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Maurizio Botta

University of Siena

60H-index
626Paper Count
1.5WCitation Count
Published Papers 226
Publication Date
Investigating the potential of the SI306 Src inhibitor and its liposomal formulation in the non-small cell lung cancer treatment
err2025-07-25
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PREAI
errFederica Poggialini; Enrico Rango; Chiara Vagaggini; Sara Diana; Annalaura Brai; Giancarlo Grossi; Maria Frosini; Francesca Musumeci; Anna Carbone; Maurizio Botta; Elena Dreassi; Silvia Schenone
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The Pyrazolo[3,4-d]Pyrimidine Derivative Si306 Encapsulated into Anti-GD2-Immunoliposomes as Therapeutic Treatment of Neuroblastoma
err2022-03-12
err9
errOAAI
errRango, Enrico; Pastorino, Fabio; Brignole, Chiara; Mancini, Arianna; Poggialini, Federica; Di Maria, Salvatore; Zamperini, Claudio; Iovenitti, Giulia; Fallacara, Anna Lucia; Sabetta, Samantha; Clementi, Letizia; Valoti, Massimo; Schenone, Silvia; Angelucci, Adriano; Ponzoni, Mirco; Dreassi, Elena; Botta, Maurizio
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Si113-prodrugs selectively activated by plasmin against hepatocellular and ovarian carcinoma
err2021-11-01
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PREAI
errRango, Enrico; D'Antona, Lucia; Iovenitti, Giulia; Brai, Annalaura; Mancini, Arianna; Zamperini, Claudio; Trivisani, Claudia Immacolata; Marianelli, Stefano; Fallacara, Anna Lucia; Molinari, Alessio; Cianciusi, Annarita; Schenone, Silvia; Perrotti, Nicola; Dreassi, Elena; Botta, Maurizio
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DDX3X inhibitors, an effective way to overcome HIV-1 resistance targeting host proteins
err2020-08-01
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errOAAI
errBrai, Annalaura; Riva, Valentina; Saladini, Francesco; Zamperini, Claudio; Trivisani, Claudia Immacolata; Garbelli, Anna; Pennisi, Carla; Giannini, Alessia; Boccuto, Adele; Bugli, Francesca; Martini, Maurizio; Sanguinetti, Maurizio; Zazzi, Maurizio; Dreassi, Elena; Botta, Maurizio; Maga, Giovanni
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Unique Domain for a Unique Target: Selective Inhibitors of Host Cell DDX3X to Fight Emerging Viruses
err2020-07-30
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errRiva, Valentina; Garbelli, Anna; Brai, Annalaura; Casiraghi, Federica; Fazi, Roberta; Trivisani, Claudia I.; Boccuto, Adele; Saladini, Francesco; Vicenti, Ilaria; Martelli, Francesco; Zazzi, Maurizio; Giannecchini, Simone; Dreassi, Elena; Botta, Maurizio; Maga, Giovanni
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Dual SMO/BRAF Inhibition by Flavonolignans from Silybum marianum
err2020-05-05
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errOAAI
errDiukendjieva, Antonia; Zaharieva, Maya M.; Mori, Mattia; Alov, Petko; Tsakovska, Ivanka; Pencheva, Tania; Najdenski, Hristo; Kren, Vladimir; Felici, Chiara; Bufalieri, Francesca; Di Marcotullio, Lucia; Botta, Bruno; Botta, Maurizio; Pajeva, Ilza
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Exploring the Implication of DDX3X in DENV Infection: Discovery of the First-in-Class DDX3X Fluorescent Inhibitor
err2020-04-09
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errOAAI
errBrai, Annalaura; Boccuto, Adele; Monti, Martina; Marchi, Serena; Vicenti, Ilaria; Saladini, Francesco; Trivisani, Claudia Immacolata; Pollutri, Alessandro; Trombetta, Claudia Maria; Montomoli, Emanuele; Riva, Valentina; Garbelli, Anna; Nola, Emanuele Maria; Zazzi, Maurizio; Maga, Giovanni; Dreassi, Elena; Botta, Maurizio
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5,6-Dihydroxypyrimidine Scaffold to Target HIV-1 Nucleocapsid Protein
err2020-03-19
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errOAAI
errMalancona, Savina; Mori, Mattia; Fezzardi, Paola; Santoriello, Marisabella; Basta, Andreina; Nibbio, Martina; Kovalenko, Lesia; Speziale, Roberto; Battista, Maria Rosaria; Cellucci, Antonella; Gennari, Nadia; Monteagudo, Edith; Di Marco, Annalise; Giannini, Alessia; Sharma, Rajhans; Pires, Manuel; Real, Eleonore; Zazzi, Maurizio; Lang, Maria Chiara Dasso; De Forni, Davide; Saladini, Francesco; Mely, Yves; Summa, Vincenzo; Harper, Steven; Botta, Maurizio
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Identification of Phosphate-Containing Compounds as New Inhibitors of 14-3-3/c-Abl Protein-Protein Interaction
err2020-03-06
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PREAI
errIralde-Lorente, Leire; Tassone, Giusy; Clementi, Letizia; Franci, Lorenzo; Munier, Claire C.; Cau, Ylenia; Mori, Mattia; Chiariello, Mario; Angelucci, Adriano; Perry, Matthew W. D.; Pozzi, Cecilia; Mangani, Stefano; Botta, Maurizio
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AuNP Pyrazolo[3,4-d]pyrimidine Nanosystem in Combination with Radiotherapy against Glioblastoma
err2020-03-05
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errOAAI
errMolinari, Alessio; Iovenitti, Giulia; Mancini, Arianna; Gravina, Giovanni Luca; Chebbi, Monia; Caruana, Maura; Vignaroli, Giulia; Orofino, Francesco; Rango, Enrico; Angelucci, Adriano; Dreassi, Elena; Schenone, Silvia; Botta, Maurizio
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Predictive Gene Signature for Pyrazolopyrimidine Derivative c-Src Inhibitor 10a Sensitivity in Melanoma Cells
err2020-02-18
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errOAAI
errKucukkaraduman, Baris; Turk, Can; Fallacara, Anna L.; Isbilen, Murat; Senses, Kerem M.; Ayyildiz, Zeynep O.; Akbar, Muhammad W.; Lotem, Michal; Botta, Maurizio; Gure, Ali O.
