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Zhengfang Yi

Institute of Biomedical Sciences and School of Life Sciences

49H-index
179Paper Count
8.1KCitation Count
Published Papers 98
Publication Date
Synthesis and biological evaluation of cyanoenone- and enone-fused 4-androstene-3,17-dione derivatives against triple-negative breast cancer
err2026-09-13
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PREAI
errJing-Zan Zhang; Yunxuan Li; Jin-Hui Huang; Min Wu; Qiaobing Yue; Mingyao Liu; Chen-Chen Li; Zhengfang Yi; Wen-Wei Qiu
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A novel small-molecule inhibitor of IRF4 selectively suppresses multiple myeloma
err2026-04-03
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errOAAI
errLin Zhang; Xin Ding; Min Wu; Jing-Zan Zhang; Huang Chen; Mingyao Liu; Wen-Wei Qiu; Zhengfang Yi
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Design and synthesis of novel N-phenyl-4-pyrimidine-diamine BCL6 inhibitors with anti-tumor activities
err2025-09-01
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PREAI
errLi, Yan; Xing, Yajing; Huang, Dongxia; Xie, Jiuqing; Peng, Yangrui; Yi, Zhengfang; Chen, Yihua
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Selectively targeting BCL6 using a small-molecule inhibitor is a potential therapeutic strategy for glioblastoma
err2025-04-15
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errOAAI
errMin Wu; Lin Zhang; Weikai Guo; Shiyi Lv; Wangrui Jin; Shuangshuang Zhu; Huang Chen; Shuyi Jian; Layang Liu; Yajing Xing; Shihong Peng; Mingyao Liu; Yihua Chen; Zhengfang Yi
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Design, synthesis and biological evaluation of bisnoralcohol derivatives as novel IRF4 inhibitors for the treatment of multiple myeloma
err2025-03-01
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PREAI
errZhang, Jing-Zan; Zhang, Lin; Ding, Xin; Wu, Min; Zhang, De-Jie; Wu, Yujie; Liu, Mingyao; Li, Chen-Chen; Yi, Zhengfang; Qiu, Wen-Wei
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IRE1α inhibitor reduces cisplatin resistance in ovarian cancer by modulating IRE1α/XBP1 pathway
err2024-11-20
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PREAI
errLv, Shiyi; Zhang, Lin; Wu, Min; Zhu, Shuangshuang; Wang, Yixue; Liu, Layang; Li, Yunxuan; Zhang, Ting; Wu, Yujie; Chen, Huang; Liu, Mingyao; Yi, Zhengfang
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A Small-Molecule BCL6 Inhibitor as an Anti-Proliferative Agent for Diffuse Large B-Cell Lymphoma
err2024-10-10
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PREAI
errXing, Yajing; Guo, Weikai; Wu, Min; Xie, Jiuqing; Huang, Dongxia; Hu, Pan; Zhou, Miaoran; Zhang, Lin; Zhong, Yadong; Liu, Mingyao; Chen, Yihua; Yi, Zhengfang
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Remodeling the immune microenvironment for gastric cancer therapy through antagonism of prostaglandin E2 receptor 4
err2024-07-01
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errOAAI
errGuo, Mengmeng; Hu, Pan; Xie, Jiayi; Tang, Kefu; Hu, Shixiu; Sun, Jialiang; He, Yundong; Li, Jing; Lu, Weiqiang; Liu, Huirong; Liu, Mingyao; Yi, Zhengfang; Peng, Shihong
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IRE1α inhibitor enhances paclitaxel sensitivity of triple-negative breast cancer cells
err2024-06-18
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PREAI
errWu, Min; Zhang, Lin; Pi, Lifu; Liu, Layang; Wang, Siyu; Wu, Yujie; Pan, Hongli; Liu, Mingyao; Yi, Zhengfang
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Targeting STAT3 by a small molecule suppresses pancreatic cancer progression (vol 40, pg 1440, 2021)
err2024-06-05
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errOAAI
errChen, Huang; Bian, Aiwu; Yang, Lian-fang; Yin, Xuan; Wang, Jie; Ti, Chaowen; Miao, Ying; Peng, Shihong; Xu, Shifen; Liu, Mingyao; Qiu, Wen-Wei; Yi, Zhengfang
