arrow
返回
M

Marco Siderius

vrije universiteit

30H指数
92论文数
2.8K被引数
收录论文 36
发表时间
Constitutive activity of an atypical chemokine receptor revealed by inverse agonistic nanobodies由反向激动剂纳米抗体揭示的非典型趋化因子受体的固有活性
err2025-12-02
err0
errOAAI
errClaudia V. Perez Almeria; Omolade Otun; Roman Schlimgen; Thomas D. Lamme; Lotte Di Niro; Caitrin Crudden; Jan Paul Bebelman; Noureldine Youssef; Lejla Musli; Shawn Jenjak; Vladimir Bobkov; Julia Drube; Carsten Hoffmann; Brian F. Volkman; Sébastien Granier; Cherine Bechara; Marco Siderius; Raimond Heukers; Christopher T. Schafer; Martine J. Smit
err分享
err收藏
Pharmacological characterization of a clinical candidate, TG-0 054, a small molecule inverse agonist targeting CXCR4TG-0 054临床候选药物的药理学表征,TG-0 054是一种靶向CXCR4的小分子反向激动剂
err2025-01-01
err0
PREAI
errPan, Kylie S.; Wang, Ziming; Pfeil, Cy; Bergkamp, Nick D.; Mobach, Simon; Roth, Susanne; Rizk, Aurelien; Lohse, Martin J.; Annibale, Paolo; Siderius, Marco; Zimmermann, Mirjam; Smit, Martine J.; Bosma, Reggie
err分享
err收藏
Multivalent CXCR4-targeting nanobody formats differently affect affinity, receptor clustering, and antagonism
err2024-09-01
err1
errOAAI
errAnbuhl, Stephanie M.; Dervillez, Xavier; Neubacher, Saskia; Schriek, Angela I.; Bobkov, Vladimir; de Taeye, Steven W.; Szpakowska, Martyna; Siderius, Marco; Grossmann, Tom N.; Chevigne, Andy; Smit, Martine J.; Heukers, Raimond
err分享
err收藏
A virally encoded GPCR drives glioblastoma through feed-forward activation of the SK1-S1P1 signaling axis
err2023-08-15
err4
PREAI
errBergkamp, Nick D.; van Senten, Jeffrey R.; Brink, Hendrik J.; Bebelman, Maarten P.; van den Bor, Jelle; Cobanoglu, Tugce S.; Dinkla, Kasper; Koester, Johannes; Klau, Gunnar; Siderius, Marco; Smit, Martine J.
err分享
err收藏
Discovery of 5-Phenylpyrazolopyrimidinone Analogs as Potent Antitrypanosomal Agents with In Vivo Efficacy
err2023-07-20
err5
errOAAI
errZheng, Yang; van den Kerkhof, Magali; van der Meer, Tiffany; Gul, Sheraz; Kuzikov, Maria; Ellinger, Bernhard; de Esch, Iwan J. P.; Siderius, Marco; Matheeussen, An; Maes, Louis; Sterk, Geert Jan; Caljon, Guy; Leurs, Rob
err分享
err收藏
The middle domain of Hsp90 acts as a discriminator between different types of client proteins
err2023-03-27
err114
errOAAI
errHawle, Patricija; Siepmann, Martin; Harst, Anja; Siderius, Marco; Reusch, H. Peter; Obermann, Wolfgang M. J.
err分享
err收藏
NanoB2 to monitor interactions of ligands with membrane proteins by combining nanobodies and NanoBRET
err2023-03-01
err5
errOAAI
errvan den Bor, Jelle; Bergkamp, Nick D.; Anbuhl, Stephanie M.; Dekker, Francoise; Comez, Dehan; Almeria, Claudia V. Perez; Bosma, Reggie; White, Carl W.; Kilpatrick, Laura E.; Hill, Stephen J.; Siderius, Marco; Smit, Martine J.; Heukers, Raimond
err分享
err收藏
Fusicoccin-A Targets Cancerous Inhibitor of Protein Phosphatase 2A by Stabilizing a C-Terminal Interaction with 14-3-3
err2022-10-18
err9
errOAAI
errBrink, Hendrik J.; van Senten, Jeffrey R.; De Vries-van Leeuwen, Ingrid J.; Pereira, Daniel da Costa; Piersma, Sander R.; Jimenez, Connie R.; Centorrino, Federica; Ottmann, Christian; Siderius, Marco; Smit, Martine J.; de Boer, Albertus H.
err分享
err收藏
3-nitroimidazo[1,2-b]pyridazine as a novel scaffold for antiparasitics with sub-nanomolar anti-Giardia lamblia activity
err2022-08-01
err7
errOAAI
errZheng, Yang; Mueller, Joachim; Kunz, Stefan; Siderius, Marco; Maes, Louis; Caljon, Guy; Mueller, Norbert; Hemphill, Andrew; Sterk, Geert Jan; Leurs, Rob
err分享
err收藏
Selective targeting of ligand-dependent and -independent signaling by GPCR conformation-specific anti-US28 intrabodies
err2021-07-16
err22
errOAAI
errDe Groof, Timo W. M.; Bergkamp, Nick D.; Heukers, Raimond; Giap, Truc; Bebelman, Maarten P.; Goeij-de Haas, Richard; Piersma, Sander R.; Jimenez, Connie R.; Garcia, K. Christopher; Ploegh, Hidde L.; Siderius, Marco; Smit, Martine J.
