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Seiya Kitamura

albert einstein college of medicine

18H-index
76Paper Count
1.3KCitation Count
Published Papers 24
Publication Date
CDK9 inhibition sensitizes intrinsically resistant BRAF V600E mutant colorectal cancer to BRAF inhibitors
err2026-05-18
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errOAAI
errNing Wei; Natalie Thielen; Mahshid Mohammadi; Muzaffer Ahmed Bhat; Terence Li; Yan Sun; Seiya Kitamura; Edward Chu; Chaoyuan Kuang
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High-throughput screening identifies NT-1 that synergizes with MRTX1133 against acquired resistant KRASG12D colorectal cancer
err2026-04-08
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errOAAI
errNatalie Thielen; Ning Wei; Emiko Nagai; Michele Houston; Leonard H. Augenlicht; Alice E. Shin; Joel T. Gabre; Anil K. Rustgi; Grace Ha; Lindsay M. LaFave; Edward Chu; Seiya Kitamura; Chaoyuan Kuang
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Novel Taxol-Derivative, STO-1, Induces Selective Anti-Tumor Immunity and Sustained Remission of Glioblastoma Without Triggering Autoimmune Reactions
err2025-10-30
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errOAAI
errShubhasmita Mohapatra; Adrian Guerrero; Neha Rahman; Khondoker Takia Zaman; Jing Wu; Callistus Onyeagba; Chanyue Hu; Matteo Pellegrini; Jayaram Vankudoth; Seiya Kitamura; Lauren O’Donnell; Youssef Zaim Wadghiri; Probal Banerjee
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Diversity oriented clicking for modular synthesis
err2025-08-07
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PREAI
errZifei Wang; Joshua A. Homer; Elias K. Zegeye; Lucas Dada; Dennis W. Wolan; Seiya Kitamura; John E. Moses
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SuFEx-enabled high-throughput medicinal chemistry for developing potent tamoxifen analogs as Ebola virus entry inhibitors
err2025-04-28
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errOAAI
errDada, Lucas; Nagai, Emiko; Agrawal, Sashank; Wirchnianski, Ariel S.; Wilson, Ian A.; Chandran, Kartik; Kitamura, Seiya
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In Vivo-Active Soluble Epoxide Hydrolase-Targeting PROTACs with Improved Potency and Stability
err2024-10-03
err0
PREAI
errNakane, Keita; Morisseau, Christophe; Dowker-Key, Presley D.; Benitez, Gabrielle; Aguilan, Jennifer T.; Nagai, Emiko; Sidoli, Simone; Hammock, Bruce D.; Bettaieb, Ahmed; Shinoda, Kosaku; Kitamura, Seiya
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Ultrapotent influenza hemagglutinin fusion inhibitors developed through SuFEx- enabled highthroughput medicinal chemistry
err2024-05-16
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PREAI
errKitamura, Seiya; Lin, Ting Hui; Lee, Chang Chun David; Takamura, Akihiro; Kadam, Rameshwar U.; Zhang, Ding; Zhu, Xueyong; Dada, Lucas; Nagai, Emiko; Yu, Wenli; Yao, Yao; Sharpless, K. Barry; Wilson, Ian A.; Wolan, Dennis W.
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SuFEx-based chemical diversification for the systematic discovery of CRBN molecular glues
err2024-04-01
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errOAAI
errCarter, Trever R.; Milosevich, Natalia; Dada, Lucas; Shaum, James B.; Sharpless, K. Barry; Kitamura, Seiya; Erb, Michael A.
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PROTAC-Mediated Selective Degradation of Cytosolic Soluble Epoxide Hydrolase Enhances ER Stress Reduction
err2023-03-22
err3
errOAAI
errWang, Yuxin; Morisseau, Christophe; Takamura, Akihiro; Wan, Debin; Li, Dongyang; Sidoli, Simone; Yang, Jun; Wolan, Dennis W.; Hammock, Bruce D.; Kitamura, Seiya
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Diversity oriented clicking delivers ?-substituted alkenyl sulfonyl fluorides as covalent human neutrophil elastase inhibitors br
err2022-09-07
err22
errOAAI
errCheng, Yunfei; Li, Gencheng; Smedley, Christopher J.; Giel, Marie -Claire; Kitamura, Seiya; Woehl, Jordan L.; Bianco, Giulia; Forli, Stefano; Homer, Joshua A.; Cappiello, John R.; Wolan, Dennis W.; Moses, John E.; Sharpless, K. Barry
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The Development of the Bengamides as New Antibiotics against Drug-Resistant Bacteria
err2022-05-31
err8
errOAAI
errPorras-Alcala, Cristina; Moya-Utrera, Federico; Garcia-Castro, Miguel; Sanchez-Ruiz, Antonio; Lopez-Romero, Juan Manuel; Pino-Gonzalez, Maria Soledad; Diaz-Morilla, Amelia; Kitamura, Seiya; Wolan, Dennis W.; Prados, Jose; Melguizo, Consolacion; Cheng-Sanchez, Ivan; Sarabia, Francisco
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Metabolomics activity screening of T cell-induced colitis reveals anti-inflammatory metabolites
err2021-09-28
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errOAAI
errMontenegro-Burke, J. Rafael; Kok, Bernard P.; Guijas, Carlos; Domingo-Almenara, Xavier; Moon, Clara; Galmozzi, Andrea; Kitamura, Seiya; Eckmann, Lars; Saez, Enrique; Siuzdak, Gary E.; Wolan, Dennis W.
