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Design, synthesis and antiproliferative activity evaluation of new 3,7-disubstituted pyrrolo[2,3-c]pyridines Zografistou, Marianthi; Georgiou, Maria; Mikropoulou, Eleni, V; Halabalaki, Maria; Lougiakis, Nikolaos; Pouli, Nicole; Marakos, Panagiotis; Mavrogonatou, Eleni; Pratsinis, Harris; Kletsas, Dimitris Share Save
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Generation of a selective senolytic platform using a micelle-encapsulated Sudan Black B conjugated analog (vol 5, pg 162, 2025) Magkouta, Sophia; Veroutis, Dimitris; Papaspyropoulos, Angelos; Georgiou, Maria; Lougiakis, Nikolaos; Pippa, Natassa; Havaki, Sophia; Palaiologou, Anastasia; Thanos, Dimitris-Foivos; Kambas, Konstantinos; Lagopati, Nefeli; Boukos, Nikos; Pouli, Nicole; Marakos, Panagiotis; Kotsinas, Athanassios; Thanos, Dimitris; Evangelou, Konstantinos; Sampaziotis, Fotios; Tamvakopoulos, Constantin; Pispas, Stergios; Petty, Russell; Kotopoulos, Nicholas; Gorgoulis, Vassilis G. Share Save
Generation of a selective senolytic platform using a micelle-encapsulated Sudan Black B conjugated analog Magkouta, Sophia; Veroutis, Dimitris; Papaspyropoulos, Angelos; Georgiou, Maria; Lougiakis, Nikolaos; Pippa, Natassa; Havaki, Sophia; Palaiologou, Anastasia; Thanos, Dimitris-Foivos; Kambas, Konstantinos; Lagopati, Nefeli; Boukos, Nikos; Pouli, Nicole; Marakos, Panagiotis; Kotsinas, Athanassios; Thanos, Dimitris; Evangelou, Konstantinos; Sampaziotis, Fotios; Tamvakopoulos, Constantin; Pispas, Stergios; Petty, Russell; Kotopoulos, Nicholas; Gorgoulis, Vassilis G. Share Save
The pyrazolo[4,3-c]pyrazole core as a novel and versatile scaffold for developing dual DYRK1A-CLK1 inhibitors targeting key processes of Alzheimer's disease pathology Bakalakou, Vaia-Argyro; Mavroidi, Barbara; Kalampaliki, Amalia D.; Josselin, Beatrice; Bach, Stephane; Skaltsounis, Alexios-Leandros; Marakos, Panagiotis; Pouli, Nicole; Pelecanou, Maria; Myrianthopoulos, Vassilios; Ruchaud, Sandrine; Kostakis, Ioannis K. Share Save
The pyrazolo[4,3-c]pyrazole core as a novel and versatile scaffold for developing dual DYRK1A-CLK1 inhibitors targeting key processes of Alzheimer's disease pathology (vol 12, 100193, 2024) Bakalakou, Vaia-Argyro; Mavroidi, Barbara; Kalampaliki, Amalia D.; Josselin, Beatrice; Bach, Stephane; Skaltsounis, Alexios-Leandros; Marakos, Panagiotis; Pouli, Nicole; Pelecanou, Maria; Myrianthopoulos, Vassilios; Ruchaud, Sandrine; Kostakis, Ioannis K. Share Save
Hit-to-Lead Optimization of Heterocyclic Carbonyloxycarboximidamides as Selective Antagonists at Human Adenosine A3 Receptor Huang, Xianglin; Chorianopoulou, Anna; Kalkounou, Panagoula; Georgiou, Maria; Pousias, Athanasios; Davies, Amy; Pearce, Abigail; Harris, Matthew; Lambrinidis, George; Marakos, Panagiotis; Pouli, Nicole; Kolocouris, Antonios; Lougiakis, Nikolaos; Ladds, Graham Share Save
Synthesis, cytotoxic activity evaluation and mechanistic investigation of novel 3,7-diarylsubstituted 6-azaindoles Lougiakis, Nikolaos; Sakalis, Nikolaos; Georgiou, Maria; Marakos, Panagiotis; Pouli, Nicole; Skaltsounis, Alexios-Leandros; Mavrogonatou, Eleni; Pratsinis, Harris; Kletsas, Dimitris Share Save
