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Christopher D. Cox

University of California System

37H指数
112论文数
4.2K被引数
收录论文 42
发表时间
Preclinical evaluation of MK-8189: A novel phosphodiesterase 10A inhibitor for the treatment of schizophreniaMK-8189的临床前评估: 一种用于治疗精神分裂症的新型磷酸二酯酶10A抑制剂
err2025-01-01
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errOAAI
errSmith, Sean M.; Toolan, Dawn; Kandebo, Monika; Vardigan, Joshua; Raheem, Izzat; Layton, Mark E.; Kern, Jeffrey C.; Cox, Christopher; Gantert, Liza; Riffel, Kerry; Hostetler, Eric; Uslaner, Jason M.
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Discovery of Broad-Spectrum Herpes Antiviral Oxazolidinone Amide Derivatives and Their Structure-Activity Relationships
err2024-07-09
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PREAI
errPlotkin, Michael A.; Labroli, Marc; Schubert, Jeffrey; Shaw, Anthony; Schlegel, Kelly-Ann S.; Berger, Richard; Cooke, Andrew J.; Hayes, Robert P.; Armacost, Kira A.; Kinek, Keith; Krosky, Paula; Burlein, Christine; Meng, Shi; Dinunzio, Edward; Murray, Edward M.; Agrawal, Sony; Madeira, Maria; Flattery, Amy; Yao, Huifang; Leithead, Andrew; Rose, William A.; Cox, Christopher; Tellers, David M.; McKenna, Philip M.; Raheem, Izzat
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Discovery of MK-8189, a Highly Potent and Selective PDE10A Inhibitor for the Treatment of Schizophrenia
err2023-01-10
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errLayton, Mark E.; Kern, Jeffrey C.; Hartingh, Timothy J.; Shipe, William D.; Raheem, Izzat; Kandebo, Monika; Hayes, Robert P.; Huszar, Sarah; Eddins, Donnie; Ma, Bennett; Fuerst, Joy; Wollenberg, Gordon K.; Li, Jing; Fritzen, Jeff; McGaughey, Georgia B.; Uslaner, Jason M.; Smith, Sean M.; Coleman, Paul J.; Cox, Christopher D.
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Redefining the Histone Deacetylase Inhibitor Pharmacophore: High Potency with No Zinc Cofactor Interaction
err2021-03-07
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errBeshore, Douglas C.; Adam, Gregory C.; Barnard, Richard J. O.; Burlein, Christine; Gallicchio, Steven N.; Holloway, M. Katharine; Krosky, Daniel; Lemaire, Wei; Myers, Robert W.; Patel, Sangita; Plotkin, Michael A.; Powell, David A.; Rada, Vanessa; Cox, Christopher D.; Coleman, Paul J.; Klein, Daniel J.; Wolkenberg, Scott E.
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Discovery of an Anion-Dependent Farnesyltransferase Inhibitor from a Phenotypic Screen
err2020-12-23
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errBukhtiyarova, Marina; Cook, Erica M.; Hancock, Paula J.; Hruza, Alan W.; Shaw, Anthony W.; Adam, Gregory C.; Barnard, Richard J. O.; McKenna, Philip M.; Holloway, M. Katharine; Bell, Ian M.; Carroll, Steve; Cornella-Taracido, Ivan; Cox, Christopher D.; Kutchukian, Peter S.; Powell, David A.; Strickland, Corey; Trotter, B. Wesley; Tudor, Matthew; Wolkenberg, Scott; Li, Jing; Tellers, David M.
