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SaveCLIPSing Melanotan-II to Discover Multiple Functionally Selective hMCR Agonists
Tomassi, Stefano; Dimmito, Marilisa Pia; Cai, Minying; D'Aniello, Antonia; Del Bene, Alessandra; Messere, Anna; Liu, Zekun; Zhu, Tingyi; Hruby, Victor J.; Stefanucci, Azzurra; Cosconati, Sandro; Mollica, Adriano; Di Maro, Salvatore
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SaveAntagonism of the mu-delta opioid receptor heterodimer enhances opioid antinociception by activating Src and calcium/calmodulin-dependent protein kinase II signaling
Keresztes, Attila; Olson, Keith; Nguyen, Paul; Lopez-Pier, Marissa A.; Hecksel, Ryan; Barker, Natalie K.; Liu, Zekun; Hruby, Victor; Konhilas, John; Langlais, Paul R.; Streicher, John M.
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SaveMultifunctional Enkephalin Analogs with a New Biological Profile: MOR/DOR Agonism and KOR Antagonism
Lee, Yeon Sun; Remesic, Michael; Ramos-Colon, Cyf; Wu, Zhijun; LaVigne, Justin; Molnar, Gabriella; Tymecka, Dagmara; Misicka, Aleksandra; Streicher, John M.; Hruby, Victor J.; Porreca, Frank
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SaveMultiple Applications of a Novel Biarsenical Imaging Probe in Fluorescence and PET Imaging of Melanoma
Kondrashov, Mikhail; Svensson, Samuel P. S.; Strom, Peter; Westermark, Andreas; Jacobson-Ingemyr, Hanna; Takano, Akihiro; Tari, Lenke; Toth, Miklos; Cai, Minying; Hruby, Victor J.; Schou, Magnus
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SaveDevelopment of Macrocyclic Peptidomimetics Containing Constrained α,α-Dialkylated Amino Acids with Potent and Selective Activity at Human Melanocortin Receptors
Merlino, Francesco; Zhou, Yang; Cai, Minying; Carotenuto, Alfonso; Yousif, Ali M.; Brancaccio, Diego; Di Maro, Salvatore; Zappavigna, Silvia; Limatola, Antonio; Novellino, Ettore; Grieco, Paolo; Hruby, Victor J.
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SaveDevelopment of Novel Melanocortin Receptor Agonists Based on the Cyclic Peptide Framework of Sunflower Trypsin Inhibitor-1
Durek, Thomas; Cromm, Philipp M.; White, Andrew M.; Schroeder, Christina I.; Kaas, Quentin; Weidmann, Joachim; Fuaad, Abdullah Ahmad; Cheneval, Olivier; Harvey, Peta J.; Daly, Norelle L.; Zhou, Yang; Dellsen, Anita; Osterlund, Torben; Larsson, Niklas; Knerr, Laurent; Bauer, Udo; Kessler, Horst; Cai, Minying; Hruby, Victor J.; Plowright, Alleyn T.; Craik, David J.
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SaveDynamics of Membrane Proteins Studied by Solid State 2H NMR Relaxation
Xu, Xiaolin; Struts, Andrey V.; Giri, Aswini Kumar; Molugu, Trivikram R.; Guruge, Charitha; Faylough, Samira; Nascimento, Carolina L.; Nesnas, Nasri; Hruby, Victor J.; Brown, Michael F.
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SaveMelanocortin 1 Receptor Signaling Regulates Cholesterol Transport in Macrophages
Rinne, Petteri; Rami, Martina; Nuutinen, Salla; Santovito, Donato; van der Vorst, Emiel P. C.; Guillamat-Prats, Raquel; Lyytikainen, Leo-Pekka; Raitoharju, Emma; Oksala, Niku; Ring, Larisa; Cai, Minying; Hruby, Victor J.; Lehtimaki, Terho; Weber, Christian; Steffens, Sabine
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