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J

Jérôme Amaudrut

irbm

10H-index
18Paper Count
1.1KCitation Count
Published Papers 10
Publication Date
An allosteric inhibitor of the Zika virus NS2B-NS3 protease with oral efficacy in mouse models
err2026-02-10
err0
errOAAI
errJesus M. Ontoria; Esther Torrente; Antonino Missineo; Cristina Alli; Rita Graziani; Silvia Conti; Monica Bisbocci; Antonio Quotadamo; Federica Ferrigno; Alessandra Corio; Giovanni Ievoli; Leda Bencheva; Jérôme Amaudrut; Silvana Vasile; Elisa Beghetto; Chantal Paolini; Nadine Alaimo; Maria Veneziano; Martina Nibbio; Maria V. Orsale; Giulia Proto; Fabrizio Colaceci; Laura Orsatti; Vincenzo Pucci; Romano Di Fabio; Licia Tomei; Christian Montalbetti; Alberto Bresciani; Carlo Toniatti; Giacomo Paonessa
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Viruses traverse the human proteome through peptide interfaces that can be biomimetically leveraged for drug discovery
err2024-01-22
err0
errOAAI
errSchickin, Laurene Meyniel; Amaudrut, Jerome; Mallinjoud, Pierre; Guillier, Fabrice; Mangeot, Philippe E.; Lines, Laetitia; Aublin-Gex, Anne; Scholtes, Caroline; Punginelli, Claire; Joly, Stephane; Vasseur, Florence; Manet, Evelyne; Gruffat, Henri; Henry, Thomas; Halitim, Fares; Paparin, Jean-Laurent; Machin, Peter; Darteil, Raphael; Sampson, Diane; Mikaelian, Ivan; Lane, Lydie; Navratil, Vincent; Golinelli-Coher, Marie-Pierre; Terzi, Fabiola; Andre, Patrice; Lotteau, Vincent; Vonderscher, Jacky; Meldrum, Eric C.; de Chassey, Benoit
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Discovery of a Novel Series of Potent SHP2 Allosteric Inhibitors
err2023-04-17
err6
errOAAI
errPetrocchi, Alessia; Grillo, Alessandro; Ferrante, Luca; Randazzo, Pietro; Prandi, Adolfo; De Matteo, Marilenia; Iaccarino, Costanza; Bisbocci, Monica; Cellucci, Antonella; Alli, Cristina; Nibbio, Martina; Pucci, Vincenzo; Amaudrut, Jerome; Montalbetti, Christian; Toniatti, Carlo; Di Fabio, Romano
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Discovery of a Novel Series of Imidazopyrazine Derivatives as Potent SHP2 Allosteric Inhibitors
err2023-01-10
err10
PREAI
errTorrente, Esther; Fodale, Valentina; Ciammaichella, Alina; Ferrigno, Federica; Ontoria, Jesus M.; Ponzi, Simona; Rossetti, Ilaria; Sferrazza, Alessio; Amaudrut, Jerome; Missineo, Antonino; Esposito, Simone; Palombo, Simone; Nibbio, Martina; Cerretani, Mauro; Bisbocci, Monica; Cellucci, Antonella; di Marco, Annalise; Alli, Cristina; Pucci, Vincenzo; Toniatti, Carlo; Petrocchi, Alessia
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SAR evolution towards potent C-terminal carboxamide peptide inhibitors of Zika virus NS2B-NS3 protease
err2022-03-01
err6
PREAI
errColarusso, Stefania; Ferrigno, Federica; Ponzi, Simona; Pavone, Francesca; Conte, Immacolata; Abate, Luigi; Beghetto, Elisa; Missineo, Antonino; Amaudrut, Jerome; Bresciani, Alberto; Paonessa, Giacomo; Tomei, Licia; Montalbetti, Christian; Bianchi, Elisabetta; Toniatti, Carlo; Ontoria, Jesus M. M.
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Design, Synthesis, and Evaluation of a Novel Series of Indole Sulfonamide Peroxisome Proliferator Activated Receptor (PPAR) α/γ/δ Triple Activators: Discovery of Lanifibranor, a New Antifibrotic Clinical Candidate
err2018-02-15
err98
PREAI
errBoubia, Benaissa; Poupardin, Olivia; Barth, Martine; Binet, Jean; Peralba, Philippe; Mounier, Laurent; Jacquier, Elise; Gauthier, Emilie; Lepais, Valerie; Chatar, Maryline; Ferry, Stephanie; Thourigny, Anne; Guillier, Fabrice; Llacer, Jonathan; Amaudrut, Jerome; Dodey, Pierre; Lacombe, Olivier; Masson, Philippe; Montalbetti, Christian; Wettstein, Guillaume; Luccarini, Jean-Michel; Legendre, Christiane; Junien, Jean-Louis; Broqua, Pierre
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Electron delocalization in the radical cation of 1,3,6,8-tetraazatricyclo[4.4.1.13,8]dodecane, a 4-nitrogen-7-electron system
err2001-12-13
err12
PREAI
errZwier, JM; Brouwer, AM; Keszthelyi, T; Balakrishnan, G; Offersgaard, JF; Wilbrandt, R; Barbosa, F; Buser, U; Amaudrut, J; Gescheidt, G; Nelsen, SF; Little, CD
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