未登录 Discovery of a Novel Benzodiazepine Series of Cbl-b Inhibitors for the Enhancement of Antitumor Immunity Boerth, Jeffrey A.; Chinn, Alex J.; Schimpl, Marianne; Bommakanti, Gayathri; Chan, Christina; Code, Erin L.; Giblin, Kathryn A.; Gohlke, Andrea; Hansel, Catherine S.; Jin, Meizhong; Kavanagh, Stefan L.; Lamb, Michelle L.; Lane, Jordan S.; Larner, Carrie J. B.; Mfuh, Adelphe M.; Moore, Rachel K.; Puri, Taranee; Quinn, Taylor R.; Ye, Minwei; Robbins, Kevin J.; Gancedo-Rodrigo, Miguel; Tang, Haoran; Walsh, Jarrod; Ware, Jamie; Wrigley, Gail L.; Reddy, Iswarya Karapa; Zhang, Yun; Grimster, Neil P. 分享 收藏
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Nuisance compounds in cellular assays Dahlin, Jayme L.; Auld, Douglas S.; Rothenaigner, Ina; Haney, Steve; Sexton, Jonathan Z.; Nissink, J. Willem M.; Walsh, Jarrod; Lee, Jonathan A.; Strelow, John M.; Willard, Francis S.; Ferrins, Lori; Baell, Jonathan B.; Walters, Michael A.; Hua, Bruce K.; Hadian, Kamyar; Wagner, Bridget K. 分享 收藏
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Identification and Characterization of Dual Inhibitors of the USP25/28 Deubiquitinating Enzyme Subfamily Wrigley, Jonathan D.; Gavory, Gerald; Simpson, Iain; Preston, Marian; Plant, Helen; Bradley, Jenna; Goeppert, Anne U.; Rozycka, Ewelina; Davies, Gareth; Walsh, Jarrod; Valentine, Andrea; McClelland, Keeva; Odrzywol, Krzysztofa Ewa; Renshaw, Jonathan; Boros, Joanna; Tart, Jonathan; Leach, Lindsey; Nowak, Thorsten; Ward, Richard A.; Harrison, Timothy; Andrews, David M. 分享 收藏
Discovery of Imidazo[1,2-a]pyridine Ethers and Squaramides as Selective and Potent Inhibitors of Mycobacterial Adenosine Triphosphate (ATP) Synthesis Tantry, Subramanyam J.; Markad, Shankar D.; Shinde, Vikas; Bhat, Jyothi; Balakrishnan, Gayathri; Gupta, Amit K.; Ambady, Anisha; Raichurkar, Anandkumar; Kedari, Chaitanyakumar; Sharma, Sreevalli; Mudugal, Naina V.; Narayan, Ashwini; Kumar, C. N. Naveen; Nanduri, Robert; Bharath, Sowmya; Reddy, Jitendar; Panduga, Vijender; Prabhakar, K. R.; Kandaswamy, Karthikeyan; Saralaya, Ramanatha; Kaur, Parvinder; Dinesh, Neela; Guptha, Supreeth; Rich, Kirsty; Murray, David; Plant, Helen; Preston, Marian; Ashton, Helen; Plant, Darren; Walsh, Jarrod; Alcock, Peter; Naylor, Kathryn; Collier, Matthew; Whiteaker, James; McLaughlin, Robert E.; Mallya, Meenakshi; Panda, Manoranjan; Rudrapatna, Suresh; Ramachandran, Vasanthi; Shandil, Radha; Sambandamurthy, Vasan K.; Mdluli, Khisi; Cooper, Christopher B.; Rubin, Harvey; Yano, Takahiro; Iyer, Pravin; Narayanan, Shridhar; Kavanagh, Stefan; Mukherjee, Kakoli; Balasubramanian, V.; Hosagrahara, Vinayak P.; Solapure, Suresh; Ravishankar, Sudha; Hameed, Shahul P. 分享 收藏
Discovery and Optimization of Allosteric Inhibitors of Mutant Isocitrate Dehydrogenase 1 (R132H IDH1) Displaying Activity in Human Acute Myeloid Leukemia Cells Jones, Stuart; Ahmet, Jonathan; Ayton, Kelly; Ball, Matthew; Cockerill, Mark; Fairweather, Emma; Hamilton, Nicola; Harper, Paul; Hitchin, James; Jordan, Allan; Levy, Colin; Lopez, Ruth; McKenzie, Eddie; Packer, Martin; Plant, Darren; Simpson, Iain; Simpson, Peter; Sinclair, Ian; Somervaille, Tim C. P.; Small, Helen; Spencer, Gary J.; Thomson, Graeme; Tonge, Michael; Waddell, Ian; Walsh, Jarrod; Waszkowycz, Bohdan; Wigglesworth, Mark; Wiseman, Daniel H.; Ogilvie, Donald 分享 收藏