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SaveIn vitro and in vivo evaluation of Bombesin-MMAE conjugates for targeted tumour therapy
Gomena, Jacopo; Modena, Daniela; Cordella, Paola; Vari, Balazs; Randelovic, Ivan; Borbely, Adina; Bottani, Michela; Vari-Mezo, Diana; Halmos, Gabor; Juhasz, Eva; Steinkuhler, Christian; Tovari, Jozsef; Mezo, Gabor
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SaveMapping protein binding sites by photoreactive fragment pharmacophores
Abranyi-Balogh, Peter; Bajusz, David; Orgovan, Zoltan; Keeley, Aaron B.; Petri, Laszlo; Peczka, Nikolett; Szalai, Tibor Viktor; Palfy, Gyula; Gadanecz, Marton; Grant, Emma K.; Imre, Timea; Takacs, Tamas; Randelovic, Ivan; Baranyi, Marcell; Marton, Andras; Schlosser, Gitta; Ashraf, Qirat F.; de Araujo, Elvin D.; Karancsi, Tamas; Buday, Laszlo; Tovari, Jozsef; Perczel, Andras; Bush, Jacob T.; Keseru, Gyoergy M.
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SaveContribution of Noncovalent Recognition and Reactivity to the Optimization of Covalent Inhibitors: A Case Study on KRasG12C
Peczka, Nikolett; Randelovic, Ivan; Orgovan, Zoltan; Csorba, Noemi; Egyed, Attila; Petri, Laszlo; Abranyi-Balogh, Peter; Gadanecz, Marton; Perczel, Andras; Tovari, Jozsef; Schlosser, Gitta; Takacs, Tamas; Mihalovits, Levente M.; Ferenczy, Gyorgy G.; Buday, Laszlo; Keseru, Gyorgy M.
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SaveFarnesyl-transferase inhibitors show synergistic anticancer effects in combination with novel KRAS-G12C inhibitors
Baranyi, Marcell; Molnar, Eszter; Hegedus, Luca; Gabriel, Zsofia; Petenyi, Flora Greta; Bordas, Fanni; Lener, Violetta; Randelovic, Ivan; Cserepes, Mihaly; Tovari, Jozsef; Hegedus, Balazs; Timar, Jozsef
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SaveActivation-Free Sulfonyl Fluoride Probes for Fragment Screening
Petri, Laszlo; Aabranyi-Balogh, Peter; Csorba, Noemi; Keeley, Aaron; Simon, Jozsef; Randelovic, Ivan; Tovari, Jozsef; Schlosser, Gitta; Szabo, Daniel; Drahos, Laszlo; Keseru, Gyoergy M.
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SaveCovalent fragment mapping of KRasG12C revealed novel chemotypes with in vivo potency
Orgovan, Zoltan; Peczka, Nikolett; Petri, Laszlo; Abranyi-Balogh, Peter; Randelovic, Ivan; Toth, Szilard; Szakacs, Gergely; Nyiri, Kinga; Vertessy, Beata; Palfy, Gyula; Vida, Istvan; Perczel, Andras; Tovari, Jozsef; Keseru, Gyorgy M.
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SaveSREKA-targeted liposomes for highly metastatic breast cancer therapy
Vari, Balazs; Dokus, Levente; Borbely, Adina; Gaal, Aniko; Vari-Mezo, Diana; Randelovic, Ivan; Solyom-Tisza, Anna; Varga, Zoltan; Szoboszlai, Norbert; Mezo, Gabor; Tovari, Jozsef
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SaveCorrelations of genetic variation R521K of EGF receptor and the in vitro, in vivo and clinical phenotypes of head and neck cancers after cetuximab treatment
Cserepes, Mihaly T.; Hegedus, Zita; Randelovic, Ivan; Kenessey, Istvan; Meilinger-Dobra, Monika; Csiko, Kristof G.; Ladanyi, Andrea; Remenar, Eva; Tovari, Jozsef
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SaveSequence modification of heptapeptide selected by phage display as homing device for HT-29 colon cancer cells to improve the anti-tumour activity of drug delivery systems
Kiss, Krisztina; Biri-Kovacs, Beata; Szabo, Rita; Randelovic, Ivan; Enyedi, Kata Nora; Schlosser, Gitta; Orosz, Adam; Kapuvari, Bence; Tovari, Jozsef; Mezo, Gabor
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SaveAnticancer Potential of (Pentamethylcyclopentadienyl)chloridoiridium(III) Complexes Bearing κP and κP,κS-Coordinated Ph2PCH2CH2CH2S(O)xPh (x=0-2) Ligands
Ludwig, Gerd; Randelovic, Ivan; Maksimovic-Ivanic, Danijela; Mijatovic, Sanja; Bulatovic, Mirna Z.; Miljkovic, Djordje; Korb, Marcus; Lang, Heinrich; Steinborn, Dirk; Kaluderovic, Goran N.
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