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Václav Bazgier

palacky university olomouc

H指数:18

被引数:2,426

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Development of 2,6,9-Trisubstituted Purines as Neuroprotective Agents Targeting Butyrylcholinesterase and Cannabinoid CB2 Receptor

2,6,9-三取代嘌呤作为靶向丁酰胆碱酯酶和大麻素CB2受体的神经保护剂的开发

European Journal of Medicinal Chemistry

IF5.9

2025-09-260

PRE

MOLEonline: a web-based tool for analysing channels, tunnels, and pores (2025 update)

MOLEonline：一个用于分析通道、隧道和孔隙的基于网络的工具（2025更新）

IF5.4

2025-09-010

OAAI

ChannelsDB 2.0: a comprehensive database of protein tunnels and pores in AlphaFold era

NUCLEIC ACIDS RESEARCH

IF13.1

2023-11-133

OAAI

Expanding the squaramide library as mycobacterial ATP synthase inhibitors: Innovative synthetic pathway and biological evaluation

BIOORGANIC & MEDICINAL CHEMISTRY

IF3

2023-11-012

OAAI

Novel heterocyclic hydroxamates as inhibitors of the mycobacterial zinc metalloprotease Zmp1 to probe its mechanism of function

EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

IF5.9

2022-12-016

PRE

Metabolic interactions of benzodiazepines with oxycodone ex vivo and toxicity depending on usage patterns in an animal model

BRITISH JOURNAL OF PHARMACOLOGY

IF7.7

2022-01-222

OAAI

Mol* Viewer: modern web app for 3D visualization and analysis of large biomolecular structures

Mol * Viewer: 用于3D可视化和分析大型生物分子结构的现代web应用程序

NUCLEIC ACIDS RESEARCH

IF13.1

2021-05-06587

OAAI

Novel thiazolidinedione-hydroxamates as inhibitors of Mycobacterium tuberculosis virulence factor Zmp1

EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

IF5.9

2020-01-0117

PREAI

Synthesis of novel galeterone derivatives and evaluation of their in vitro activity against prostate cancer cell lines

EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

IF5.9

2019-10-0118

PREAI

MolMeDB: Molecules on Membranes Database

DATABASE-THE JOURNAL OF BIOLOGICAL DATABASES AND CURATION

IF3.6

2019-06-2714

OAAI

Membrane-attached mammalian cytochromes P450: An overview of the membrane's effects on structure, drug binding, and interactions with redox partners

JOURNAL OF INORGANIC BIOCHEMISTRY

IF3.2

2018-06-01141

OAAI

MOLEonline: a web-based tool for analyzing channels, tunnels and pores (2018 update)

MOLEonline: 用于分析渠道、隧道和孔隙的基于网络的工具 (2018更新)

NUCLEIC ACIDS RESEARCH

IF13.1

2018-04-30203

OAAI

Discovery of N2-(4-Amino-cyclohexyl)-9-cyclopentyl-N6-(4-morpholin-4-ylmethyl-phenyl)-9H-purine-2,6-diamine as a Potent FLT3 Kinase Inhibitor for Acute Myeloid Leukemia with FLT3 Mutations

JOURNAL OF MEDICINAL CHEMISTRY

IF6.8

2018-04-1937

PREAI

Channelsdb and Moleonline - Database and Tool for Analysis of Biomacromolecular Tunnels and Pores

BIOPHYSICAL JOURNAL

IF3.1

2018-02-010

OAAI

Mole 2.5-Tool for Detection and Analysis of Macromolecular Pores and Channels

BIOPHYSICAL JOURNAL

IF3.1

2017-02-015

OAAI

Novel N-substituted indole Schiff bases as dual inhibitors of cyclooxygenase-2 and 5-lipoxygenase enzymes: Synthesis, biological activities in vitro and docking study

EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

IF5.9

2016-11-0183

PREAI

Exponential Repulsion Improves Structural Predictability of Molecular Docking

JOURNAL OF COMPUTATIONAL CHEMISTRY

IF4.8

2016-09-1310

PREAI

Novel thidiazuron-derived inhibitors of cytokinin oxidase/dehydrogenase

PLANT MOLECULAR BIOLOGY

IF3.8

2016-07-1550

PREAI

Synthesis, biological evaluation and molecular modeling of a novel series of 7-azaindole based tri-heterocyclic compounds as potent CDK2/Cyclin E inhibitors

EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

IF5.9

2016-01-0140

PREAI

Characterization of a Pyrazolo[4,3-d]pyrimidine Inhibitor of Cyclin-dependent Kinases 2 and 5 and Aurora A With Pro-Apoptotic and Anti-Angiogenic Activity In Vitro

CHEMICAL BIOLOGY & DRUG DESIGN

IF3.3

2015-09-1613

PREAI