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György M. Keserű

Research Centre for Natural Sciences

50H-index
415Paper Count
1.3WCitation Count
Published Papers 180
Publication Date
Probing 3-Amino-2H-Azaindazoles as Allosteric Inhibitors of the Protein Tyrosine Phosphatase SHP2
err2026-06-14
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errMachoud Amoussa; Nina-Louisa Efrém; Feng Li; Ziqiong Guo; Yvette Roske; Katrin Jana Frank; Szymon Pach; Clemens Alexander Wolf; Feng Bo; Marina Lesina; Mika Kintzel; Rana Alsalim; Victoria Zeitz; Noémi Csorba; Silke Radetzki; György M. Keserű; Oliver Daumke; Hana Algül; Gerhard Wolber; Jia Li; Marc Nazaré
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Fragment-Based Design of Targeted Covalent Inhibitors: The Scope and Limitation of Linking Approaches
err2026-05-22
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errLevente Kollár; Levente M. Mihalovits; Dávid Bajusz; Damijan Knez; József Simon; Blake H. Balcomb; Daren Fearon; Stanislav Gobec; György M. Keserű
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α-Halothioamide warheads with enhanced cysteine reactivity and specificity for covalent protein labelling
err2026-05-14
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errLászló Petri; Ronen Gabizon; Nikolett Péczka; Péter Ábrányi-Balogh; József Simon; Tímea Imre; György G. Ferenczy; Nir London; György M. Keserű
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Merging Micellar Catalysis and C-H Activation: Silver-Free Direct Arylation of Fluoroarenes in Water
err2026-05-14
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errBelnome, Federico; Garami, Kristof N.; Varga, Zoltan; Mihaly, Judith; Hauk, Pascal; Hergert, Tamas; Keseru, Gyorgy M.; Gallou, Fabrice; Wencel-Delord, Joanna; Abranyi-Balogh, Peter
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Mapping the SHP2 Allosteric Pocket With Target-Biased Covalent Fragments
err2026-04-24
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errNina-Louisa Efrém; Noémi Csorba; Machoud Amoussa; Péter Ábrányi-Balogh; Ziqiong Guo; László Petri; Feng Bo; Vincenzo Di Lorenzo; Yvette Roske; Tibor Viktor Szalai; Levente Mihalovits; József Simon; Jia Li; Oliver Daumke; György M. Keserű; Marc Nazaré
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Efficiency landscape of bioorthogonal click reactions producing bispecific antibody conjugates
err2026-04-21
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errLászló Petri; Írisz K. Kovács; Boglárka Szabó; Tímea Imre; Anita Rácz; Vijay Chudasama; Peter A. Szijj; György M. Keserű
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Benchmarking pKa Prediction Algorithms against an Extensive; Public Data Set
err2026-04-05
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errLevente Sipos-Szabó; Dávid Bajusz; György T. Balogh; György M. Keserű
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The Discovery of RGH-706; a Highly Efficacious MCH1 Receptor Antagonist; for the Treatment of Obesity and Insatiable Hunger
err2026-01-22
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errGyula Beke; András Boros; György M. Keserű; Balázs Krámos; Krisztina Katalin Szalai; Anikó Gere; Mónika Vastag; Márta Thán; Balázs Varga; Ottilia Balázs; Sándor Farkas; Balázs Lendvai; István Greiner; János Éles
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Covalent Activation of the C-type Lectin DC-SIGN
err2025-11-24
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errJonathan Lefèbre; Maurice Besch; Noémi Csorba; Kristóf Garami; Zoltán Orgován; Gitta Schlosser; Iris Bermejo; Péter Ábrányi-Balogh; György M. Keserű; Prof. Dr. Christoph Rademacher
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The impact of secondary site interactions on the binding specificity of bitopic dopamine D2/D3 receptor ligands
err2025-10-20
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errAttila Egyed; Dóra Judit Kiss; Zsófia Pável; Keve Rajna; Supriya A. Gaitonde; Mariam Dubiel; María Isabel Loza; Edina Szűcs; Éva Borbély; Zsófia Hajna; Grzegorz Satala; Márton Vass; Pál Szabó; Katalin Jósvay; Andrzej J. Bojarski; Holger Stark; Zsuzsanna Helyes; Erika Pintér; Michel Bouvier; György M. Keserű
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Versatile Palladium-Catalyzed C-H Arylation of Fluoroarenes with 2-Chloropyridine Derivatives
err2025-09-27
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errFederico Belnome; Péter P. Fehér; András Stirling; Csongor G. Németh; Tamás Hergert; György M. Keserű; Péter Ábrányi-Balogh
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Structure-Guided Discovery of Nitrobenzo-2-Oxa-1,3-Diazole (NBD) Scaffold-based PFKFB4 Inhibitors for Cancer Therapy
err2025-08-28
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PREAI
errYiliang Chen; Shihong Wei; Qi Wang; Muhammad Salman Hameed; Jiawei Bao; Jufen Yan; György M. Keserű; Xinya Han
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Discovering Uncharted Binding Pockets on E3 Ligases Leads to the Identification of FBW7 Allosteric Modulators
err2025-08-20
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errMíriam Martínez-Cartró; Álvaro Serrano-Morrás; Andrea Bertran-Mostazo; Roger Castaño-Muñiz; Salvatore Scaffidi; Varbina Ivanova; Noémi Csorba; József Simon; Péter Ábrányi-Balogh; Yunfeng Li; György M. Keserü; Bing Hao; Xavier Barril; Carles Galdeano
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Covalent ligand efficiency
err2025-08-13
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errGyörgy G. Ferenczy; György M. Keserű
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The changing landscape of medicinal chemistry optimization
err2025-07-07
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PREAI
errAnita Rácz; Levente M. Mihalovits; Maximilian Beckers; Nikolas Fechner; Nikolaus Stiefl; Finton Sirockin; William McCoull; Emma Evertsson; Malin Lemurell; Gergely Makara; György M. Keserű
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Ultrahigh-Throughput Virtual Screening Strategies against PPI Targets: A Case Study of STAT Inhibitors
err2025-07-04
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errTibor Viktor Szalai; Nikolett Péczka; Levente Sipos-Szabó; László Petri; Dávid Bajusz; György M. Keserű
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Fluorescent tools for imaging class A G-protein coupled receptors
err2025-06-01
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errSzabo, Renata; Hornyanszky, Agnes; Kiss, Dora Judit; Keseru, Gyorgy Miklos
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Allosteric Covalent Inhibitors of the STAT3 Transcription Factor from Virtual Screening
err2025-05-06
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errSzalai, TV; di Lorenzo, V; Péczka, N; Mihalovits, LM; Petri, L; Ashraf, QF; de Araujo, ED; Honti, V; Bajusz, D; Keseru, GM
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