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Sandip B. Bharate

department of natural products and medicinal chemistry

47H指数
261论文数
8.0K被引数
收录论文 102
发表时间
Discovery of 2-(4-Ureido-piperidin-1-yl)-4-morpholinothieno [3; 2-D] Pyrimidines as Orally Bioavailable Phosphoinositide-3-Kinase Inhibitors with In Vitro and In Vivo Antitumor Efficacy in Triple-Negative Breast Cancer作为口服可利用的磷脂酰肌醇-3-激酶抑制剂,2-(4-脲基-哌啶-1-基)-4-吗啉基噻吩并[3;2-D]嘧啶在体外和体内对三阴性乳腺癌均显示出抗肿瘤疗效。
err2025-10-06
err0
PREAI
errShabber Mohammed; Shabu Thakur; Diksha Manhas; Chilakala Nagarjuna Reddy; Abhisheik Eedara; Santosh K. Guru; Ajeet Singh; Mahir Bhardwaj; Vaishnavi Kambhampati; Ramajayan Pandian; Boobalan Gopu; Shashi Bhushan; Ram A. Vishwakarma; Sai Balaji Andugulapati; Shashank K. Singh; Utpal Nandi; Sandip B. Bharate
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Improving the oral bioavailability of berberine: A crystal engineering approach提高小檗碱口服生物利用度:一种晶体工程方法
err2025-09-17
err0
PREAI
errAnuja Venkata Sai Durga Surampudi; Sai Ram Prasad; Pujitha Ramanujam; Debasish Swain; Bhagyashri N. Wadje; Sandip B. Bharate; Umanath Kamalakannan; Muralidharan Kathirvel; Sridhar Balasubramanian
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Silicon incorporated tacrine: design, synthesis, and evaluation of biological and pharmacokinetic parameters
err2025-03-01
err0
PREAI
errKulkarni, Akshay S.; Ramana, Sreenivasa Rao; Nuthakki, Vijay K.; Bhatt, Shipra; Jamwal, Ashiya; Nandawadekar, Laxman D.; Jotshi, Anshika; Kumar, Ajay; Nandi, Utpal; Bharate, Sandip B.; Reddy, D. Srinivasa
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Sinigrin Selectively Mitigates the Acute-Cardiac Inflammatory Response Through an AMPK-Dependent Mechanism
err2025-02-01
err0
PREAI
errVeeram, Anjali; Patekar, Rohan R.; Bharate, Sandip B.; Andugulapati, Sai Balaji; Sistla, Ramakrishna
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Unfolding the Potential of Pyrrole- and Indole-Based Allylidene Hydrazine Carboximidamides as Antimicrobial Agents
err2025-01-13
err0
PREAI
errSharma, Amit; Jain, Sonali J.; Jha, Prabhat Nath; Rudrawar, Santosh; Bharate, Sandip B.; Jadhav, Hemant R.
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Structure-Based Virtual Screening and Biological Characterization of Novel BACE-1 and Amyloid-β Aggregation Inhibitors
err2024-12-20
err0
PREAI
errSharma, Ankita; Nayak, Madhusmita; Thakur, Shikha; Jadhav, Hemant R.; Bharate, Sandip B.
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Natural Products Driven Medicinal Chemistry
err2024-12-04
err0
PREAI
errBharate, Sandip B.; Lindsley, Craig W.
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N-Benzyl piperidine Fragment in Drug Discovery
err2024-08-23
err4
errOAAI
errSharma, Ankita; Sharma, Mohit; Bharate, Sandip B.
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Synthesis and Biological Evaluation of Colchicine-Aryl/Alkyl Amine Hybrids as Potential Noncytotoxic Cholinesterase Inhibitors: Identification of SBN-284 as a Dual Inhibitor of Cholinesterases and NLRP3 Inflammasome
err2024-07-26
err2
PREAI
errReddy, Chilakala Nagarjuna; Nuthakki, Vijay K.; Sharma, Ankita; Malik, Sumera; Tabassum, Misbah; Kumar, Rajesh; Choudhary, Sushil; Iqbal, Fiza; Tufail, Ziya; Mondhe, Dilip M.; Kumar, Ajay; Bharate, Sandip B.
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Benzopyrone, a privileged scaffold in drug discovery: An overview of FDA-approved drugs and clinical candidates
err2024-03-26
err5
PREAI
errSharma, Venu; Sharma, Ankita; Wadje, Bhagyashri N.; Bharate, Sandip B.
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Orally bioavailable styryl derivative of rohitukine-N-oxide inhibits CDK9/T1 and the growth of pancreatic cancer cells
err2023-10-01
err5
PREAI
errBhurta, Deendyal; Hossain, Md Mehedi; Bhardwaj, Mahir; Showket, Farheen; Nandi, Utpal; Dar, Mohd Jamal; Bharate, Sandip B.
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Methoxy-naphthyl-Linked N-Benzyl Pyridinium Styryls as Dual Cholinesterase Inhibitors: Design, Synthesis, Biological Evaluation, and Structure-Activity Relationship
err2023-05-09
err7
errOAAI
errAbdullaha, Mohd; Banoo, Razia; Nuthakki, Vijay K.; Sharma, Mohit; Kaur, Sukhleen; Thakur, Shikha; Kumar, Ajay; Jadhav, Hemant R.; Bharate, Sandip B.
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In vitro and in vivo anticancer potential and molecular targets of the new colchicine analog IIIM-067
err2023-01-01
err6
PREAI
errMalik, Sumera; Mintoo, Mubashir J.; Reddy, Chilakala Nagarjuna; Kumar, Rajesh; Kotwal, Pankul; Bharate, Sandip B.; Nandi, Utpal; Mondhe, Dilip M.; Shukla, Sanket K.
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