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Chemical Inhibition of ENL/AF9 YEATS Domains in Acute Leukemia
err2021-04-30
err57
errOAAI
errGarnar-Wortzel, Leopold; Bishop, Timothy R.; Kitamura, Seiya; Milosevich, Natalia; Asiaban, Joshua N.; Zhang, Xiaoyu; Zheng, Qinheng; Chen, Emily; Ramos, Anissa R.; Ackerman, Christopher J.; Hampton, Eric N.; Chatterjee, Arnab K.; Young, Travis S.; Hull, Mitchell, V; Sharpless, K. Barry; Cravatt, Benjamin F.; Wolan, Dennis W.; Erb, Michael A.
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Synthetic Elaboration of Native DNA by RASS (SENDR) (vol 6, pg 1789, 2020)
err2020-10-23
err0
errOAAI
errFlood, Dillon T.; Knouse, Kyle W.; Vantourout, Julien C.; Kitamura, Seiya; Sanchez, Brittany B.; Sturgell, Emily J.; Chen, Jason S.; Wolan, Dennis W.; Baran, Phil S.; Dawson, Philip E.
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Synthetic Elaboration of Native DNA by RASS (SENDR)
err2020-10-05
err14
errOAAI
errFlood, Dillon T.; Knouse, Kyle W.; Vantourout, Julien C.; Kitamura, Seiya; Sanchez, Brittany B.; Sturgell, Emily J.; Chen, Jason S.; Wolan, Dennis W.; Baran, Phil S.; Dawson, Philip E.
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An influenza A hemagglutinin small-molecule fusion inhibitor identified by a new high-throughput fluorescence polarization screen
err2020-07-20
err34
errOAAI
errYao, Yao; Kadam, Rameshwar U.; Lee, Chang-Chun David; Woehl, Jordan L.; Wu, Nicholas C.; Zhu, Xueyong; Kitamura, Seiya; Wilson, Ian A.; Wolan, Dennis W.
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An Irreversible Inhibitor to Probe the Role of Streptococcus pyogenes Cysteine Protease SpeB in Evasion of Host Complement Defenses
err2020-07-14
err8
errOAAI
errWoehl, Jordan L.; Kitamura, Seiya; Dillon, Nicholas; Han, Zhen; Edgar, Landon J.; Nizet, Victor; Wolan, Dennis W.
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Discovery of small-molecule enzyme activators by activity-based protein profiling
err2020-06-08
err37
errOAAI
errKok, Bernard P.; Ghimire, Srijana; Kim, Woojoo; Chatterjee, Shreyosree; Johns, Tyler; Kitamura, Seiya; Eberhardt, Jerome; Ogasawara, Daisuke; Xu, Janice; Sukiasyan, Ara; Kim, Sean M.; Godio, Cristina; Bittencourt, Julia M.; Cameron, Michael; Galmozzi, Andrea; Forli, Stefano; Wolan, Dennis W.; Cravatt, Benjamin F.; Boger, Dale L.; Saez, Enrique
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Sulfur(VI) Fluoride Exchange (SuFEx)-Enabled High-Throughput Medicinal Chemistry
err2020-06-01
err110
errOAAI
errKitamura, Seiya; Zheng, Qinheng; Woehl, Jordan L.; Solania, Angelo; Chen, Emily; Dillon, Nicholas; Hull, Mitchell, V; Kotaniguchi, Miyako; Cappiello, John R.; Kitamura, Shinichi; Nizet, Victor; Sharpless, K. Barry; Wolan, Dennis W.
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SuFEx-enabled, agnostic discovery of covalent inhibitors of human neutrophil elastase
err2019-09-04
err142
errOAAI
errZheng, Qinheng; Woehl, Jordan L.; Kitamura, Seiya; Santos-Martins, Diogo; Smedley, Christopher J.; Li, Gencheng; Forli, Stefano; Moses, John E.; Wolan, Dennis W.; Sharpless, K. Barry
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