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SaveDiscovery of Novel 3-Phenylpiperidine Derivatives Targeting the β-Catenin/B-Cell Lymphoma 9 Interaction as a Single Agent and in Combination with the Anti-PD-1 Antibody for the Treatment of Colorectal Cancer
Zhang, Hao; Liu, Chenglong; Chen, Qiushi; Shen, Li-An; Xiao, Wenting; Li, Jiayi; Wang, Yonghui; Zhu, Di; Zhang, Qingwei; Li, Jianqi
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SaveTargeting actin-bundling protein L-plastin as an anabolic therapy for bone loss
Li, Xiaoqun; Wang, Lipeng; Huang, Biaotong; Gu, Yanqiu; Luo, Ying; Zhi, Xin; Hu, Yan; Zhang, Hao; Gu, Zhengrong; Cui, Jin; Cao, Liehu; Guo, Jiawei; Wang, Yajun; Zhou, Qirong; Jiang, Hao; Fang, Chao; Weng, Weizong; Chen, Xiaofei; Chen, Xiao; Su, Jiacan
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SaveN-(7-Cyano-6-(4-fluoro-3-(2-(3-(trifluoromethyl)phenyl)acetarnido)phenoxy)benzo[d]thiazol-2-yl)cyclopropanecarboxamide (TAK-632) Analogues as Novel Necroptosis Inhibitors by Targeting Receptor-Interacting Protein Kinase 3 (RIPK3): Synthesis, Structure-Activity Relationships, and in Vivo Efficacy
Zhang, Hao; Xu, Lijuan; Qin, Xia; Chen, Xiaofei; Cong, Hui; Hu, Longmiao; Chen, Long; Miao, Zhenyuan; Zhang, Wannian; Cai, Zhenyu; Zhuang, Chunlin
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SaveIdentification of the Raf kinase inhibitor TAK-632 and its analogues as potent inhibitors of necroptosis by targeting RIPK1 and RIPK3
Chen, Xiaofei; Zhuang, Chunlin; Ren, Yibin; Zhang, Hao; Qin, Xia; Hu, Longmiao; Fu, Jing; Miao, Zhenyuan; Chai, Yifeng; Li, Zheng-gang; Zhang, Haibing; Cai, Zhenyu; Wang, Hong-yang
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SaveATF4 destabilizes RET through nonclassical GRP78 inhibition to enhance chemosensitivity to bortezomib in human osteosarcoma
Luo, Jie; Xia, Yuanzheng; Yin, Yong; Luo, Jun; Liu, Mingming; Zhang, Hao; Zhang, Chao; Zhao, Yucheng; Yang, Lei; Kong, Lingyi
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SaveFragment-growing guided design of Keap1-Nrf2 protein-protein interaction inhibitors for targeting myocarditis
Meng, Ning; Tang, Hua; Zhang, Hao; Jiang, Chengshi; Su, Li; Min, Xiao; Zhang, Wannian; Zhang, Hua; Miao, Zhenyuan; Zhang, Wen; Zhuang, Chunlin
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SaveDifferential effects on lung and bone metastasis of breast cancer by Wnt signalling inhibitor DKK1
Zhuang, Xueqian; Zhang, Hao; Li, Xiaoyan; Li, Xiaoxun; Cong, Min; Peng, Fangli; Yu, Jingyi; Zhang, Xue; Yang, Qifeng; Hu, Guohong
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