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Marcin Kołaczkowski

faculty of pharmacy

34H指数
180论文数
4.1K被引数
收录论文 95
发表时间
Casticin inhibits AKR1C3 and enhances abiraterone efficacy in castration-resistant prostate cancerCasticin抑制AKR1C3并增强阿比特龙在去势抵抗性前列腺癌中的疗效
err2025-12-10
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errOAAI
errKamil Piska; Michał Zubek; Adam Bucki; Maria Świtalska; Paulina Koczurkiewicz-Adamczyk; Benedykt Władyka; Marcin Kołaczkowski; Elżbieta Pękala
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Simultaneous modulation of 5-HT6 and SERT by MM394: a dual-target ligand providing neuroprotection against amyloid-β toxicity, memory preservation, and alleviation of BPSD symptomsMM394对5-HT6和SERT的同时调节:一种双靶点配体,可提供抗淀粉样β毒性、记忆保留和改善BPSD症状的神经保护作用
err2025-11-10
err0
PREAI
errAgata Siwek; Monika Marcinkowska; Barbara Mordyl; Monika Głuch-Lutwin; Małgorzata Wolak; Magdalena Jastrzębska-Więsek; Natalia Wilczyńska-Zawal; Elżbieta Wyska; Katarzyna Szafrańska; Anna Wesołowska; Marcin Kołaczkowski
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Machine Learning-Driven Discovery of GABA-A Ligands with Pronounced Neuroprotective Efficacy and Resistance to P-gp Efflux机器学习驱动的具有显著神经保护功效且能抵抗P-gp外排的GABA-A配体的发现
err2025-11-03
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PREAI
errKatarzyna Szafrańska; Konstantin Koch; Jakub Jończyk; Barbara Mordyl; Monika Głuch-Lutwin; Bartosz Wojdyła; Dominika Krzysztofik; Agata Siwek; Małgorzata Wolak; Krzysztof Więckowski; Marcin Kołaczkowski; Monika Marcinkowska
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JP-14: A Trace Amine-Associated Receptor 1 Agonist with Anti-Metabolic Disorder PotentialJP-14:一种 Trace Amine-Associated Receptor 1 激动剂,具有抗代谢紊乱的潜力
err2025-10-15
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errOAAI
errMonika Marcinkowska; Joanna Sniecikowska; Monika Głuch-Lutwin; Barbara Mordyl; Marek Bednarski; Adam Bucki; Michał Sapa; Monika Kubacka; Agata Siwek; Agnieszka Zagórska; Jacek Sapa; Marcin Kołaczkowski; Magdalena Kotańska
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Zolpidem suppresses cortical spreading depolarization and protects against ischemia/reperfusion injury and resulting neurological dysfunctions唑吡坦抑制皮层扩散性去极化,并保护缺血/再灌注损伤及由此引起的神经功能障碍
err2025-07-04
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PREAI
errBartosz Pomierny; Mateusz W. Kucharczyk; Weronika Krzyżanowska; Alicja Skórkowska; Jakub Jurczyk; Ewa Niedzielska-Andres; Katarzyna Szafrańska; Małgorzata Wolak; Maria Walczak; Maciej Gawlik; Małgorzata Szafarz; Katarzyna Przejczowska-Pomierny; Elżbieta Wyska; Marcin Kolaczkowski; Lucyna Pomierny-Chamioło; Monika Marcinkowska
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Preferential Synaptic Type of GABA-A Receptor Ligands Enhancing Neuronal Survival and Facilitating Functional Recovery After Ischemic Stroke
err2024-12-13
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PREAI
errMordyl, Barbara; Fajkis-Zajaczkowska, Nikola; Szafranska, Katarzyna; Siwek, Agata; Gluch-Lutwin, Monika; Zmudzki, Pawel; Jonczyk, Jakub; Karcz, Tadeusz; Sloczynska, Karolina; Pekala, Elzbieta; Pomierny, Bartosz; Krzyzanowska, Weronika; Jurczyk, Jakub; Skorkowska, Alicja; Salach, Aleksandra; Jastrzebska-Wiesek, Magdalena; Walczak, Maria; Gawlik, Maciej Tadeusz; Smolik, Magdalena; Kolaczkowski, Marcin; Marcinkowska, Monika
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Dual 5-HT6/SERT ligands for mitigating neuropsychiatric symptoms of dementia exerting neuroprotection against amyloid-β toxicity, memory preservation, and antidepressant-like properties
err2024-09-01
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PREAI
errSiwek, Agata; Marcinkowska, Monika; Gluch-Lutwin, Monika; Mordyl, Barbara; Wolak, Malgorzata; Jastrzebska-Wiesek, Magdalena; Wilczynska-Zawal, Natalia; Wyska, Elzbieta; Szafranska, Katarzyna; Karcz, Tadeusz; Ostrowska, Olga; Bucki, Adam; Kolaczkowski, Marcin
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Novel 1-(1-Arylimiazolin-2-Yl)-3-Arylalkilurea Derivatives with Modulatory Activity on Opioid MOP Receptors
err2024-01-24
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errOAAI
errStraszak, Dominik; Wozniak, Sylwia; Siwek, Agata; Gluch-Lutwin, Monika; Kolaczkowski, Marcin; Pietrzak, Aldona; Drop, Bartlomiej; Matosiuk, Dariusz
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Neuroprotective Activity of Enantiomers of Salsolinol and N-Methyl-(R)-salsolinol: In Vitro and In Silico Studies
err2023-10-05
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errOAAI
