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Targeting microbial β-CAs: bridging in silico screening with in vitro validation Tondo, Anna Rita; Fantacuzzi, Marialuigia; Carradori, Simone; D'Agostino, Ilaria; Angeli, Andrea; Supuran, Claudiu T.; Capasso, Clemente; Gambacorta, Nicola; Piemontese, Luca; Laghezza, Antonio; Nicolotti, Orazio; Tortorella, Paolo; Agamennone, Mariangela 分享 收藏
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Deep Eutectic Solvents (DESs) as Alternative Sustainable Media for the Extraction and Characterization of Bioactive Compounds from Winemaking Industry Wastes Roselli, Vincenzo; Leuci, Rosalba; Pugliese, Gianluca; Barbarossa, Alexia; Laghezza, Antonio; Paparella, Marco; Carocci, Alessia; Tufarelli, Vincenzo; Gambacorta, Lucia; Piemontese, Luca 分享 收藏
A chemical modification of a peroxisome proliferator-activated receptor pan agonist produced a shift to a new dual alpha/gamma partial agonist endowed with mitochondrial pyruvate carrier inhibition and antidiabetic properties (vol 275, 116567, 2024) Laghezza, Antonio; Cerchia, Carmen; Genovese, Massimo; Montanari, Roberta; Capelli, Davide; Wackerlig, Judith; Simic, Stefan; Falbo, Emanuele; Pecora, Lucia; Leuci, Rosalba; Brunetti, Leonardo; Piemontese, Luca; Tortorella, Paolo; Biswas, Abanish; Singh, Ravi Pratap; Tambe, Suhas; Sudeep, C. A.; Pattnaik, Ashok Kumar; Jayaprakash, Venkatesan; Paoli, Paolo; Lavecchia, Antonio; Loiodice, Fulvio 分享 收藏
A chemical modification of a peroxisome proliferator-activated receptor pan agonist produced a shift to a new dual alpha/gamma partial agonist endowed with mitochondrial pyruvate carrier inhibition and antidiabetic properties Laghezza, Antonio; Cerchia, Carmen; Genovese, Massimo; Montanari, Roberta; Capelli, Davide; Wackerlig, Judith; Simic, Stefan; Falbo, Emanuele; Pecora, Lucia; Leuci, Rosalba; Brunetti, Leonardo; Piemontese, Luca; Tortorella, Paolo; Biswas, Abanish; Singh, Ravi Pratap; Tambe, Suhas; Sudeep, C. A.; Pattnaik, Ashok Kumar; Jayaprakash, Venkatesan; Paoli, Paolo; Lavecchia, Antonio; Loiodice, Fulvio 分享 收藏
Chiral pyrrolidines as multipotent agents in Alzheimer and neurodegenerative diseases Carrieri, Antonio; Barbarossa, Alexia; de Candia, Modesto; Samarelli, Francesco; Altomare, Cosimo Damiano; Czarnota-Lydka, Kinga; Sudol-Talaj, Sylwia; Latacz, Gniewomir; Handzlik, Jadwiga; Brunetti, Leonardo; Piemontese, Luca; Limongelli, Francesco; Lentini, Giovanni; Carocci, Alessia 分享 收藏
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A New Antidiabetic Agent Showing Short- and Long-Term Effects Due to Peroxisome Proliferator-Activated Receptor Alpha/Gamma Dual Agonism and Mitochondrial Pyruvate Carrier Inhibition Laghezza, Antonio; Cerchia, Carmen; Genovese, Massimo; Leuci, Rosalba; Pranzini, Erica; Santi, Alice; Brunetti, Leonardo; Piemontese, Luca; Tortorella, Paolo; Biswas, Abanish; Singh, Ravi Pratap; Tambe, Suhas; Ca, Sudeep; Pattnaik, Ashok Kumar; Jayaprakash, Venkatesan; Paoli, Paolo; Lavecchia, Antonio; Loiodice, Fulvio 分享 收藏
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Novel Phenothiazine/Donepezil-like Hybrids Endowed with Antioxidant Activity for a Multi-Target Approach to the Therapy of Alzheimer's Disease Carocci, Alessia; Barbarossa, Alexia; Leuci, Rosalba; Carrieri, Antonio; Brunetti, Leonardo; Laghezza, Antonio; Catto, Marco; Limongelli, Francesco; Chaves, Silvia; Tortorella, Paolo; Altomare, Cosimo Damiano; Santos, Maria Amelia; Loiodice, Fulvio; Piemontese, Luca 分享 收藏
Food Industry Byproducts as Starting Material for Innovative, Green Feed Formulation: A Sustainable Alternative for Poultry Feeding Brunetti, Leonardo; Leuci, Rosalba; Colonna, Maria Antonietta; Carrieri, Rossana; Celentano, Francesco Emanuele; Bozzo, Giancarlo; Loiodice, Fulvio; Selvaggi, Maria; Tufarelli, Vincenzo; Piemontese, Luca 分享 收藏
Structure-based design of novel donepezil-like hybrids for a multi-target approach to the therapy of Alzheimer's disease Brunetti, Leonardo; Leuci, Rosalba; Carrieri, Antonio; Catto, Marco; Occhineri, Sara; Vinci, Giuseppe; Gambacorta, Lucia; Baltrukevich, Hanna; Chaves, Silvia; Laghezza, Antonio; Altomare, Cosimo Damiano; Tortorella, Paolo; Santos, M. Amelia; Loiodice, Fulvio; Piemontese, Luca 分享 收藏
Novel Rivastigmine Derivatives as Promising Multi-Target Compounds for Potential Treatment of Alzheimer's Disease 新型卡巴拉汀衍生物作为潜在的治疗阿尔茨海默病的多靶点化合物 Vicente-Zurdo, David; Rosales-Conrado, Noelia; Eugenia Leon-Gonzalez, M.; Brunetti, Leonardo; Piemontese, Luca; Raquel Pereira-Santos, A.; Cardoso, Sandra M.; Madrid, Yolanda; Chaves, Silvia; Amelia Santos, M. 分享 收藏
A chemoinformatics search for peroxisome proliferator-activated receptors ligands revealed a new pan-agonist able to reduce lipid accumulation and improve insulin sensitivity 对过氧化物酶体增殖物激活受体配体的化学信息学搜索揭示了一种新的泛激动剂,能够减少脂质积累并改善胰岛素敏感性 Sblano, Sabina; Cerchia, Carmen; Laghezza, Antonio; Piemontese, Luca; Brunetti, Leonardo; Leuci, Rosalba; Gilardi, Federica; Thomas, Aurelien; Genovese, Massimo; Santi, Alice; Tortorella, Paolo; Paoli, Paolo; Lavecchia, Antonio; Loiodice, Fulvio 分享 收藏
A New Series of Aryloxyacetic Acids Endowed with Multi-Target Activity towards Peroxisome Proliferator-Activated Receptors (PPARs), Fatty Acid Amide Hydrolase (FAAH), and Acetylcholinesterase (AChE) Leuci, Rosalba; Brunetti, Leonardo; Laghezza, Antonio; Piemontese, Luca; Carrieri, Antonio; Pisani, Leonardo; Tortorella, Paolo; Catto, Marco; Loiodice, Fulvio 分享 收藏
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