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Discovery of small molecule inhibitors of Leishmania braziliensis Hsp90 chaperone
err2020-02-12
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errOAAI
errBatista, Fernanda A. H.; Ramos, Sergio L., Jr.; Tassone, Giusy; Leitao, Andrei; Montanari, Carlos A.; Botta, Maurizio; Mori, Mattia; Borges, Julio C.
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(Thia)calixarenephosphonic Acids as Potent Inhibitors of the Nucleic Acid Chaperone Activity of the HIV-1 Nucleocapsid Protein with a New Binding Mode and Multitarget Antiviral Activity
err2020-02-11
err9
errOAAI
errHumbert, Nicolas; Kovalenko, Lesia; Saladini, Francesco; Giannini, Alessia; Pires, Manuel; Botzanowski, Thomas; Cherenok, Sergiy; Boudier, Christian; Sharma, Kamal K.; Real, Eleonore; Zaporozhets, Olga A.; Cianferani, Sarah; Seguin-Devaux, Carole; Poggialini, Federica; Botta, Maurizio; Zazzi, Maurizio; Kalchenko, Vitaly, I; Mori, Mattia; Mely, Yves
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Synthesis and Antiproliferative Activity of Nitric Oxide-Donor Largazole Prodrugs
err2020-02-07
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errOAAI
errBorgini, Matteo; Zamperini, Claudio; Poggialini, Federica; Ferrante, Luca; Summa, Vincenzo; Botta, Maurizio; Di Fabio, Romano
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Synthesis and Antiviral Activity of Novel 1,3,4-Thiadiazole Inhibitors of DDX3X
err2019-11-04
err34
errOAAI
errBrai, Annalaura; Ronzini, Stefania; Riva, Valentina; Botta, Lorenzo; Zamperini, Claudio; Borgini, Matteo; Trivisani, Claudia Immacolata; Garbelli, Anna; Pennisi, Carla; Boccuto, Adele; Saladini, Francesco; Zazzi, Maurizio; Maga, Giovanni; Botta, Maurizio
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Identification of a new family of pyrazolo[3,4-d]pyrimidine derivatives as multitarget Fyn-Blk-Lyn inhibitors active on B- and T-lymphoma cell lines
err2019-11-01
err13
PREAI
errFallacara, Anna Lucia; Passannanti, Raffaele; Mori, Mattia; Iovenitti, Giulia; Musumeci, Francesca; Greco, Chiara; Crespan, Emmanuele; Kissova, Miroslava; Maga, Giovanni; Tarantelli, Chiara; Spriano, Filippo; Gaudio, Eugenio; Bertoni, Francesco; Botta, Maurizio; Schenone, Silvia
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A Molecular Tool Targeting the Base-Flipping Activity of Human UHRF1
err2019-09-13
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PREAI
errZaayter, Liliyana; Mori, Mattia; Ahmad, Tanveer; Ashraf, Waseem; Boudier, Christian; Kilin, Vasyl; Gavvala, Krishna; Richert, Ludovic; Eiler, Sylvia; Ruff, Marc; Botta, Maurizio; Bronner, Christian; Mousli, Marc; Mely, Yves
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Synthesis of distal and proximal fleximer base analogues and evaluation in the nucleocapsid protein of HIV-1
err2019-07-01
err9
errOAAI
errKu, Therese; Lopresti, Natalie; Shirley, Matthew; Mori, Mattia; Marchant, Jan; Heng, Xiao; Botta, Maurizio; Summers, Michael F.; Seley-Radtke, Katherine L.
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Preclinical development of novel pyrazolo[3,4-d]pyrimidines structure-based TKIs for the treatment of glioblastoma
err2019-07-01
err0
PREAI
errMancini, Arianna; Fallacara, Anna Lucia; Zamperini, Claudio; Iovenitti, Giulia; Molinari, Alessio; Rango, Enrico; Angelucci, Adriano; Schenone, Silvia; Botta, Maurizio
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