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Discovery of the Highly Selective and Potent STAT3 Inhibitor for Pancreatic Cancer Treatment
err2024-02-10
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errOAAI
errChen, Huang; Bian, Aiwu; Zhou, Wenbo; Miao, Ying; Ye, Jiangnan; Li, Jiahui; He, Peng; Zhang, Qiansen; Sun, Yue; Sun, Zhenliang; Ti, Chaowen; Chen, Yihua; Yi, Zhengfang; Liu, Mingyao
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WB518, a novel STAT3 inhibitor, effectively alleviates IMQ and TPA-induced animal psoriasis by inhibiting STAT3 phosphorylation and Keratin 17
err2024-01-01
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PREAI
errTi, Chaowen; Chen, Huang; Zhou, Wenbo; Bian, Aiwu; Hu, Pan; Miao, Ying; Shao, Ting; Liu, Mingyao; Chen, Yihua; Yi, Zhengfang
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Discovery of a Highly Potent and Selective MYOF Inhibitor with Improved Water Solubility for the Treatment of Gastric Cancer
err2023-12-06
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PREAI
errGu, Haijun; Zhang, Ting; Guan, Tian; Wu, Min; Li, Shen; Li, Yunqi; Guo, Mengmeng; Zhang, Lin; Peng, Yangrui; Mi, Dazhao; Liu, Mingyao; Yi, Zhengfang; Chen, Yihua
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A small molecule BCL6 inhibitor as chemosensitizers in acute myeloid leukemia
err2023-10-01
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errOAAI
errZhang, Lin; Wu, Min; Guo, Weikai; Zhu, Shuangshuang; Li, Shen; Lv, Shiyi; Li, Yan; Liu, Layang; Xing, Yajing; Chen, Huang; Liu, Mingyao; Peng, Shihong; Chen, Yihua; Yi, Zhengfang
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Combined treatment of disulfiram with PARP inhibitors suppresses ovarian cancer
err2023-04-18
err7
errOAAI
errTang, Bin; Wu, Min; Zhang, Lin; Jian, Shuyi; Lv, Shiyi; Lin, Tongyuan; Zhu, Shuangshuang; Liu, Layang; Wang, Yixue; Yi, Zhengfang; Jiang, Feiyun
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Discovery of 1,5-diaryl-1,2,4-triazole derivatives as myoferlin inhibitors and their antitumor effects in pancreatic cancer
err2022-09-27
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PREAI
errGu, Haijun; Zhang, Ting; Li, Yunqi; He, Yuan; Guan, Tian; Kan, Weiqiong; He, Peng; Yi, Zhengfang; Chen, Yihua
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Discovery of a Novel Potent STAT3 Inhibitor HP590 with Dual p-Tyr705/Ser727 Inhibitory Activity for Gastric Cancer Treatment
err2022-09-14
err11
PREAI
errHe, Peng; Miao, Ying; Sun, Yue; Bian, Aiwu; Jin, Wangrui; Ye, Jiangnan; Chen, Huang; He, Jia; Peng, Yangrui; Gu, Haijun; Liu, Mingyao; Yi, Zhengfang; Chen, Yihua
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Discovery of 2-Amino-3-cyanothiophene Derivatives as PotentSTAT3 Inhibitors for the Treatment of Osteosarcoma Growth and Metastasis
err2022-04-27
err19
PREAI
errJin, Wangrui; Zhang, Tao; Zhou, Wenbo; He, Peng; Sun, Yue; Hu, Shijia; Chen, Huang; Ma, Xinglong; Peng, Yangrui; Yi, Zhengfang; Liu, Mingyao; Chen, Yihua
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A novel small-molecule activator of unfolded protein response suppresses castration-resistant prostate cancer growth
err2022-04-01
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PREAI
errChen, Huang; Miao, Ying; Bian, Aiwu; Ye, Jiangnan; Wang, Jing; Cong, Xiaonan; Jian, Shuyi; Yi, Zhengfang; Liang, Lin; Sun, Zhenliang; Yang, Fan; Ding, Tao
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An orally available small molecule BCL6 inhibitor effectively suppresses diffuse large B cell lymphoma cells growth in vitro and in vivo
err2022-03-01
err12
errOAAI
errXing, Yajing; Guo, Weikai; Wu, Min; Xie, Jiuqing; Huang, Dongxia; Hu, Pan; Zhou, Miaoran; Zhang, Lin; Zhang, Qiansen; Wang, Peili; Wang, Xin; Wang, Guixue; Wu, Huangan; Zhou, Cili; Chen, Yihua; Liu, Mingyao; Yi, Zhengfang; Sun, Zhenliang
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