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T

Terry Kenakin

University of North Carolina

62H指数
403论文数
1.7W被引数
收录论文 101
发表时间
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Receptor kinetics: Binding flux-based approaches offer complementary insight into how ligand binding evolves with time受体动力学：基于结合通量的方法为配体结合如何随时间演变提供了互补的见解
errBritish Journal of Pharmacology
IF7.7
err2026-08-15
err0
errOAAI
errGeorges Vauquelin; Terry Kenakin; Dominique Maes
err分享
err收藏
Kinetic Benefit(s) of Allosteric Receptor Blockade by Positive Allosteric Modulator Antagonists正别构调节剂拮抗剂对别构受体阻滞的动力学益处
errACS Pharmacology & Translational Science
IF3.7
err2026-08-14
err0
PREAI
errGeorges Vauquellin; Terry Kenakin
err分享
err收藏
Biased Signaling as Allosteric Probe Dependence: Everything Old Is New Again偏向性信号作为别构探针依赖性：旧貌换新颜
errBiochemistry
IF3
err2026-04-29
err0
PREAI
errTerry Kenakin
err分享
err收藏
Structure-based design of an opioid receptor modulator for enhanced morphine analgesia基于结构的阿片受体调节剂的设计，以增强吗啡镇痛效果
errScience Advances
IF12.5
err2026-02-11
err0
errOAAI
errYue Wang; Ping Luo; Haiyan Xu; Li Zhan; Kensuke Sakamoto; Mingyu Li; Jing Wang; Xi-Ping Huang; Jianhui Zhou; Tao Liu; Yanrui Suo; Wenjia Fan; Xinheng He; Youwei Xu; Yongjie Cai; Chao Wang; Yuxi Zhao; Antao Dai; Yali Lai; Qingning Yuan; Wen Hu; Kai Wu; Dehua Yang; Xi Cheng; Xiaojie Lu; Brian Krumm; Terry Kenakin; Jian Zhang; Bryan L. Roth; Zhaobing Gao; H. Eric Xu; Youwen Zhuang
err分享
err收藏
Differential Effects of Sodium on Agonist-Induced Conformational Transitions and Signaling at μ and κ Opioid Receptors钠离子对μ和κ阿片受体激动剂诱导的构象转变和信号传导的差异性影响
errBIOCHEMISTRY
IF3
err2025-12-01
err0
PREAI
errKuijer, Michael Bram; Fulton, Camryn J.; Albert, Talia L.; Knobloch, Paloma; Wang, Jing; Krumm, Brian E.; Che, Tao; Varga, Balazs R.; Majumdar, Susruta; Katritch, Vsevolod; Gumpper, Ryan H.; Kenakin, Terry; Huang, Xi-Ping; Roth, Bryan L.
err分享
err收藏
Molecular mechanisms of inverse agonism via κ-opioid receptor-G protein complexesκ-阿片受体-G蛋白复合物的反向激动分子机制
errNATURE CHEMICAL BIOLOGY
IF13.7
err2025-01-07
err0
errOAAI
errTyson, Aaliyah S.; Khan, Saif; Motiwala, Zenia; Han, Gye Won; Zhang, Zixin; Ranjbar, Mohsen; Styrpejko, Daniel; Ramos-Gonzalez, Nokomis; Woo, Stone; Villers, Kelly; Landaker, Delainey; Kenakin, Terry; Shenvi, Ryan; Majumdar, Susruta; Gati, Cornelius
err分享
err收藏
Intracellular Allosteric Antagonist of the Olfactory Receptor OR51E2 S
errMOLECULAR PHARMACOLOGY
IF3
err2024-07-01
err0
errOAAI
errAbaffy, Tatjana; Fu, Olivia; Harume-Nagai, Maira; Goldenberg, Josh M.; Kenyon, Victor; Kenakin, Terry
err分享
err收藏
Know your molecule: pharmacological characterization of drug candidates to enhance efficacy and reduce late-stage attrition了解您的分子: 候选药物的药理学表征，以增强疗效并减少后期损耗
errNATURE REVIEWS DRUG DISCOVERY
IF101.8
err2024-06-18
err1
PREAI
errKenakin, Terry
err分享
err收藏
A Pharmacological perspective on the temporal properties of sweeteners
errPHARMACOLOGICAL RESEARCH
IF10.5
err2024-06-01
err1
errOAAI
errServant, Guy; Kenakin, Terry
err分享
err收藏
Bias translation: The final frontier?
errBRITISH JOURNAL OF PHARMACOLOGY
IF7.7
err2024-02-29
err2
errOAAI
errKenakin, Terry
err分享
err收藏
Allostery: The Good, the Bad, and the Ugly
errJOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS
IF3.8
err2024-01-01
err4
errOAAI
errKenakin, Terry
err分享
err收藏
Community guidelines for GPCR ligand bias: IUPHAR review 32GPCR配体偏倚的社区指南: IUPHAR综述32
errBRITISH JOURNAL OF PHARMACOLOGY
