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收藏Design and Discovery of Substituted 1,3,4-Thiadiazole-1,3,5-Triazine Hybrids as Human Immunodeficiency Virus-1 Non-Nucleoside Reverse Transcriptase Inhibitors with Anti-SARS-CoV-2 and Antibacterial Activities设计并发现取代的1,3,4-噻二唑-1,3,5-三嗪杂合物作为具有抗SARS-CoV-2和抗菌活性的人类免疫缺陷病毒-1非核苷类反转录酶抑制剂
Singh, Saumya; Srivastava, Kumar Saurabh; Kumawat, Mukesh Kumar; Bhat, Hans Raj; Corona, Angela; Tramontano, Enzo; Mitra, Debashis; Singh, Udaya Pratap
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收藏Design, discovery, molecular docking, dynamics and in-silico ADME-T evaluation of novel hybrids of 1,3,5-triazine-morpholi-no-thiazine as an anti-diabetic agent in Wistar rats via inhibition of DPP-4 (vol 1332, 141707, 2025)设计、发现、分子对接、动力学及对新型1,3,5-三嗪-吗啉基-噻唑嗪杂交物的计算机辅助ADME-T评价,作为通过抑制DPP-4发挥作用的抗糖尿病药物(在Wistar大鼠中的研究)(卷1332,141707,2025)
Gupta, Akanksha; Anand, Ananya Anurag; Samanta, Sintu Kumar; Bhat, Hans Raj; Singh, Udaya Pratap
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收藏Design, discovery, molecular docking, dynamics and in-silico ADME-T evaluation of novel hybrids of 1,3,5-triazine-morpholino-thiazine as an anti-diabetic agent in Wistar rats via inhibition of DPP-41,3,5-三嗪-吗啉基噻嗪的新型杂合体的设计,发现,分子对接,动力学和硅adme-t评估通过抑制DPP-4在Wistar大鼠中作为抗糖尿病药
Gupta, Akanksha; Anand, Ananya Anurag; Samanta, Sintu Kumar; Bhat, Hans Raj; Singh, Udaya Pratap
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收藏In Silico Study, Synthesis, and In Vitro Evaluation of Nicotinamide-Substituted 1,3,5-Triazine Derivatives as Inhibitors of Acetylcholinesterase and Butyrylcholinesterase
Kalita, Tutumoni; Dutta, Swarnendu; Shakya, Anshul; Ghosh, Surajit Kumar; Singh, Udaya Pratap; Bhat, Hans Raj
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收藏Ebselen: A Review on its Synthesis, Derivatives, Anticancer Efficacy and Utility in Combating SARS-COV-2
Ali, Farak; Alom, Shahnaz; Ali, Sheikh Rezzak; Kondoli, Biswanarayan; Sadhu, Prativa; Borah, Chinmoyee; Kakoti, Bibhuti Bushan; Ghosh, Surajit Kumar; Shakya, Anshul; Ahmed, Abdul Baquee; Singh, Udaya Pratap; Bhat, Hans Raj
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收藏Microwave-assisted synthesis of hybrid PABA-1,3,5-triazine derivatives as an antimalarial agent
Kashyap, Ankita; Choudhury, Ayesha A. K.; Saha, Ashmita; Adhikari, Nayana; Ghosh, Surajit K.; Shakya, Anshul; Patgiri, Saurav J.; Bhattacharyya, Dibya R.; Singh, Udaya P.; Bhat, Hans R.
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收藏In silico study, synthesis, and evaluation of the antimalarial activity of hybrid dimethoxy pyrazole 1,3,5-triazine derivatives
Gogoi, Pinku; Shakya, Anshul; Ghosh, Surajit K.; Gogoi, Neelutpal; Gahtori, Prashant; Singh, Nardev; Bhattacharyya, Dibya R.; Singh, Udaya P.; Bhat, Hans R.
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收藏In silico ADMET study, docking, synthesis and antimalarial evaluation of thiazole-1,3,5-triazine derivatives as Pf-DHFR inhibitor
Sahu, Supriya; Ghosh, Surajit Kumar; Gahtori, Prashant; Singh, Udaya Pratap; Bhattacharyya, Dibya Ranjan; Bhat, Hans Raj
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