Hydrolytic Activity of Mitochondrial F1FO-ATP Synthase as a Target for Myocardial Ischemia-Reperfusion Injury: Discovery and In Vitro and In Vivo Evaluation of Novel Inhibitors Nikolaou, Panagiota-Efstathia; Lambrinidis, George; Georgiou, Maria; Karagiannis, Dimitrios; Efentakis, Panagiotis; Bessis-Lazarou, Pavlos; Founta, Konstantina; Kampoukos, Stavros; Konstantin, Vasilis; Palmeira, Carlos M.; Davidson, Sean M.; Lougiakis, Nikolaos; Marakos, Panagiotis; Pouli, Nicole; Mikros, Emmanuel; Andreadou, Ioanna Share Save
A fluorophore-conjugated reagent enabling rapid detection, isolation and live tracking of senescent cells Magkouta, Sophia; Veroutis, Dimitris; Pousias, Athanasios; Papaspyropoulos, Angelos; Pippa, Natassa; Lougiakis, Nikolaos; Kambas, Konstantinos; Lagopati, Nefeli; Polyzou, Aikaterini; Georgiou, Maria; Chountoulesi, Maria; Pispas, Stergios; Foutadakis, Spyros; Pouli, Nicole; Marakos, Panagiotis; Kotsinas, Athanassios; Verginis, Panayotis; Valakos, Dimitrios; Mizi, Athanasia; Papantonis, Argyris; Vatsellas, Giannis; Galanos, Panagiotis; Bartek, Jiri; Petty, Russell; Serrano, Manuel; Thanos, Dimitris; Roussos, Charis; Demaria, Marco; Evangelou, Konstantinos; Gorgoulis, Vassilis G. Share Save
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Novel H2S-Releasing Bifunctional Antihistamine Molecules with Improved Antipruritic and Reduced Sedative Actions Antoniadou, Ivi; Georgiou, Maria; Dotsikas, Yannis; Lamprou, Alexandra; Lougiakis, Nikolaos; Pouli, Nicole; Karousis, Nikolaos; Loukas, Yannis; Tseti, Ioulia; Marakos, Panagiotis; Papapetropoulos, Andreas Share Save
Discovery of New 1,4,6-Trisubstituted-1H-pyrazolo[3,4-b]pyridines with Anti-Tumor Efficacy in Mouse Model of Breast Cancer Georgiou, Maria; Lougiakis, Nikolaos; Tenta, Roxane; Gioti, Katerina; Baritaki, Stavroula; Gkaralea, Lydia-Evangelia; Deligianni, Elisavet; Marakos, Panagiotis; Pouli, Nicole; Stellas, Dimitris Share Save
Dual A1/A3 Adenosine Receptor Antagonists: Binding Kinetics and Structure-Activity Relationship Studies Using Mutagenesis and Alchemical Binding Free Energy Calculations Stampelou, Margarita; Suchankova, Anna; Tzortzini, Efpraxia; Dhingra, Lakshiv; Barkan, Kerry; Lougiakis, Nikolaos; Marakos, Panagiotis; Pouli, Nicole; Ladds, Graham; Kolocouris, Antonios Share Save
Discovery of a High Affinity Adenosine A1/A3 Receptor Antagonist with a Novel 7-Amino-pyrazolo[3,4-d]pyridazine Scaffold Suchankova, Anna; Stampelou, Margarita; Koutsouki, Klontiana; Pousias, Athanasios; Dhingra, Lakshiv; Barkan, Kerry; Pouli, Nicole; Marakos, Panagiotis; Tenta, Roxane; Kolocouris, Antonios; Lougiakis, Nikolaos; Ladds, Graham Share Save
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New bioactive 5-arylcarboximidamidopyrazolo[3,4-c]pyridines: Synthesis, cytotoxic activity, mechanistic investigation and structure-activity relationships Papastathopoulos, Athanasios; Lougiakis, Nikolaos; Kostakis, Ioannis K.; Marakos, Panagiotis; Pouli, Nicole; Pratsinis, Harris; Kletsas, Dimitris Share Save
Synthesis of novel xanthone and acridone carboxamides with potent antiproliferative activities Georgakopoulos, Antonios; Kalampaliki, Amalia D.; Gioti, Katerina; Hamdoun, Sami; Giannopoulou, Aikaterini F.; Efferth, Thomas; Stravopodis, Dimitrios J.; Tenta, Roxane; Marakos, Panagiotis; Pouli, Nicole; Kostakis, Ioannis K. Share Save
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