IF7.7
err2022-03-27
err101
errOAAI
errKolb, Peter; Kenakin, Terry; Alexander, Stephen P. H.; Bermudez, Marcel; Bohn, Laura M.; Breinholt, Christian S.; Bouvier, Michel; Hill, Stephen J.; Kostenis, Evi; Martemyanov, Kirill A.; Neubig, Rick R.; Onaran, H. Ongun; Rajagopal, Sudarshan; Roth, Bryan L.; Selent, Jana; Shukla, Arun K.; Sommer, Martha E.; Gloriam, David E.
err分享
err收藏
Development of 3-(4-Chlorophenyl)-1-(phenethyl)urea Analogues as Allosteric Modulators of the Cannabinoid Type-1 Receptor: RTICBM-189 is Brain Penetrant and Attenuates Reinstatement of Cocaine-Seeking Behavior
errJOURNAL OF MEDICINAL CHEMISTRY
IF6.8
err2021-12-20
err7
errOAAI
errThuy Nguyen; Gamage, Thomas F.; Finlay, David B.; Decker, Ann M.; Langston, Tiffany L.; Barrus, Daniel; Glass, Michelle; Li, Jun-Xu; Kenakin, Terry P.; Zhang, Yanan
err分享
err收藏
Biased signaling as allosteric probe dependence
errCELLULAR SIGNALLING
IF3.7
err2021-03-01
err12
PREAI
errKenakin, Terry
err分享
err收藏
GB001 is a potent, insurmountable DP2 antagonist with long receptor residence time and extended pharmacodynamic effects
errEUROPEAN RESPIRATORY JOURNAL
IF21
err2020-10-28
err0
PREAI
errSahdeo, Sunil; Meadows, Kristen Taylor; Hoare, Sam; Kenakin, Terry; Murphy, Susan; Salter-Cid, Tomas; Ortega, Hector; Opiteck, Gregory; Salter-Cid, Luisa; Carter, Laura
err分享
err收藏
Preclinical Testing of Nalfurafine as an Opioid-sparing Adjuvant that Potentiates Analgesia by the Mu Opioid Receptor-targeting Agonist Morphine
errJOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS
IF3.8
err2019-11-01
err44
errOAAI
errKaski, Shane W.; White, Allison N.; Gross, Joshua D.; Trexler, Kristen R.; Wix, Kim; Harland, Aubrie A.; Prisinzano, Thomas E.; Aube, Jeffrey; Kinsey, Steven G.; Kenakin, Terry; Siderovski, David P.; Setola, Vincent
err分享
err收藏
Discovery and Characterization of a Cellular Potent Positive Allosteric Modulator of the Polycomb Repressive Complex 1 Chromodomain, CBX7
errCELL CHEMICAL BIOLOGY
IF7.2
err2019-10-01
err48
errOAAI
errLamb, Kelsey N.; Bsteh, Daniel; Dishman, Sarah N.; Moussa, Hagar F.; Fan, Huitao; Stuckey, Jacob I.; Norris, Jacqueline L.; Cholensky, Stephanie H.; Li, Dongxu; Wang, Jingkui; Sagum, Cari; Stanton, Benjamin Z.; Bedford, Mark T.; Pearce, Kenneth H.; Kenakin, Terry P.; Kireev, Dmitri B.; Wang, Gang Greg; James, Lindsey I.; Bell, Oliver; Frye, Stephen V.
err分享
err收藏
Can we use Nature's Structure-Activity-Relationships to Make Better Drugs?
errDRUG DISCOVERY TODAY
IF7.5
err2019-09-01
err0
PREAI
errKenakin, Terry
err分享
err收藏
Design, Synthesis, and Characterization of Ogerin-Based Positive Allosteric Modulators for G Protein-Coupled Receptor 68 (GPR68)
errJOURNAL OF MEDICINAL CHEMISTRY
IF6.8
err2019-07-12
err21
errOAAI
errYu, Xufen; Huang, Xi-Ping; Kenakin, Terry P.; Slocum, Samuel T.; Chen, Xin; Martini, Michael L.; Liu, Jing; Jin, Jian
err分享
err收藏
Prescient Indices of Activity: The Application of Functional System Sensitivity to Measurement of Drug Effect有先见之明的活性指标: 功能系统敏感性在药物作用测量中的应用
errTRENDS IN PHARMACOLOGICAL SCIENCES
IF19.9
err2019-07-01
err0
PREAI
errKenakin, Terry
err分享
err收藏

研究方向

暂无研究方向
合作学者
合作期刊
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William A. Catterall
H 指数: 162 · 论文数: 652
B
Bryan L. Roth
H 指数: 139 · 论文数: 971
J
John A. Cidlowski
H 指数: 115 · 论文数: 551
M
Michel Bouvier
H 指数: 108 · 论文数: 808
H
H. Eric Xu
H 指数: 100 · 论文数: 623
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