errKurnik-Lucka, Magdalena; Latacz, Gniewomir; Bucki, Adam; Rivera-Meza, Mario; Khan, Nadia; Konwar, Jahnobi; Skowron, Kamil; Kolaczkowski, Marcin; Gil, Krzysztof
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Metabolic and cardiovascular benefits and risks of 4-hydroxy guanabenz hydrochloride: a2-adrenoceptor and trace amine-associated receptor 1 ligand
err2023-08-25
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errOAAI
errKotanska, Magdalena; Marcinkowska, Monika; Kuder, Kamil J.; Walczak, Maria; Bednarski, Marek; Siwek, Agata; Kolaczkowski, Marcin
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In Silico and In Vitro Assessment of Carbonyl Reductase 1 Inhibition Using ASP9521-A Potent Aldo-Keto Reductase 1C3 Inhibitor with the Potential to Support Anticancer Therapy Using Anthracycline Antibiotics
err2023-04-27
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errOAAI
errJamrozik, Marek; Piska, Kamil; Bucki, Adam; Koczurkiewicz-Adamczyk, Paulina; Sapa, Michal; Wladyka, Benedykt; Pekala, Elzbieta; Kolaczkowski, Marcin
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Dual Molecules Targeting 5-HT6 and GABA-A Receptors as a New Approach to Combat Depression Associated with Neuroinflammation
err2023-04-04
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errOAAI
errMarcinkowska, Monika; Mordyl, Barbara; Siwek, Agata; Gluch-Lutwin, Monika; Karcz, Tadeusz; Gawalska, Alicja; Sapa, Michal; Bucki, Adam; Szafranska, Katarzyna; Pomierny, Bartosz; Pytka, Karolina; Kotanska, Magdalena; Mika, Kamil; Kolaczkowski, Marcin
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Potential Anti-Amnesic Activity of a Novel Multimodal Derivative of Salicylamide, JJGW08, in Mice
err2023-03-06
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errOAAI
errZmudzka, Elzbieta; Lustyk, Klaudia; Salaciak, Kinga; Siwek, Agata; Jaskowska, Jolanta; Kolaczkowski, Marcin; Sapa, Jacek; Pytka, Karolina
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Ultrasound assisted one-pot synthesis and preliminary in vitro studies of salicylamide arylpiperazines as dual 5-HT1A/5-HT7 ligands
err2023-03-01
err7
PREAI
errJaskowska, Jolanta; Drabczyk, Anna Karolina; Sliwa, Pawel; Jodlowski, Przemyslaw; Pindelska, Edyta; Kulaga, Damian; Zareba, Przemyslaw; Majka, Zbigniew; Siwek, Agata; Wolak, Malgorzata; Kolaczkowski, Marcin
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2-(4-Fluorophenyl)-1H-benzo[d]imidazole as a Promising Template for the Development of Metabolically Robust, α1β2γ2GABA-A Receptor-Positive Allosteric Modulators
err2023-02-27
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errOAAI
errMarcinkowska, Monika; Fajkis-Zajaczkowska, Nikola; Szafranska, Katarzyna; Jonczyk, Jakub; Siwek, Agata; Mordyl, Barbara; Karcz, Tadeusz; Latacz, Gniewomir; Kolaczkowski, Marcin
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Hybrid molecules combining GABA-A and serotonin 5-HT6 receptors activity designed to tackle neuroinflammation associated with depression
err2023-02-01
err10
PREAI
errMarcinkowska, Monika; Mordyl, Barbara; Fajkis-Zajaczkowska, Nikola; Siwek, Agata; Karcz, Tadeusz; Gawalska, Alicja; Bucki, Adam; Zmudzki, Pawel; Partyka, Anna; Jastrzebska-Wiesek, Magdalena; Pomierny, Bartosz; Walczak, Maria; Smolik, Magdalena; Pytka, Karolina; Mika, Kamil; Kotanskad, Magdalena; Kolaczkowski, Marcin
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Spontaneous head twitches in aged rats: behavioral and molecular study
err2022-10-24
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errZakrzewska-Sito, Alicja; Bienkowski, Przemyslaw; Kolaczkowski, Marcin; Nalepa, Irena; Zelek-Molik, Agnieszka; Bielawski, Adam; Chorazka, Katarzyna; Kuczynska, Julita; Mierzejewski, Pawel
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Cinnamamide derivatives with 4-hydroxypiperidine moiety enhance effect of doxorubicin to cancer cells and protect cardiomyocytes against drug-induced toxicity through CBR1 inhibition mechanism
err2022-09-01
err6
PREAI
errKoczurkiewicz-Adamczyk, Paulina; Gasiorkiewicz, Bartosz; Piska, Kamil; Gunia-Krzyzak, Agnieszka; Jamrozik, Marek; Bucki, Adam; Sloczynska, Karolina; Bojdo, Patrycja; Wojcik-Pszczola, Katarzyna; Wladyka, Benedykt; Kolaczkowski, Marcin; Pekala, Elzbieta
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Structural Modeling of TRPA1 Ion Channel-Determination of the Binding Site for Antagonists
err2022-05-11
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errOAAI
errGawalska, Alicja; Kolaczkowski, Marcin; Bucki, Adam
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