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Deciphering the RNA recognition by Musashi-1 to design protein and RNA variants for in vitro and in vivo applications Perez-Rafols, Anna; Perez-Ropero, Guillermo; Cerofolini, Linda; Sperotto, Luca; Roca-Martinez, Joel; Higuera-Rodriguez, R. Anahi; Russomanno, Pasquale; Kaiser, Wolfgang; Vranken, Wim; Danielson, U. Helena; Provenzani, Alessandro; Martelli, Tommaso; Sattler, Michael; Buijs, Jos; Fragai, Marco Share Save
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The Role of Water Networks in Phosphodiesterase Inhibitor Dissociation and Kinetic Selectivity Blaazer, Antoni R.; Singh, Abhimanyu K.; Zara, Lorena; Boronat, Pierre; Bautista, Lady J.; Irving, Steve; Majewski, Maciej; Barril, Xavier; Wijtmans, Maikel; Danielson, U. Helena; Sterk, Geert Jan; Leurs, Rob; van Muijlwijk-Koezen, Jacqueline E.; Brown, David G.; de Esch, Iwan J. P. Share Save
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Discovery of the 4-aminopiperidine-based compound EM127 for the site-specific covalent inhibition of SMYD3 Parenti, Marco Daniele; Naldi, Marina; Manoni, Elisabetta; Fabini, Edoardo; Cederfelt, Daniela; Talibov, Vladimir O.; Gressani, Valeria; Guven, Ummu; Grossi, Valentina; Fasano, Candida; Sanese, Paola; De Marco, Katia; Shtil, Alexander A.; V. Kurkin, Alexander; Altieri, Andrea; Danielson, U. Helena; Caretti, Giuseppina; Simone, Cristiano; Varchi, Greta; Bartolini, Manuela; Del Rio, Alberto Share Save
Monitoring drug-target interactions through target engagement-mediated amplification on arrays and in situ Al-Amin, Rasel A.; Johansson, Lars; Abdurakhmanov, Eldar; Landegren, Nils; Lof, Liza; Arngarden, Linda; Blokzijl, Andries; Svensson, Richard; Hammond, Maria; Lonn, Peter; Haybaeck, Johannes; Kamali-Moghaddam, Masood; Jensen, Annika Jenmalm; Danielson, U. Helena; Artursson, Per; Lundback, Thomas; Landegren, Ulf Share Save
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Ultralarge Virtual Screening Identifies SARS-CoV-2 Main Protease Inhibitors with Broad-Spectrum Activity against Coronaviruses Luttens, Andreas; Gullberg, Hjalmar; Abdurakhmanov, Eldar; Duy Duc Vo; Akaberi, Dario; Talibov, Vladimir O.; Nekhotiaeva, Natalia; Vangeel, Laura; De Jonghe, Steven; Jochmans, Dirk; Krambrich, Janina; Tas, Ali; Lundgren, Bo; Gravenfors, Ylva; Craig, Alexander J.; Atilaw, Yoseph; Sandstrom, Anja; Moodie, Lindon W. K.; Lundkvist, Ake; van Hemert, Martijn J.; Neyts, Johan; Lennerstrand, Johan; Kihlberg, Jan; Sandberg, Kristian; Danielson, U. Helena; Carlsson, Jens Share Save
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A real-time cell-binding assay reveals dynamic features of STxB-Gb3 cointernalization and STxB-mediated cargo delivery into cancer cells Encarnacao, Joao; Napolitano, Valeria; Opassi, Giulia; Danielson, U. Helena; Dubin, Grzegorz; Popowicz, Grzegorz M.; Munier-Lehmann, Helene; Buijs, Jos; Andersson, Karl; Bjorkelund, Hanna Share Save
Macrocyclic Peptides Uncover a Novel Binding Mode for Reversible Inhibitors of LSD1 Yang, Jie; Talibov, Vladimir O.; Peintner, Stefan; Rhee, Claire; Poongavanam, Vasanthanathan; Geitmann, Matthis; Sebastiano, Matteo Rossi; Simon, Bernd; Hennig, Janosch; Dobritzsch, Doreen; Danielson, U. Helena; Kihlberg, Jan Share Save
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Noelin1 Affects Lateral Mobility of Synaptic AMPA Receptors Pandya, Nikhil J.; Seeger, Christian; Babai, Norbert; Gonzalez-Lozano, Miguel A.; Mack, Volker; Lodder, Johannes C.; Gouwenberg, Yvonne; Mansvelder, Huibert D.; Danielson, U. Helena; Li, Ka Wan; Heine, Martin; Spijker, Sabine; Frischknecht, Renato; Smit, August B. Share Save
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