未登录

I

Ingebrigt Sylte

uit—the arctic university of norway

H指数:31

被引数:3,404

个人简介

暂无内容

教育背景

暂无内容

工作经历

暂无内容

荣誉奖项

暂无内容

Identification of novel N-benzyloxy-amino acid hydroxamates as inhibitors of the virulence factor LasB from Pseudomonas aeruginosa

新型苄氧基氨基酸羟酰胺作为铜绿假单胞菌毒力因子LasB抑制剂的鉴定

IF3.6

2025-08-140

PRE

Identification of Orthosteric GABAB Receptor Ligands by Virtual Screening and In Vitro Validation

通过虚拟筛选和体外验证鉴定正构GABAB受体配体

IF4.3

2025-05-160

OA

Zinc-Chelating Compounds as Inhibitors of Human and Bacterial Zinc Metalloproteases

IF4.6

2021-12-225

OAAI

Inhibition of bacterial and human zinc-metalloproteases by bisphosphonate- and catechol-containing compounds

JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY

IF5.4

2021-03-236

OAAI

The GABABReceptor-Structure, Ligand Binding and Drug Development

IF4.6

2020-07-0777

OAAI

Protonation states of central amino acids in a zinc metalloprotease complexed with inhibitor: Molecular mechanics optimizations and ab initio molecular orbital calculations

BIOPHYSICAL CHEMISTRY

IF2.2

2020-06-016

OAAI

Exploring Conformational Dynamics of the Extracellular Venus flytrap Domain of the GABAB Receptor: A Path-Metadynamics Study

JOURNAL OF CHEMICAL INFORMATION AND MODELING

IF5.3

2020-04-018

OAAI

Molecular modelling, synthesis, and biological evaluations of a 3,5-disubstituted isoxazole fatty acid analogue as a PPARα-selective agonist

作为ppar α 选择性激动剂的3，5-二取代异恶唑脂肪酸类似物的分子建模，合成和生物学评估

BIOORGANIC & MEDICINAL CHEMISTRY

IF3

2019-09-016

OAAI

In Silico Methods for the Discovery of Orthosteric GABAB Receptor Compounds

IF4.6

2019-03-079

OAAI

In Silico Site-Directed Mutagenesis Informs Species-Specific Predictions of Chemical Susceptibility Derived From the Sequence Alignment to Predict Across Species Susceptibility (SeqAPASS) Tool

TOXICOLOGICAL SCIENCES

IF4.1

2018-07-2722

OAAI

In Vitro and in Silico Competitive Binding of Brominated Polyphenyl Ether Contaminants with Human and Gull Thyroid Hormone Transport Proteins

ENVIRONMENTAL SCIENCE & TECHNOLOGY

IF11.3

2018-01-1618

OAAI

Serotonin transporter and receptor ligands with antidepressant activity as neuroprotective and proapoptotic agents

PHARMACOLOGICAL REPORTS

IF3.8

2017-06-0123

PREAI

From Homology Models to a Set of Predictive Binding Pockets-a 5-HT1A Receptor Case Study

JOURNAL OF CHEMICAL INFORMATION AND MODELING

IF5.3

2017-01-1822

OAAI

Environmental Chemicals Modulate Polar Bear (Ursus maritimus) Peroxisome Proliferator-Activated Receptor Gamma (PPARG) and Adipogenesis in Vitro

ENVIRONMENTAL SCIENCE & TECHNOLOGY

IF11.3

2016-09-1938

PREAI

Synthesis, experimental evaluation and molecular modelling of hydroxamate derivatives as zinc metalloproteinase inhibitors

EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

IF5.9

2016-01-0115

OAAI

Synthesis, biological evaluation and molecular modeling studies of the PPARβ/δ antagonist CC618

EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

IF5.9

2015-04-0110

OAAI

Inhibition of pseudolysin and thermolysin by hydroxamate-based MMP inhibitors

EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

IF5.9

2015-01-0120

PREAI

Ligand-directed trafficking of receptor stimulus

PHARMACOLOGICAL REPORTS

IF3.8

2014-12-019

PREAI

Development of new LXR modulators that regulate LXR target genes and reduce lipogenesis in human cell models

EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

IF5.9

2014-03-017

PREAI

Identification of Novel Serotonin Transporter Compounds by Virtual Screening

JOURNAL OF CHEMICAL INFORMATION AND MODELING

IF5.3

2014-02-2634

OAAI