err分享
err收藏
From recipe to research: introducing undergraduate students to the nature o science using a hybrid practical course centred on drug discovery for neglected diseases
err2021-06-01
err6
errOAAI
errWijtmans, Maikel; Edink, Ewald; van Linden, Oscar P. J.; Zheng, Yang; Blaazer, Antoni R.; Siderius, Marco; van Muijlwijk-Koezen, Jacqueline E.
err分享
err收藏
Differential Involvement of ACKR3 C-Tail in β-Arrestin Recruitment, Trafficking and Internalization
errCELLS
IF5.2
err2021-03-11
err21
errOAAI
errZarca, Aurelien; Perez, Claudia; van den Bor, Jelle; Bebelman, Jan Paul; Heuninck, Joyce; de Jonker, Rianna J. F.; Durroux, Thierry; Vischer, Henry F.; Siderius, Marco; Smit, Martine J.
err分享
err收藏
Discovery of Diaryl Ether Substituted Tetrahydrophthalazinones as TbrPDEB1 Inhibitors Following Structure-Based Virtual Screening
err2021-01-21
err4
errOAAI
errde Heuvel, Erik; Kooistra, Albert J.; Edink, Ewald; van Klaveren, Sjors; Stuijt, Jeffrey; van der Meer, Tiffany; Sadek, Payman; Mabille, Dorien; Caljon, Guy; Maes, Louis; Siderius, Marco; de Esch, Iwan J. P.; Sterk, Geert Jan; Leurs, Rob
err分享
err收藏
The CXCL12/CXCR4/ACKR3 Axis in the Tumor Microenvironment: Signaling, Crosstalk, and Therapeutic Targeting
err2021-01-06
err43
errOAAI
errSmit, Martine J.; Schlecht-Louf, Geraldine; Neves, Maria; van den Bor, Jelle; Penela, Petronila; Siderius, Marco; Bachelerie, Francoise; Mayor, Federico, Jr.
err分享
err收藏
Cloning and functional complementation of ten Schistosoma mansoni phosphodiesterases expressed in the mammalian host stages
err2020-07-30
err3
errOAAI
errMunday, Jane C.; Kunz, Stefan; Kalejaiye, Titilola D.; Siderius, Marco; Schroeder, Susanne; Paape, Daniel; Alghamdi, Ali H.; Abbasi, Zainab; Huang, Sheng Xiang; Donachie, Anne-Marie; William, Samia; Sabra, Abdel Nasser; Sterk, Geert Jan; Botros, Sanaa S.; Brown, David G.; Hoffman, Charles S.; Leurs, Rob; de Koning, Harry P.
err分享
err收藏
Viral G protein-coupled receptors as modulators of cancer hallmarks
err2020-06-01
err18
errOAAI
errvan Senten, Jeffrey R.; Fan, Tian Shu; Siderius, Marco; Smit, Martine J.
err分享
err收藏
Human Cytomegalovirus-Encoded G Protein-Coupled Receptor UL33 Facilitates Virus Dissemination via the Extracellular and Cell-to-Cell Route
err2020-05-30
err10
errOAAI
errvan Senten, Jeffrey R.; Bebelman, Maarten P.; van Gasselt, Puck; Bergkamp, Nick D.; van den Bor, Jelle; Siderius, Marco; Smit, Martine J.
err分享
err收藏
Lead Optimization of Phthalazinone Phosphodiesterase Inhibitors as Novel Antitrypanosomal Compounds
err2020-03-20
err11
errOAAI
errSalado, Irene G.; Singh, Abhimanyu K.; Moreno-Cinos, Carlos; Sakaine, Guna; Siderius, Marco; Van der Veken, Pieter; Matheeussen, An; van der Meer, Tiffany; Sadek, Payman; Gul, Sheraz; Maes, Louis; Sterk, Geert-Jan; Leurs, Rob; Brown, David; Augustyns, Koen
err分享
err收藏
The human cytomegalovirus-encoded G protein?coupled receptor UL33 exhibits oncomodulatory properties人类巨细胞病毒编码的g蛋白?偶联受体UL33具有调节功能
err2019-11-01
err23
errOAAI
errvan Senten, Jeffrey R.; Bebelman, Maarten P.; Tian Shu Fan; Heukers, Raimond; Bergkamp, Nick D.; van Gasselt, Puck; Langemeijer, Ellen V.; Slinger, Erik; Lagerweij, Tonny; Rahbar, Afsar; Stigter-van Walsum, Marijke; Maussang, David; Leurs, Rob; Musters, Rene J. P.; van Dongen, Guus A. M. S.; Soderberg-Naucler, Cecilia; Wurdinger, Thomas; Siderius, Marco; Smit, Martine J.
err分享
err收藏
Alkynamide phthalazinones as a new class of TbrPDEB1 inhibitors
err2019-09-01
err16
errOAAI
errde Heuvel, Erik; Singh, Abhimanyu K.; Edink, Ewald; van der Meer, Tiffany; van der Woude, Melanie; Sadek, Payman; Krell-Jorgensen, Mikkel P.; van den Bergh, Toine; Veerman, Johan; Caljon, Guy; Kalejaiye, Titilola D.; Wijtmans, Maikel; Maes, Louis; de Koning, Harry P.; Sterk, Geert Jan; Siderius, Marco; de Esch, Iwan J. P.; Brown, David G.; Leurs, Rob
err分享
err收藏