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Glucagon Like Peptide 1 Receptor Agonists for Targeted Delivery of Antisense Oligonucleotides to Pancreatic Beta CellJOURNAL OF THE AMERICAN CHEMICAL SOCIETYIF15.62021-02-2440PREAI
Novel Chemical Series of 5-Lipoxygenase-Activating Protein Inhibitors for Treatment of Coronary Artery DiseaseJOURNAL OF MEDICINAL CHEMISTRYIF6.82019-03-3010PREAI
Discovery and Early Clinical Development of an Inhibitor of 5-Lipoxygenase Activating Protein (AZD5718) for Treatment of Coronary Artery DiseaseJOURNAL OF MEDICINAL CHEMISTRYIF6.82019-03-1430PREAI
Discovery of a Series of Indole-2 Carboxamides as Selective Secreted Phospholipase A2 Type X (sPLA2-X) InhibitorsACS MEDICINAL CHEMISTRY LETTERSIF42018-06-239OAAI
Design of Selective sPLA2-X Inhibitor (-)-2-{2-[Carbamoyl-6-(trifluoromethoxy)-1H-indol-1-yl]pyridine-2-yl}propanoic AcidACS MEDICINAL CHEMISTRY LETTERSIF42018-06-235OAAI
A Practical Telescoped Three-Step Sequence for the Preparation of (1R,2R)-2-(4-Bronnobenzoyl)cyclohexanecarboxylic Acid: A Key Building Block Used in One of Our Drug Development ProjectsORGANIC PROCESS RESEARCH & DEVELOPMENTIF3.52018-04-2713PREAI
Discovery of AZD6642, an Inhibitor of 5-Lipoxygenase Activating Protein (FLAP) for the Treatment of Inflammatory DiseasesJOURNAL OF MEDICINAL CHEMISTRYIF6.82014-12-2238PREAI
Discovery of Agonists of Cannabinoid Receptor 1 with Restricted Central Nervous System Penetration Aimed for Treatment of Gastroesophageal Reflux DiseaseJOURNAL OF MEDICINAL CHEMISTRYIF6.82012-12-2411PREAI
Design of small molecule inhibitors of acetyl-CoA carboxylase 1 and 2 showing reduction of hepatic malonyl-CoA levels in vivo in obese Zucker ratsBIOORGANIC & MEDICINAL CHEMISTRYIF32011-05-0138PRE
Preparation of a diglycosylated hydroxylysine building block used in solid-phase synthesis of a glycopeptide from type II collagenJOURNAL OF ORGANIC CHEMISTRYIF3.61999-10-3047PREAI
T cells recognize a glycopeptide derived from type II collagen in a model for rheumatoid arthritisJOURNAL OF THE AMERICAN CHEMICAL SOCIETYIF15.61998-07-2381PREAI