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A first-in-class Wiskott-Aldrich syndrome protein activator with antitumor activity in hematologic cancers Spriano, Filippo; Sartori, Giulio; Sgrignani, Jacopo; Barnabei, Laura; Arribas, Alberto J.; Guala, Matilde; Del Amor, Ana Maria Carrasco; Tomasso, Meagan R.; Tarantelli, Chiara; Cascione, Luciano; Golino, Gaetanina; Riveiro, Maria E.; Bortolozzi, Roberta; Lupia, Antonio; Paduano, Francesco; Huguet, Samuel; Rezai, Keyvan; Rinaldi, Andrea; Margheriti, Francesco; Ventura, Pedro; Guarda, Greta; Costa, Giosue; Rocca, Roberta; Furlan, Alberto; Verdonk, Luuk M.; Innocenti, Paolo; Martin, Nathaniel I.; Viola, Giampietro; Driessen, Christoph; Zucca, Emanuele; Stathis, Anastasios; Gahtory, Digvijay; van den Nieuwboer, Maurits; Bornhauser, Beat; Alcaro, Stefano; Trapasso, Francesco; Cristobal, Susana; Padrick, Shae B.; Pazzi, Natalina; Cavalli, Franco; Cavalli, Andrea; Gaudio, Eugenio; Bertoni, Francesco 分享 收藏
On the effects of 30.5 GHz sinusoidal wave exposure on glioblastoma organoids Rampazzo, Elena; Persano, Luca; Karim, Nissar; Hodgking, George; Pinto, Rosanna; Casciati, Arianna; Tanori, Mirella; Zambotti, Alessandro; Bresolin, Silvia; Cani, Alice; Pannicelli, Alessandro; Davies, Ilan W.; Hancock, Cristopher; Palego, Cristiano; Viola, Giampietro; Mancuso, Mariateresa; Merla, Caterina 分享 收藏
Design, synthesis and biological evaluation of novel 2,4-thiazolidinedione derivatives able to target the human BAG3 protein Budassi, Federica; Marchioro, Chiara; Canton, Martina; Favaro, Annagiulia; Sturlese, Mattia; Urbinati, Chiara; Rusnati, Marco; Romagnoli, Romeo; Viola, Giampietro; Mariotto, Elena 分享 收藏
Molecular and functional profiling of chemotolerant cells unveils nucleoside metabolism-dependent vulnerabilities in medulloblastoma Mariotto, Elena; Rampazzo, Elena; Bortolozzi, Roberta; Rruga, Fatlum; Zeni, Ilaria; Manfreda, Lorenzo; Marchioro, Chiara; Canton, Martina; Cani, Alice; Magni, Ruben; Luchini, Alessandra; Bresolin, Silvia; Viola, Giampietro; Persano, Luca 分享 收藏
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Design, synthesis, and biological investigation of selective human carbonic anhydrase II, IX, and XII inhibitors using 7-aryl/heteroaryl triazolopyrimidines bearing a sulfanilamide scaffold Romagnoli, Romeo; De Ventura, Tiziano; Manfredini, Stefano; Baldini, Erika; Supuran, Claudiu T.; Nocentini, Alessio; Brancale, Andrea; Bortolozzi, Roberta; Manfreda, Lorenzo; Viola, Giampietro 分享 收藏
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Identification of pyrrolo[3′,4′:3,4]cyclohepta[1,2-d][1,2]oxazoles as promising new candidates for the treatment of lymphomas Barreca, Marilia; Spano, Virginia; Rocca, Roberta; Bivacqua, Roberta; Gualtieri, Gianmarco; Raimondi, Maria Valeria; Gaudio, Eugenio; Bortolozzi, Roberta; Manfreda, Lorenzo; Bai, Ruoli; Montalbano, Alessandra; Alcaro, Stefano; Hamel, Ernest; Bertoni, Francesco; Viola, Giampietro; Barraja, Paola 分享 收藏
