未登录 Transaminases Provide Key Chiral Building Blocks for the Synthesis of Selective M1/M4 Agonists Thomson, Christopher G.; Boss, Kelly; Calhoun, Amy; Fridrich, Cary; Gardinier, Kevin M.; Hall, Edward C.; Jendza, Keith; Kirman, Louise; Labbe-Giguere, Nancy; Laumen, Kurt; Qian, Ming; Sanyal, Sanjit; Shultz, Michael D.; Snajdrova, Radka; Tan, Kian; Wang, Kate Yaping; Yang, Fan; Gao, Feng; Hong, Tao; Dale, Elena; Kuzmiski, Brent; Ortuno, Danny; Palacios, Daniel S. 分享 收藏
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Systematic Chemogenetic Library Assembly Canham, Stephen M.; Wang, Yuan; Cornett, Allen; Auld, Douglas S.; Baeschlin, Daniel K.; Patoor, Maude; Skaanderup, Philip R.; Honda, Ayako; Llamas, Luis; Wendel, Greg; Mapa, Felipa A.; Aspesi, Peter, Jr.; Labbe-Giguere, Nancy; Gamber, Gabriel G.; Palacios, Daniel S.; Schuffenhauer, Ansgar; Deng, Zhan; Nigsch, Florian; Frederiksen, Mathias; Bushell, Simon M.; Rothman, Deborah; Jain, Rishi K.; Hemmerle, Horst; Briner, Karin; Porter, Jeffery A.; Tallarico, John A.; Jenkins, Jeremy L. 分享 收藏
Scaffold Morphing Identifies 3-Pyridyl Azetidine Ureas as Inhibitors of Nicotinamide Phosphoribosyltransferase (NAMPT) Palacios, Daniel S.; Meredith, Erik L.; Kawanami, Toshio; Adams, Christopher M.; Chen, Xin; Darsigny, Veronique; Palermo, Mark; Baird, Daniel; George, Elizabeth L.; Guy, Chantale; Hewett, Jeffrey; Tierney, Laryssa; Thigale, Sachin; Wang, Louis; Weihofen, Wilhelm A. 分享 收藏
Nicotinamide Phosphoribosyltransferase Inhibitor as a Novel Payload for Antibody-Drug Conjugates 烟酰胺磷酸核糖转移酶抑制剂作为抗体-药物缀合物的新型有效载荷 Karpov, Alexei S.; Abrams, Tinya; Clark, Suzanna; Raikar, Ankita; D'Alessio, Joseph A.; Dillon, Michael P.; Gesner, Thomas G.; Jones, Darryl; Lacaud, Marion; Mallet, William; Martyniuk, Piotr; Meredith, Erik; Mohseni, Morvarid; Nieto-Oberhuber, Cristina M.; Palacios, Daniel; Perruccio, Francesca; Piizzi, Grazia; Zurini, Mauro; Bialucha, Carl Uli 分享 收藏
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