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J

Jonathan B. Baell

monash university

52H指数
351论文数
1.5W被引数
收录论文 152
发表时间
Biological Activity and Structural Biology of Current KAT6A Inhibitor Chemotypes当前KAT6A抑制剂化学骨架的生物活性与结构生物学
err2026-01-29
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errOAAI
errAdi Suwandi; Jianwen Jin; Yichao Zhao; Ramesh Mudududdla; Yi Sing Gee; Girdhar Singh Deora; Yuxin Sun; Heping Wei; Fei Huang; Jin-Shu He; Amee J. George; Stefan J. Hermans; David J. Leaver; Michael W. Parker; Jonathan B. Baell
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Fluorinated pyrimidine 5-carboxamides as potential tools for MERTK targeted fluorine-18-PET-radioligand development氟化嘧啶-5-甲酰胺作为MERTK靶向氟-18-PET放射性配体的潜在开发工具
err2025-12-04
err0
PREAI
errRamesh Mudududdla †; Siu Wai Wong †; Nghi Nguyen; Lian Xue; Michael A. Stashko; Xiaodong Wang; Lucy Vivash; Michele D. Binder; Uwe Ackermann; Ylva E. Bozikis; Trevor J. Kilpatrick; Jonathan B. Baell
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Formylpeptide receptors: A novel target to treat cardiometabolic complications甲酰肽受体:治疗心血管代谢并发症的新型靶点
err2025-10-26
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errOAAI
errChen Huei Leo; Elizabeth A. Vecchio; Ting Fu; Xiangyan Yi; Cheng Peng; Peishen Zhao; Owen L. Woodman; Jonathan Baell; Rebecca H. Ritchie; Cheng Xue Qin
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Development of potent glutathione transferase Omega-1 inhibitors with applications in inflammation and cancer therapy开发具有抗炎和癌症治疗应用的高效谷胱甘肽转移酶Omega-1抑制剂
err2025-08-23
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PREAI
errYiyue Xie; Yuji Nakano; Padmaja Tummala; Aaron J. Oakley; Adi Suwandi; Matthew E. Cuellar; Jessica M. Strasser; Jayme L. Dahlin; Michael A. Walters; Marco G. Casarotto; Philip G. Board; Jonathan B. Baell
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Dual inhibition of AXL and MER kinase: scope for lung and breast cancer therapeuticsAXL和MER激酶的双重抑制:在肺癌和乳腺癌治疗中的应用前景
err2025-08-19
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PREAI
errBalaji Dashrath Sathe; Pratibha Kumari; Hemant Kumar; Madhav Shivaji Mane; Ramesh Mudududdla; Jonathan Baell; Roshan Kumar; Shareen Singh; D.K. Pawar; Damodara N. Kommi; Ganesh Bushi; Prateek Pathak; Ashish R. Dwivedi
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Unlocking pH-responsive dual payload release through hydrazone linkage chemistry
err2025-03-01
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PREAI
errAbd-Ellah, Heba S.; Zhao, Dan; Zhou, Yayao; Baell, Jonathan B.
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Platform of Oxidative Transformation of α-Methyl Secondary Enaminones toward Tetrahydropyridines
err2025-03-01
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PREAI
errHuang, Fei; Li, Mingrui; Jiang, Quanbin; Huang, Qingyu; Zhang, Shiyu; Wei, Heping; Li, Yufeng; Yu, Yang; Zhao, Lili; Baell, Jonathan
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Heterocyclic core modifications in trypanosomacidal 2-[(phenylheteroaryl)ethyl]ureas
err2025-01-01
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PREAI
errToynton, Arthur; Ferrins, Lori; Newson, Harriet L.; Sykes, Melissa L.; Varghese, Swapna; Nguyen, Nghi; Russell, Stephanie; Rahmani, Raphael; Cheang, Jeremy; Flematti, Gavin R.; Skelton, Brian W.; Zulfiqar, Bilal; Avery, Vicky M.; Baell, Jonathan B.; Piggott, Matthew J.
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A Collection of Useful Nuisance Compounds (CONS) for Interrogation of Bioassay Integrity
errJACS AU