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Targeted next-generation sequencing of 565 neuro-oncology patients at UCLA: A single-institution experience
err2020-01-29
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errJi, Matthew S.; Eldred, Blaine S. C.; Liu, Regina; Pianka, Sean T.; Molaie, Donna; Kevan, Bryan; Pan, Stephanie; Lai, Thomas J.; Nguyen, Nhung T.; Chow, Frances E.; Yong, William H.; Cox, Christopher D.; Reeh, Devin N.; Li, Tie; Liau, Linda M.; Nghiemphu, Phioanh L.; Cloughesy, Timothy F.; Li, Gang; Lai, Albert
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SPINT2 is hypermethylated in both IDH1 mutated and wild-type glioblastomas, and exerts tumor suppression via reduction of c-Met activationSPINT2在IDH1突变和野生型胶质母细胞瘤中均高甲基化,并通过减少c-met激活来抑制肿瘤
err2019-03-05
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errLiu, Fei; Cox, Christopher D.; Chowdhury, Reshmi; Dovek, Laura; Nguyen, Huytram; Li, Tie; Li, Sichen; Ozer, Byram; Chou, Arthur; Nhung Nguyen; Wei, Bowen; Antonios, Joseph; Soto, Horacio; Kornblum, Harley; Liau, Linda; Prins, Robert; Nghiemphu, P. Leia; Yong, William; Cloughesy, Timothy; Lai, Albert
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D-2-Hydroxyglutarate Is Necessary and Sufficient for Isocitrate Dehydrogenase 1 Mutant-Induced MIR148A Promoter Methylation异柠檬酸脱氢酶1突变体诱导的MIR148A启动子甲基化的D-2-Hydroxyglutarate是必要和充分的
err2018-05-31
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errLi, Tie; Cox, Christopher D.; Ozer, Byram H.; Nguyen, Nhung T.; Nguyen, HuyTram N.; Lai, Thomas J.; Li, Sichen; Liu, Fei; Kornblum, Harley I.; Liau, Linda M.; Nghiemphu, Phioanh L.; Cloughesy, Timothy F.; Lai, Albert
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Preclinical Characterization of the Phosphodiesterase 10A PET Tracer [11C]MK-8193
err2015-11-23
err9
PREAI
errHostetler, Eric D.; Fan, Hong; Joshi, Aniket D.; Zeng, Zhizhen; Eng, Waisi; Gantert, Liza; Holahan, Marie; Meng, Xianjun; Miller, Patricia; O'Malley, Stacey; Purcell, Mona; Riffel, Kerry; Salinas, Cristian; Williams, Mangay; Ma, Bennett; Buist, Nicole; Smith, Sean M.; Coleman, Paul J.; Cox, Christopher D.; Flores, Brock A.; Raheem, Izzat T.; Cook, Jacquelynn J.; Evelhoch, Jeffrey L.
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Elevating microRNA-122 in blood improves outcomes after temporary middle cerebral artery occlusion in rats
err2015-10-19
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errLiu, Da Zhi; Jickling, Glen C.; Ander, Bradley P.; Hull, Heather; Zhan, Xinhua; Cox, Christopher; Shroff, Natasha; Dykstra-Aiello, Cheryl; Stamova, Boryana; Sharp, Frank R.
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Discovery and Optimization of a Series of Pyrimidine-Based Phosphodiesterase 10A (PDE10A) Inhibitors through Fragment Screening, Structure-Based Design, and Parallel Synthesis
err2015-09-25
err52
PREAI
errShipe, William D.; Sharik, Steven S.; Barrow, James C.; McGaughey, Georgia B.; Theberge, Cory R.; Uslaner, Jason M.; Yan, Youwei; Renger, John J.; Smith, Sean M.; Coleman, Paul J.; Cox, Christopher D.
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Orexin Receptor Antagonists: New Therapeutic Agents for the Treatment of Insomnia
err2015-09-15
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PREAI
errRoecker, Anthony J.; Cox, Christopher D.; Colemant, Paul J.
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Inflammation Combined with Ischemia Produces Myelin Injury and Plaque-Like Aggregates of Myelin, Amyloid-β and AβPP in Adult Rat Brain
err2015-05-30
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errZhan, Xinhua; Cox, Christopher; Ander, Bradley P.; Liu, Dazhi; Stamova, Boryana; Jin, Lee-Way; Jickling, Glen C.; Sharp, Frank R.
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Shaping suvorexant: application of experimental and theoretical methods for driving synthetic designs
err2014-02-01
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errMcGaughey, Georgia; Bayly, Christopher I.; Cox, Christopher D.; Schreier, John D.; Breslin, Michael J.; Bogusky, Michael; Pitzenberger, Steve; Ball, Richard; Coleman, Paul J.
