii S.; Tolmachev, Andrey A.; Zhersh, Serhii; Grygorenko, Oleksandr O.
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Docking for EP4R antagonists active against inflammatory pain对炎症性疼痛具有活性的EP4R拮抗剂的对接
err2023-12-06
err12
errOAAI
errGahbauer, Stefan; DeLeon, Chelsea; Braz, Joao M.; Craik, Veronica; Kang, Hye Jin; Wan, Xiaobo; Huang, Xi-Ping; Billesbolle, Christian B.; Liu, Yongfeng; Che, Tao; Deshpande, Ishan; Jewell, Madison; Fink, Elissa A.; Kondratov, Ivan S.; Moroz, Yurii S.; Irwin, John J.; Basbaum, Allan I.; Roth, Bryan L.; Shoichet, Brian K.
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AI-Powered Virtual Screening of Large Compound Libraries Leads to the Discovery of Novel Inhibitors of Sirtuin-1
err2023-07-27
err12
PREAI
errGryniukova, Anastasiia; Kaiser, Florian; Myziuk, Iryna; Alieksieieva, Diana; Leberecht, Christoph; Heym, Peter P.; Tarkhanova, Olga O.; Moroz, Yurii S.; Borysko, Petro; Haupt, V. Joachim
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Structure-Based Discovery of Inhibitors of the SARS-CoV-2 Nsp14 N7-Methyltransferase
err2023-06-09
err14
errOAAI
errSingh, Isha; Li, Fengling; Fink, Elissa A.; Chau, Irene; Li, Alice; Rodriguez-Hernandez, Annia; Glenn, Isabella; Zapatero-Belinchon, Francisco J.; Rodriguez, M. Luis; Devkota, Kanchan; Deng, Zhijie; White, Kris; Wan, Xiaobo; Tolmachova, Nataliya A.; Moroz, Yurii S.; Kaniskan, H. Umit; Ott, Melanie; Garcia-Sastre, Adolfo; Jin, Jian; Fujimori, Danica Galonic; Irwin, John J.; Vedadi, Masoud; Shoichet, Brian K.
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Discovery, Synthesis, and In Vitro Characterization of 2,3 Derivatives of 4,5,6,7-Tetrahydro-Benzothiophene as Potent Modulators of Retinoic Acid Receptor-Related Orphan Receptor γt
err2023-05-12
err3
errOAAI
errFouda, Ahmed; Negi, Sarita; Zaremba, Oleg; Gaidar, Rita S.; Moroz, Yurii S.; Rusanov, Eduard; Paraskevas, Steven; Tchervenkov, Jean
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