IF8.7
err2024-11-25
err0
PREAI
errHu, Huabin; Yi, Xiangyan; Xue, Lian; Baell, Jonathan B.
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Phenotypic-Based Discovery and Exploration of a Resorufin Scaffold with Activity against Mycobacterium tuberculosis
err2024-10-25
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errTran, Eric; Cheung, Chen-Yi; Li, Lucy; Carter, Glen P.; Gable, Robert W.; West, Nicholas P.; Kaur, Amandeep; Gee, Yi Sing; Cook, Gregory M.; Baell, Jonathan B.; Joerg, Manuela
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Tolfenpyrad Derivatives Exhibit Potent Francisella-Specific Antibacterial Activity without Toxicity to Mammalian Cells In Vitro
err2024-10-02
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PREAI
errKhalid, Nimra; Adams, Nicole; Cunha, Federico; Taki, Aya C.; Le, Thuy G.; Baell, Jonathan B.; Heine, Henry S.; Gasser, Robin B.; Eshraghi, Aria
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Novel Diacyl-hydrazide Compounds as Potential Therapeutics for Visceral Leishmaniasis
err2024-08-22
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errOAAI
errJandl, Bernhard; Zheng, Rebecca; Muttenthaler, Markus; Baell, Jonathan
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Biased receptor signalling and intracellular trafficking profiles of structurally distinct formylpeptide receptor 2 agonists结构不同的甲酰肽受体2激动剂的偏向受体信号传导和细胞内运输概况
err2024-08-18
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errOAAI
errPeng, Cheng; Vecchio, Elizabeth A.; Nguyen, Anh T. N.; De Seram, Mia; Tang, Ruby; Keov, Peter; Woodman, Owen L.; Chen, Yung-Chih; Baell, Jonathan; May, Lauren T.; Zhao, Peishen; Ritchie, Rebecca H.; Qin, Cheng Xue
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A MOZ-TIF2 leukemia mouse model displays KAT6-dependent H3K23 propionylation and overexpression of a set of active developmental genes
err2024-06-18
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errSmolko, Anne E.; Sullivan, Daniel W.; Olsen, Sarah Naomi; Kang, Hyuckjoon; Whedon, Samuel D.; Baell, Jonathan B.; Cole, Philip A.; Armstrong, Scott A.; Kuroda, Mitzi I.
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Hit-to-lead optimization of 2-aminoquinazolines as anti-microbial agents against Leishmania donovani
err2024-04-01
err2
PREAI
errDas, Nirmal; Roy, Jayasree; Patra, Binita; Saunders, Eleanor; Sarkar, Dipika; Goon, Sunny; Sinha, Bishnu Prasad; Roy, Shreya; Roy, Swarnali; Sarif, Jafar; Bandopadhyay, Purbita; Barik, Subhasis; Mukherjee, Suravi; Mcnamara, Nicole; Varghese, Swapna; Simpson, Kaylene; Baell, Jonathan; Mcconville, Malcolm; Ganguly, Dipyaman; Talukdar, Arindam
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Novel aroyl guanidine anti-trypanosomal compounds that exert opposing effects on parasite energy metabolism
err2024-03-01
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errOAAI
errVarghese, Swapna; Srivastava, Anubhav; Wong, Siu Wai; Le, Thuy; Pitcher, Noel; Mesnard, Mathilda; Lallemand, Camille; Rahmani, Raphael; Moawad, Sarah R.; Huang, Fei; He, Tiantong; Sleebs, Brad E.; Barrett, Michael P.; Sykes, Melissa L.; Avery, Vicky M.; Creek, Darren J.; Baell, Jonathan B.
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Drug discovery and optimization based on the co-crystal structure of natural product with target
err2024-02-01
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PREAI
errChen, Xing; Varghese, Swapna; Zhang, Zhaoyan; Du, Juncheng; Ruan, Banfeng; Baell, Jonathan B.; Liu, Xinhua
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