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Discovery of 5-Chloro-N-[( 5,6-dimethoxypyridin-2-yl)methyl]-2,2′:5′,3-terpyridine-3′-carboxamide (MK-1064): A Selective Orexin 2 Receptor Antagonist (2-SORA) for the Treatment of Insomnia
err2013-12-27
err78
PREAI
errRoecker, Anthony J.; Mercer, Swati P.; Schreier, John D.; Cox, Christopher D.; Fraley, Mark E.; Steen, Justin T.; Lemaire, Wei; Bruno, Joseph G.; Harrell, C. Meacham; Garson, Susan L.; Gotter, Anthony L.; Fox, Steven V.; Stevens, Joanne; Tannenbaum, Pamela L.; Prueksaritanont, Thomayant; Cabalu, Tamara D.; Cui, Donghui; Stellabott, Joyce; Hartman, George D.; Young, Steven D.; Winrow, Christopher J.; Renger, John J.; Coleman, Paul J.
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Genetic Deletion and Pharmacological Inhibition of Phosphodiesterase 10A Protects Mice From Diet-Induced Obesity and Insulin Resistance
err2013-12-13
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errNawrocki, Andrea R.; Rodriguez, Carlos G.; Toolan, Dawn M.; Price, Olga; Henry, Melanie; Forrest, Gail; Szeto, Daphne; Keohane, Carol Ann; Pan, Yie; Smith, Karen M.; Raheem, Izzat T.; Cox, Christopher D.; Hwa, Joyce; Renger, John J.; Smith, Sean M.
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Syntheses, Thermal Reactivities, and Computational Studies of Aryl-Fused Quinoxalenediynes: Effect of Extended Benzannelation on Bergman Cyclization Energetics
err2012-10-31
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PREAI
errSpence, John D.; Rios, Andro C.; Frost, Megan A.; McCutcheon, Claire M.; Cox, Christopher D.; Chavez, Sonia; Fernandez, Ramiro; Gherman, Benjamin F.
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Discovery of [(2R,5R)-5-{[(5-Fluoropyridin-2-yl)oxy]methyl}-2-methylpiperidin-1-yl][5-methyl-2-(pyrimidin-2-yl)phenyl]methanone (MK-6096): A Dual Orexin Receptor Antagonist with Potent Sleep-Promoting Properties
err2012-02-03
err121
PREAI
errColeman, Paul J.; Schreier, John D.; Cox, Christopher D.; Breslin, Michael J.; Whitman, David B.; Bogusky, Michael J.; McGaughey, Georgia B.; Bednar, Rodney A.; Lemaire, Wei; Doran, Scott M.; Fox, Steven V.; Garson, Susan L.; Gotter, Anthony L.; Harrell, C. Meacham; Reiss, Duane R.; Cabalu, Tamara D.; Cui, Donghui; Prueksaritanont, Thomayant; Stevens, Joanne; Tannenbaum, Pamela L.; Ball, Richard G.; Stellabott, Joyce; Young, Steven D.; Hartman, George D.; Winrow, Christopher J.; Renger, John J.
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Molecular markers and mechanisms of stroke: RNA studies of blood in animals and humans
err2011-04-20
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errSharp, Frank R.; Jickling, Glen C.; Stamova, Boryana; Tian, Yingfang; Zhan, Xinhua; Liu, DaZhi; Kuczynski, Beth; Cox, Christopher D.; Ander, Bradley P.
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Discovery of the Dual Orexin Receptor Antagonist [(7R)-4-(5-Chloro-1,3-benzoxazol-2-yl)-7-methyl-1,4-diazepan-1-yl][5-methyl-2-(2H-1,2,3-triazol-2-yl)phenyl]methanone (MK-4305) for the Treatment of Insomnia
err2010-06-21
err365
PREAI
errCox, Christopher D.; Breslin, Michael J.; Whitman, David B.; Schreier, John D.; McGaughey, Georgia B.; Bogusky, Michael J.; Roecker, Anthony J.; Mercer, Swati P.; Bednar, Rodney A.; Lemaire, Wei; Bruno, Joseph G.; Reiss, Duane R.; Harrell, C. Meacham; Murphy, Kathy L.; Garson, Susan L.; Doran, Scott M.; Prueksaritanont, Thomayant; Anderson, Wayne B.; Tang, Cuyue; Roller, Shane; Cabalu, Tamara D.; Cui, Donahui; Hartman, George D.; Young, Steven D.; Koblan, Ken S.; Winrow, Christopher J.; Renger, John J.; Coleman, Paul J.
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