Identification of Homoharringtonine as a potent inhibitor of glioblastoma cell proliferation and migration Porcu, Elena; Maule, Francesca; Manfreda, Lorenzo; Mariotto, Elena; Bresolin, Silvia; Cani, Alice; Bortolozzi, Roberta; Della Puppa, Alessandro; Corallo, Diana; Viola, Giampietro; Rampazzo, Elena; Persano, Luca 分享 收藏
New bioisosteric sulphur-containing choline kinase inhibitors with a tracked mode of action Luque-Navarro, Pilar M.; Paz Carrasco-Jimenez, M.; Goracci, Laura; Paredes, Jose M.; Espinar-Barranco, Laura; Valverde-Pozo, Javier; Torretta, Archimede; Parisini, Emilio; Mariotto, Elena; Marchioro, Chiara; Laso, Alejandro; Marco, Carmen; Viola, Giampietro; Lanari, Daniela; Lopez Cara, Luisa Carlota 分享 收藏
Design, Synthesis and Biological Investigation of 2-Anilino Triazolopyrimidines as Tubulin Polymerization Inhibitors with Anticancer Activities Romagnoli, Romeo; Oliva, Paola; Prencipe, Filippo; Manfredini, Stefano; Budassi, Federica; Brancale, Andrea; Ferla, Salvatore; Hamel, Ernest; Corallo, Diana; Aveic, Sanja; Manfreda, Lorenzo; Mariotto, Elena; Bortolozzi, Roberta; Viola, Giampietro 分享 收藏
Synthesis and Biological Evaluation of Highly Active 7-Anilino Triazolopyrimidines as Potent Antimicrotubule Agents Oliva, Paola; Romagnoli, Romeo; Cacciari, Barbara; Manfredini, Stefano; Padroni, Chiara; Brancale, Andrea; Ferla, Salvatore; Hamel, Ernest; Corallo, Diana; Aveic, Sanja; Milan, Noemi; Mariotto, Elena; Viola, Giampietro; Bortolozzi, Roberta 分享 收藏
Synthesis of 2H-Imidazo[2',1':2,3] [1,3]thiazolo[4,5-e]isoindol-8-yl-phenylureas with promising therapeutic features for the treatment of acute myeloid leukemia (AML) with FLT3/ITD mutations 具有治疗特征的2h-咪唑并 [2',1':2,3] [1,3] 噻唑并 [4,5-e]isoindol-8-yl-phenylureas的合成,用于治疗具有FLT3/ITD突变的急性髓系白血病 (AML) Cilibrasi, Vincenzo; Spano, Virginia; Bortolozzi, Roberta; Barreca, Marilia; Raimondi, Maria Valeria; Rocca, Roberta; Maruca, Annalisa; Montalbano, Alessandra; Alcaro, Stefano; Ronca, Roberto; Viola, Giampietro; Barraja, Paola 分享 收藏
Biological Evaluation of New Thienopyridinium and Thienopyrimidinium Derivatives as Human Choline Kinase Inhibitors Maria Luque-Navarro, Pilar; Mariotto, Elena; Ballarotto, Marco; Rubbini, Gianluca; Jose Aguilar-Troyano, Francisco; Fasiolo, Alberto; Torretta, Archimede; Parisini, Emilio; Macchiarulo, Antonio; Laso, Alejandro; Marco, Carmen; Viola, Giampietro; Paz Carrasco-Jimenez, Maria; Carlota Lopez-Cara, Luisa 分享 收藏
Cinnamic acid derivatives linked to arylpiperazines as novel potent inhibitors of tyrosinase activity and melanin synthesis 与芳基哌嗪连接的肉桂酸衍生物是酪氨酸酶活性和黑色素合成的新型有效抑制剂 Romagnoli, Romeo; Oliva, Paola; Prencipe, Filippo; Manfredini, Stefano; Ricci, Federico; Corallo, Diana; Aveic, Sanja; Mariotto, Elena; Viola, Giampietro; Bortolozzi, Roberta; Germano, Maria Paola; De Luca, Laura 分享 收藏