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Allosteric Covalent Inhibitors of the STAT3 Transcription Factor from Virtual Screening Szalai, TV; di Lorenzo, V; Péczka, N; Mihalovits, LM; Petri, L; Ashraf, QF; de Araujo, ED; Honti, V; Bajusz, D; Keseru, GM Share Save
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The PARP inhibitor rucaparib blocks SARS-CoV-2 virus binding to cells and the immune reaction in models of COVID-19 Papp, Henrietta; Toth, Emese; Bovari-Biri, Judit; Banfai, Krisztina; Juhasz, Peter; Mahdi, Mohamed; Russo, Lilian Cristina; Bajusz, David; Sipos, Adrienn; Petri, Laszlo; Szalai, Tibor Viktor; Kemeny, Agnes; Madai, Monika; Kuczmog, Anett; Batta, Gyula; Mozner, Orsolya; Vasko, Dorottya; Hirsch, Edit; Bohus, Peter; Mehes, Gabor; Tozser, Jozsef; Curtin, Nicola J.; Helyes, Zsuzsanna; Toth, Attila; Hoch, Nicolas C.; Jakab, Ferenc; Keseru, Gyorgy M.; Pongracz, Judit E.; Bai, Peter Share Save
Site-Selective Antibody Conjugation with Dibromopyrazines Szepesi Kovacs, Denes; Pasztor, Bettina; Abranyi-Balogh, Peter; Petri, Laszlo; Imre, Timea; Simon, Jozsef; Tatrai, Eniko; Varady, Gyorgy; Tovari, Jozsef; Szijj, Peter A.; Keseru, Gyorgy M. Share Save
Mapping protein binding sites by photoreactive fragment pharmacophores Abranyi-Balogh, Peter; Bajusz, David; Orgovan, Zoltan; Keeley, Aaron B.; Petri, Laszlo; Peczka, Nikolett; Szalai, Tibor Viktor; Palfy, Gyula; Gadanecz, Marton; Grant, Emma K.; Imre, Timea; Takacs, Tamas; Randelovic, Ivan; Baranyi, Marcell; Marton, Andras; Schlosser, Gitta; Ashraf, Qirat F.; de Araujo, Elvin D.; Karancsi, Tamas; Buday, Laszlo; Tovari, Jozsef; Perczel, Andras; Bush, Jacob T.; Keseru, Gyoergy M. Share Save
Contribution of Noncovalent Recognition and Reactivity to the Optimization of Covalent Inhibitors: A Case Study on KRasG12C Peczka, Nikolett; Randelovic, Ivan; Orgovan, Zoltan; Csorba, Noemi; Egyed, Attila; Petri, Laszlo; Abranyi-Balogh, Peter; Gadanecz, Marton; Perczel, Andras; Tovari, Jozsef; Schlosser, Gitta; Takacs, Tamas; Mihalovits, Levente M.; Ferenczy, Gyorgy G.; Buday, Laszlo; Keseru, Gyorgy M. Share Save
Electrophilic MiniFrags Revealed Unprecedented Binding Sites for Covalent HDAC8 Inhibitors Keeley, Aaron B.; Kopranovic, Aleksandra; Di Lorenzo, Vincenzo; Abranyi-Balogh, Peter; Jaensch, Niklas; Lai, Linh N.; Petri, Laszlo; Orgovan, Zoltan; Poeloeske, Daniel; Orlova, Anna; Nemeth, Andras Gyoergy; Desczyk, Charlotte; Imre, Timea; Bajusz, David; Moriggl, Richard; Meyer-Almes, Franz-Josef; Keserue, Gyoergy M. Share Save
Activation-Free Sulfonyl Fluoride Probes for Fragment Screening Petri, Laszlo; Aabranyi-Balogh, Peter; Csorba, Noemi; Keeley, Aaron; Simon, Jozsef; Randelovic, Ivan; Tovari, Jozsef; Schlosser, Gitta; Szabo, Daniel; Drahos, Laszlo; Keseru, Gyoergy M. Share Save
Covalent fragment mapping of KRasG12C revealed novel chemotypes with in vivo potency Orgovan, Zoltan; Peczka, Nikolett; Petri, Laszlo; Abranyi-Balogh, Peter; Randelovic, Ivan; Toth, Szilard; Szakacs, Gergely; Nyiri, Kinga; Vertessy, Beata; Palfy, Gyula; Vida, Istvan; Perczel, Andras; Tovari, Jozsef; Keseru, Gyorgy M. Share Save
Covalent inhibitors of bacterial peptidoglycan biosynthesis enzyme MurA with chloroacetamide warhead Grabrijan, Katarina; Hrast, Martina; Proj, Matic; Dolsak, Ana; Zdovc, Irena; Imre, Timea; Petri, Laszlo; Abranyi-Balogh, Peter; Keseru, Gyorgy M.; Gobec, Stanislav Share Save
Next-Generation Heterocyclic Electrophiles as Small-Molecule Covalent MurA Inhibitors Abranyi-Balogh, Peter; Keeley, Aaron; Ferenczy, Gyorgy G.; Petri, Laszlo; Imre, Timea; Grabrijan, Katarina; Hrast, Martina; Knez, Damijan; Ilas, Janez; Gobec, Stanislav; Keseru, Gyorgy M. Share Save
Semisynthetic teicoplanin derivatives with dual antimicrobial activity against SARS-CoV-2 and multiresistant bacteria Bereczki, Ilona; Vimberg, Vladimir; Lorincz, Eszter; Papp, Henrietta; Nagy, Lajos; Keki, Sandor; Batta, Gyula; Mitrovic, Ana; Kos, Janko; Zsigmond, Aron; Hajdu, Istvan; Lorincz, Zsolt; Bajusz, David; Petri, Laszlo; Hodek, Jan; Jakab, Ferenc; Keseru, Gyorgy M.; Weber, Jan; Naesens, Lieve; Herczegh, Pal; Borbas, Aniko Share Save
A covalent strategy to target intrinsically disordered proteins: Discovery of novel tau aggregation inhibitors Petri, Laszlo; Abranyi-Balogh, Peter; Vagrys, Darius; Imre, Timea; Varro, Nikolett; Mandity, Istvan; Racz, Anita; Wittner, Lucia; Toth, Kinga; Toth, Estilla Zsofia; Juhasz, Tunde; Davis, Ben; Keseru, Gyoergy Miklos Share Save
Fragment-Sized and Bidentate (Immuno)Proteasome Inhibitors Derived from Cysteine and Threonine Targeting Warheads Kollar, Levente; Gobec, Martina; Proj, Matic; Smrdel, Lara; Knez, Damijan; Imre, Timea; Gomory, Agnes; Petri, Laszlo; Abranyi-Balogh, Peter; Csanyi, Dorottya; Ferenczy, Gyoergy G.; Gobec, Stanislav; Sosic, Izidor; Keseru, Gyoergy M. Share Save
Discovery of selective fragment-sized immunoproteasome inhibitors Kollar, Levente; Gobec, Martina; Szilagyi, Bence; Proj, Matic; Knez, Damijan; Abranyi-Balogh, Peter; Petri, Laszlo; Imre, Timea; Bajusz, David; Ferenczy, Gyorgy G.; Gobec, Stanislav; Keseru, Gyorgy M.; Sosic, Izidor Share Save
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