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收藏Identification of [1,2,4]Triazolo[4,3-a]pyrazine PARP1 inhibitors with overcome acquired resistance activities
Wang, Pingyuan; Zhu, Wen-Ting; Wang, Yajing; Song, Shan-Shan; Xi, Yong; Yang, Xin-Ying; Shen, Yan-Yan; Su, Yi; Sun, Yi-Ming; Gao, Ying-Lei; Chen, Yi; Ding, Jian; Miao, Ze-Hong; Zhang, Ao; He, Jin-Xue
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收藏YCH1899, a Highly Effective Phthalazin-1(2H)-one Derivative That Overcomes Resistance to Prior PARP Inhibitors
Sun, Yuting; Yang, Hui; Yuan, Jiaqi; Wang, Limin; Song, Shanshan; Chen, Rongrong; Bao, Xubin; Jia, Li; Yang, Tiantian; Zhang, Xiaofei; He, Qian; Gan, Yong; Miao, Zehong; He, Jinxue; Yang, Chunhao
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收藏Thioparib inhibits homologous recombination repair, activates the type I IFN response, and overcomes olaparib resistanceThioparib抑制同源重组修复,激活I型IFN反应,并克服olaparib抗性
Wang, Li-Min; Wang, Pingyuan; Chen, Xiao-Min; Yang, Hui; Song, Shan-Shan; Song, Zilan; Jia, Li; Chen, Hua-Dong; Bao, Xu-Bin; Guo, Ne; Huan, Xia-Juan; Xi, Yong; Shen, Yan-Yan; Yang, Xin-Ying; Su, Yi; Sun, Yi-Ming; Gao, Ying-Lei; Chen, Yi; Ding, Jian; Lang, Jing-Yu; Miao, Ze-Hong; Zhang, Ao; He, Jin-Xue
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收藏Design, synthesis and pharmacological evaluation of new PARP1 inhibitors by merging pharmacophores of olaparib and the natural product alantolactone
Kayumov, Muzaffar; Jia, Li; Pardaev, Azizbek; Song, Shan-Shan; Mirzaakhmedov, Sharafitdin; Ding, Chunyong; Cheng, Yong-Jun; Zhang, Ruihan (Isabella); Bao, Xubin; Miao, Ze-Hong; He, Jin-Xue; Zhang, Ao
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收藏SOMCL-19-133, a novel, selective, and orally available inhibitor of NEDD8-activating enzyme (NAE) for cancer therapy
Zhou, Li-Na; Xiong, Chaodong; Cheng, Yong-Jun; Song, Shan-Shan; Bao, Xu-Bin; Huan, Xia-Juan; Wang, Tong-Yan; Zhang, Ao; Miao, Ze-Hong; He, Jin-Xue
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收藏Design and development of a novel series of oral bivalent BET inhibitors with potent anticancer activities
Luo, Menglan; Wu, Qian; Yang, Yueyue; Sun, Lin; Huan, Xiajuan; Tian, Changqing; Xiong, Bing; Miao, Zehong; Wang, Yingqing; Chen, Danqi
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收藏Multi-omics characterization of WNT pathway reactivation to ameliorate BET inhibitor resistance in liver cancer cells
Liu, Yuwei; Xue, Mengzhu; Cao, Danyan; Qin, Lihuai; Wang, Ying; Miao, Zehong; Wang, Peng; Hu, Xin; Shen, Jingkang; Xiong, Bing
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收藏Development of Potent NEDD8-Activating Enzyme Inhibitors Bearing a Pyrimidotriazole Scaffold
Xiong, Chaodong; Zhou, Lina; Tan, Jing; Song, Shanshan; Bao, Xubin; Zhang, Ning; Ding, Huaqian; Zhao, Jiannan; He, Jin-Xue; Miao, Ze-Hong; Zhang, Ao
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收藏Discovery of MTR-106 as a highly potent G-quadruplex stabilizer for treating BRCA-deficient cancers
Li, Meng-Zhu; Meng, Tao; Song, Shan-Shan; Bao, Xu-Bin; Ma, Lan-Ping; Zhang, Ning; Yu, Ting; Zhang, Yong-Liang; Xiong, Bing; Shen, Jing-Kang; Miao, Ze-Hong; He, Jin-Xue
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