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J

Jie Xu

goethe-universitaet frankfurt
H指数:14
被引数:556

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Efficient Manufacturing Process for the Selective Estrogen Receptor Degrader GDC-9545 (Giredestrant) via a Crystallization-Driven Diastereoselective Pictet-Spengler Condensation

通过结晶驱动的非对映选择性pictet-spengler缩合的选择性雌激素受体降解GDC-9545 (giedestrant) 的有效制造工艺

2021-11-095
PREAI
First-Generation Asymmetric Synthesis of the Selective Estrogen Receptor Degrader GDC-9545 (Giredestrant) Featuring a Highly Efficient Pictet-Spengler Reaction and a C-N Coupling Reaction

选择性雌激素受体降解GDC-9545 (Giredestrant) 的第一代不对称合成,具有高效的pictet-spengler反应和c-n偶联反应

2021-11-053
PREAI