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J

James A. Nieman

University of Alberta
H指数:22
被引数:2,376

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SARS-CoV-2 Mpro Protease Variants of Concern Display Altered Viral Substrate and Cell Host Target Galectin-8 Processing but Retain Sensitivity toward Antivirals
2023-03-2124
OAAI
Improved SARS-CoV-2 Mpro inhibitors based on feline antiviral drug GC376: Structural enhancements, increased solubility, and micellar studies
2021-10-0171
OAAI
Peptidomimetic α-Acyloxymethylketone Warheads with Six-Membered Lactam P1 Glutamine Mimic: SARS-CoV-2 3CL Protease Inhibition, Coronavirus Antiviral Activity, and in Vitro Biological Stability
2021-07-0975
PREAI
Discovery of Ketone-Based Covalent Inhibitors of Coronavirus 3CL Proteases for the Potential Therapeutic Treatment of COVID-19
2020-10-15388
OAAI
Comprehensive in vitro characterization of PD-L1 small molecule inhibitors
2019-08-27104
OAAI
Discovery of a Novel Class of Boron-Based Antibacterials with Activity against Gram-Negative Bacteria
2013-03-01177
OA