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In Vivo-Active Soluble Epoxide Hydrolase-Targeting PROTACs with Improved Potency and Stability Nakane, Keita; Morisseau, Christophe; Dowker-Key, Presley D.; Benitez, Gabrielle; Aguilan, Jennifer T.; Nagai, Emiko; Sidoli, Simone; Hammock, Bruce D.; Bettaieb, Ahmed; Shinoda, Kosaku; Kitamura, Seiya Share Save
Ultrapotent influenza hemagglutinin fusion inhibitors developed through SuFEx- enabled highthroughput medicinal chemistry Kitamura, Seiya; Lin, Ting Hui; Lee, Chang Chun David; Takamura, Akihiro; Kadam, Rameshwar U.; Zhang, Ding; Zhu, Xueyong; Dada, Lucas; Nagai, Emiko; Yu, Wenli; Yao, Yao; Sharpless, K. Barry; Wilson, Ian A.; Wolan, Dennis W. Share Save
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PROTAC-Mediated Selective Degradation of Cytosolic Soluble Epoxide Hydrolase Enhances ER Stress Reduction Wang, Yuxin; Morisseau, Christophe; Takamura, Akihiro; Wan, Debin; Li, Dongyang; Sidoli, Simone; Yang, Jun; Wolan, Dennis W.; Hammock, Bruce D.; Kitamura, Seiya Share Save
Diversity oriented clicking delivers ?-substituted alkenyl sulfonyl fluorides as covalent human neutrophil elastase inhibitors br Cheng, Yunfei; Li, Gencheng; Smedley, Christopher J.; Giel, Marie -Claire; Kitamura, Seiya; Woehl, Jordan L.; Bianco, Giulia; Forli, Stefano; Homer, Joshua A.; Cappiello, John R.; Wolan, Dennis W.; Moses, John E.; Sharpless, K. Barry Share Save
The Development of the Bengamides as New Antibiotics against Drug-Resistant Bacteria Porras-Alcala, Cristina; Moya-Utrera, Federico; Garcia-Castro, Miguel; Sanchez-Ruiz, Antonio; Lopez-Romero, Juan Manuel; Pino-Gonzalez, Maria Soledad; Diaz-Morilla, Amelia; Kitamura, Seiya; Wolan, Dennis W.; Prados, Jose; Melguizo, Consolacion; Cheng-Sanchez, Ivan; Sarabia, Francisco Share Save
Metabolomics activity screening of T cell-induced colitis reveals anti-inflammatory metabolites Montenegro-Burke, J. Rafael; Kok, Bernard P.; Guijas, Carlos; Domingo-Almenara, Xavier; Moon, Clara; Galmozzi, Andrea; Kitamura, Seiya; Eckmann, Lars; Saez, Enrique; Siuzdak, Gary E.; Wolan, Dennis W. Share Save
Chemical Inhibition of ENL/AF9 YEATS Domains in Acute Leukemia Garnar-Wortzel, Leopold; Bishop, Timothy R.; Kitamura, Seiya; Milosevich, Natalia; Asiaban, Joshua N.; Zhang, Xiaoyu; Zheng, Qinheng; Chen, Emily; Ramos, Anissa R.; Ackerman, Christopher J.; Hampton, Eric N.; Chatterjee, Arnab K.; Young, Travis S.; Hull, Mitchell, V; Sharpless, K. Barry; Cravatt, Benjamin F.; Wolan, Dennis W.; Erb, Michael A. Share Save
Synthetic Elaboration of Native DNA by RASS (SENDR) (vol 6, pg 1789, 2020) Flood, Dillon T.; Knouse, Kyle W.; Vantourout, Julien C.; Kitamura, Seiya; Sanchez, Brittany B.; Sturgell, Emily J.; Chen, Jason S.; Wolan, Dennis W.; Baran, Phil S.; Dawson, Philip E. Share Save
Synthetic Elaboration of Native DNA by RASS (SENDR) Flood, Dillon T.; Knouse, Kyle W.; Vantourout, Julien C.; Kitamura, Seiya; Sanchez, Brittany B.; Sturgell, Emily J.; Chen, Jason S.; Wolan, Dennis W.; Baran, Phil S.; Dawson, Philip E. Share Save
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Discovery of small-molecule enzyme activators by activity-based protein profiling Kok, Bernard P.; Ghimire, Srijana; Kim, Woojoo; Chatterjee, Shreyosree; Johns, Tyler; Kitamura, Seiya; Eberhardt, Jerome; Ogasawara, Daisuke; Xu, Janice; Sukiasyan, Ara; Kim, Sean M.; Godio, Cristina; Bittencourt, Julia M.; Cameron, Michael; Galmozzi, Andrea; Forli, Stefano; Wolan, Dennis W.; Cravatt, Benjamin F.; Boger, Dale L.; Saez, Enrique Share Save
Sulfur(VI) Fluoride Exchange (SuFEx)-Enabled High-Throughput Medicinal Chemistry Kitamura, Seiya; Zheng, Qinheng; Woehl, Jordan L.; Solania, Angelo; Chen, Emily; Dillon, Nicholas; Hull, Mitchell, V; Kotaniguchi, Miyako; Cappiello, John R.; Kitamura, Shinichi; Nizet, Victor; Sharpless, K. Barry; Wolan, Dennis W. Share Save
SuFEx-enabled, agnostic discovery of covalent inhibitors of human neutrophil elastase Zheng, Qinheng; Woehl, Jordan L.; Kitamura, Seiya; Santos-Martins, Diogo; Smedley, Christopher J.; Li, Gencheng; Forli, Stefano; Moses, John E.; Wolan, Dennis W.; Sharpless, K. Barry Share Save