Not logged inHit-finding by Cysteine-Scanning (HCS): A method for finding druggable pockets
van Tienen, Laurens Moore; Bayoumi, Shadwa; Muneeruddin, Khaja; Leymarie, Nancy; Kornfilt, David; Bian, Yuemin; Kesar, Devishi; Li, Ruitong; Atack, Thomas; Popa, Alexandra-Mariela; Jandova, Zuzana; Trollmann, Philipp; Bergner, Andreas; Rumpel, Klaus; Kessler, Dirk; Sellers, William R.
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SaveDiscovery of potent and selective HER2 inhibitors with efficacy against HER2 exon 20 insertion-driven tumors, which preserve wild-type EGFR signaling
Wilding, Birgit; Scharn, Dirk; Boese, Dietrich; Baum, Anke; Santoro, Valeria; Chetta, Paolo; Schnitzer, Renate; Botesteanu, Dana A.; Reiser, Christoph; Kornigg, Stefan; Knesl, Petr; Hoermann, Alexandra; Koeferle, Anna; Corcokovic, Maja; Lieb, Simone; Scholz, Guido; Bruchhaus, Jens; Spina, Markus; Balla, Josef; Peric-Simov, Biljana; Zimmer, Jasmin; Mitzner, Sophie; Fett, Thomas N.; Beran, Alexandra; Lamarre, Lyne; Gerstberger, Thomas; Gerlach, Daniel; Bauer, Markus; Bergner, Andreas; Schlattl, Andreas; Bader, Gerd; Treu, Matthias; Engelhardt, Harald; Zahn, Stephan; Fuchs, Julian E.; Zuber, Johannes; Ettmayer, Peter; Pearson, Mark; Petronczki, Mark; Kraut, Norbert; McConnell, Darryl B.; Solca, Flavio; Neumuller, Ralph A.
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SaveGetting a Grip on the Undrugged: Targeting β-Catenin with Fragment-Based Methods
Kessler, Dirk; Mayer, Moriz; Zahn, Stephan K.; Zeeb, Markus; Woehrle, Simon; Bergner, Andreas; Bruchhaus, Jens; Ciftci, Tuncay; Dahmann, Georg; Dettling, Maike; Doebel, Sandra; Fuchs, Julian E.; Geist, Leonhard; Hela, Wolfgang; Kofink, Christiane; Kousek, Roland; Moser, Franziska; Puchner, Teresa; Rumpel, Klaus; Scharnweber, Maximilian; Werni, Patrick; Wolkerstorfer, Bernhard; Breitsprecher, Dennis; Baaske, Philipp; Pearson, Mark; McConnell, Darryl B.; Boettcher, Jark
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SaveStart Selective and Rigidify: The Discovery Path toward a Next Generation of EGFR Tyrosine Kinase Inhibitors
Engelhardt, Harald; Boese, Dietrich; Petronczki, Mark; Scharn, Dirk; Bader, Gerd; Baum, Anke; Bergner, Andreas; Chong, Eugene; Doebel, Sandra; Egger, Georg; Engelhardt, Christian; Ettmayer, Peter; Fuchs, Julian E.; Gerstberger, Thomas; Gonnella, Nina; Grimm, Andreas; Grondal, Elisabeth; Haddad, Nizar; Hopfgartner, Barbara; Kousek, Roland; Krawiec, Mariusz; Kriz, Monika; Lamarre, Lyne; Leung, Joyce; Mayer, Moriz; Patel, Nitinchandra D.; Simov, Biljana Peric; Reeves, Jonathan T.; Schnitzer, Renate; Schrenk, Andreas; Sharps, Bernadette; Solca, Flavio; Stadtmueller, Heinz; Tan, Zhulin; Wunberg, Tobias; Zoephel, Andreas; McConnell, Darryl B.
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SaveKRAS Binders Hidden in Nature
Bergner, Andreas; Cockcroft, Xiaoling; Fischer, Gerhard; Gollner, Andreas; Hela, Wolfgang; Kousek, Roland; Mantoulidis, Andreas; Martin, Laetitia J.; Mayer, Moriz; Muellauer, Barbara; Siszler, Gabriella; Wolkerstorfer, Bernhard; Kessler, Dirk; McConnell, Darryl B.
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