Not logged in Viruses traverse the human proteome through peptide interfaces that can be biomimetically leveraged for drug discovery Schickin, Laurene Meyniel; Amaudrut, Jerome; Mallinjoud, Pierre; Guillier, Fabrice; Mangeot, Philippe E.; Lines, Laetitia; Aublin-Gex, Anne; Scholtes, Caroline; Punginelli, Claire; Joly, Stephane; Vasseur, Florence; Manet, Evelyne; Gruffat, Henri; Henry, Thomas; Halitim, Fares; Paparin, Jean-Laurent; Machin, Peter; Darteil, Raphael; Sampson, Diane; Mikaelian, Ivan; Lane, Lydie; Navratil, Vincent; Golinelli-Coher, Marie-Pierre; Terzi, Fabiola; Andre, Patrice; Lotteau, Vincent; Vonderscher, Jacky; Meldrum, Eric C.; de Chassey, Benoit Share Save
Discovery of a Novel Series of Potent SHP2 Allosteric Inhibitors Petrocchi, Alessia; Grillo, Alessandro; Ferrante, Luca; Randazzo, Pietro; Prandi, Adolfo; De Matteo, Marilenia; Iaccarino, Costanza; Bisbocci, Monica; Cellucci, Antonella; Alli, Cristina; Nibbio, Martina; Pucci, Vincenzo; Amaudrut, Jerome; Montalbetti, Christian; Toniatti, Carlo; Di Fabio, Romano Share Save
Discovery of a Novel Series of Imidazopyrazine Derivatives as Potent SHP2 Allosteric Inhibitors Torrente, Esther; Fodale, Valentina; Ciammaichella, Alina; Ferrigno, Federica; Ontoria, Jesus M.; Ponzi, Simona; Rossetti, Ilaria; Sferrazza, Alessio; Amaudrut, Jerome; Missineo, Antonino; Esposito, Simone; Palombo, Simone; Nibbio, Martina; Cerretani, Mauro; Bisbocci, Monica; Cellucci, Antonella; di Marco, Annalise; Alli, Cristina; Pucci, Vincenzo; Toniatti, Carlo; Petrocchi, Alessia Share Save
SAR evolution towards potent C-terminal carboxamide peptide inhibitors of Zika virus NS2B-NS3 protease Colarusso, Stefania; Ferrigno, Federica; Ponzi, Simona; Pavone, Francesca; Conte, Immacolata; Abate, Luigi; Beghetto, Elisa; Missineo, Antonino; Amaudrut, Jerome; Bresciani, Alberto; Paonessa, Giacomo; Tomei, Licia; Montalbetti, Christian; Bianchi, Elisabetta; Toniatti, Carlo; Ontoria, Jesus M. M. Share Save
Design, Synthesis, and Evaluation of a Novel Series of Indole Sulfonamide Peroxisome Proliferator Activated Receptor (PPAR) α/γ/δ Triple Activators: Discovery of Lanifibranor, a New Antifibrotic Clinical Candidate Boubia, Benaissa; Poupardin, Olivia; Barth, Martine; Binet, Jean; Peralba, Philippe; Mounier, Laurent; Jacquier, Elise; Gauthier, Emilie; Lepais, Valerie; Chatar, Maryline; Ferry, Stephanie; Thourigny, Anne; Guillier, Fabrice; Llacer, Jonathan; Amaudrut, Jerome; Dodey, Pierre; Lacombe, Olivier; Masson, Philippe; Montalbetti, Christian; Wettstein, Guillaume; Luccarini, Jean-Michel; Legendre, Christiane; Junien, Jean-Louis; Broqua, Pierre Share Save
Electron delocalization in the radical cation of 1,3,6,8-tetraazatricyclo[4.4.1.13,8]dodecane, a 4-nitrogen-7-electron system Zwier, JM; Brouwer, AM; Keszthelyi, T; Balakrishnan, G; Offersgaard, JF; Wilbrandt, R; Barbosa, F; Buser, U; Amaudrut, J; Gescheidt, G; Nelsen, SF; Little, CD Share Save
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