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收藏Design, synthesis and biological evaluation of novel TMPRSS2-PROTACs with florosubstituted 4-guanidino-N-phenylbenzamide derivative ligands
Yang, Hao; Xu, Haoran; Lin, Xinxin; Cai, Zengxuan; Xia, Yong; Wang, Yu; Chen, Zejie; Zhang, Koutian; Wu, Yanling; Wang, Jianwei; Awadasseid, Annoor; Zhang, Wen
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收藏Design, synthesis, and evaluation of antitumor activity of 2-arylmethox-y-4-(2-fluoromethyl-biphenyl-3-ylmethoxy) benzylamine derivatives as PD-1/PD-l1 inhibitors
Zhang, Feng; Zhang, Hua; Zhou, Shijia; Plewka, Jacek; Wang, Ming; Sun, Shishi; Wu, Caiyun; Yu, Qimeng; Zhu, Mengyu; Awadasseid, Annoor; Wu, Yanling; Magiera-Mularz, Katarzyna; Zhang, Wen
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收藏Design, synthesis, anti-tumor activity and mechanism of novel PROTACs as degraders of PD-L1 and inhibitors of PD-1/PD-L1 interaction新型PD-L1降解剂和PD-1/PD-L1相互作用抑制剂的设计、合成、抗肿瘤活性及机制研究
Zhang, Feng; Yu, Qimeng; Wu, Caiyun; Sun, Shishi; Wang, Yu; Wang, Rui; Chen, Zejie; Zhang, Hua; Xiong, Xuqiong; Awadasseid, Annoor; Rao, Guowu; Zhao, Xiaoyin; Zhang, Wen
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收藏Design, Synthesis, and Antitumor Activity Evaluation of 2-Arylmethoxy-4-(2,2′-dihalogen-substituted biphenyl-3-ylmethoxy) Benzylamine Derivatives as Potent PD-1/PD-L1 Inhibitors
Zhang, Hua; Zhou, Shijia; Plewka, Jacek; Wu, Caiyun; Zhu, Mengyu; Yu, Qimeng; Musielak, Bogdan; Wang, Xiao; Awadasseid, Annoor; Magiera-Mularz, Katarzyna; Wu, Yanling; Zhang, Wen
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收藏PD-L1 dimerisation induced by biphenyl derivatives mediates anti-breast cancer activity via the non-immune PD-L1-AKT-mTOR/Bcl2 pathway
Zhang, Hua; Zhou, Shi-Jia; Shen, Chen-Feng; Zhou, Yong-Nan; Wu, Cai-Yun; Zhu, Meng-Yu; Yu, Qi-Meng; Awadasseid, Annoor; Wu, Yan-Ling; Zhang, Wen
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收藏Design, synthesis and bioactivity of novel naphthalimide-benzotriazole conjugates against A549 cells via targeting BCL2 G-quadruplex and inducing autophagy
Wang, Xiao; Zhang, Mi; Xiong, Xu-Qiong; Yang, Hao; Wang, Panpan; Zhang, Koutian; Awadasseid, Annoor; Narva, Suresh; Wu, Yan-Ling; Zhang, Wen
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收藏Design, synthesis and anti-tumor activity of novel benzothiophenonaphthalimide derivatives targeting mitochondrial DNA (mtDNA) G-quadruplex
Huang, Qiong; Wang, Xiao; Chen, An; Zhang, Hua; Yu, Qimeng; Shen, Chenfeng; Awadasseid, Annoor; Zhao, Xiaoyin; Xiong, Xuqiong; Wu, Yanling; Zhang, Wen
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