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Hiroyuki Kusuhara

the university of tokyo

84H-index
457Paper Count
2.0WCitation Count
Published Papers 194
Publication Date
A novel selective stabilizer of the ryanodine receptor 2 prevents stress-induced ventricular arrhythmias without impairing cardiac function
err2026-04-27
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errNagomi Kurebayashi; Masami Kodama; Hana Inoue; Masato Konishi; Masami Sugihara; Takashi Murayama; Ryosuke Ishida; Koichiro Ishii; Shuichi Mori; Yukari Endo; Xi Zeng; Yukiko U. Inoue; Takayoshi Inoue; Satoru Noguchi; Hajime Nishio; Eri Nakashima; Norio Suzuki; Noriko Nakaya; Ryushi Sato; Yuya Otori; Ayuna Tsutsumi; Mirei Takahashi; Takayuki Oka; Haruo Ogawa; Kayoko Kanamitsu; Hiroyuki Kusuhara; Utako Yokoyama; Junko Kurokawa; Hiroyuki Kagechika; Takashi Sakurai
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Continuous bile excretion from polarized hepatocytes on a microchannel-patterned device
err2026-03-31
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errOAAI
errFumiya Tokito; Hiroshi Arakawa; Yuya Nakazono; Mikito Kiyofuji; Yang Liang; Fukino Kono; Mathieu Danoy; Hyunjin Choi; Ya Gong; Katsuhiro Esashika; Jingjing Yang; Satoshi Yamasaki; Natsuko F. Inagaki; Taichi Ito; Kenpei Tai; Hiroyuki Kusuhara; Yusuke Masuo; Yukio Kato; Ikumi Tamai; Takeshi Katsuda
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Discovery of an HDAC2-Selective Inhibitor via Enzyme−Inhibitor-Binding Thermodynamics/Kinetics as a Prospective Neurological Disorder Drug
err2026-01-01
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PREAI
errT Tojo; Yukihiro Itoh; Takashi Kurohara; Ying Li; Ritesh Singh; Remy Narozny; Alexander M. A. van der Wiel; Rio Furutani; Yuka Miyake; Yasunobu Yamashita; Hiroyuki Kusuhara; Kayoko Kanamitsu; Naotaka Horiguchi; Hiroko Ono; Ken‐ichi Kusakabe; Shusaku Uchida; Takayoshi Suzuki
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Intracerebral Distribution of Drugs with Diverse Blood–brain Barrier Transport Characteristics: In vivo Analysis using Brain Microdialysis in Cynomolgus Monkeys
err2025-12-16
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PREAI
errTakuya Fujita; Yukari Kamikozawa; Makoto Ozawa; Yoriko Tajima; Toshiki Kurosawa; Yuki Katagiri; Hiroko Kawaguchi; Akito Kakuuchi; Rei Miyamoto; Kentaro Wakayama; Mika Nagai; Takayuki Taguchi; Koji Bessho; Daisuke Watanabe; Takuo Ogihara; Hiroyuki Kusuhara; Yoshiharu Deguchi
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Removing Extracellular Matrix From the Cell Surface Prior to Seeding Enhances the Adhesion of Primary Human Hepatocytes to the Culture Vessel
err2025-11-01
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PREAI
errMiyai, Manami; Tanaka-Yachi, Rieko; Aizawa, Kazuko; Okamura, Kohji; Kusuhara, Hiroyuki; Akutsu, Hidenori; Nakamura, Kazuaki
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Development of Single-Molecule Enzyme Activity Assay for Serine Hydrolases Using Activity-Based Protein Labeling Probes
err2025-09-01
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errOAAI
errIshii, Seiya; Minoda, Mayano; Mizuno, Tadahaya; Iwasaka, Takumi; Kusuhara, Hiroyuki; Honda, Kazufumi; Urano, Yasuteru; Komatsu, Toru
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The role of FLVCR1 and FLVCR2 in choline transport in the Caco-2 intestinal epithelial cell model and rat small intestine
err2025-06-18
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PREAI
errYasujima, Tomoya; Namba, Chitaka; Azuma, Yosuke; Shinoda, Yutaro; Matake, Isamu; Yamasaki, Mione; Morimoto, Haruka; Namai, Mana; Kusuhara, Hiroyuki; Inoue, Katsuhisa; Yamashiro, Takahiro; Yuasa, Hiroaki
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Contribution of Japanese scientists to drug metabolism and disposition
err2025-05-01
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PREAI
errNakajima, Miki; Yamazaki, Hiroshi; Yoshinari, Kouichi; Kobayashi, Kaoru; Ishii, Yuji; Nakai, Daisuke; Kamimura, Hidetaka; Kume, Toshiyuki; Saito, Yoshiro; Maeda, Kazuya; Kusuhara, Hiroyuki; Tamai, Ikumi
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Characterization of intestinal transporters in human ileal spheroid-derived differentiated cells for the prediction of intestinal drug absorption
err2025-05-01
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PREAI
errMichiba, Kazuyoshi; Namai, Mana; Hashimoto, Yoshiki; Shimomura, Osamu; Miyazaki, Yoshihiro; Hashimoto, Shinji; Ohara, Yusuke; Enomoto, Tsuyoshi; Oda, Tatsuya; Maeda, Kazuya; Kusuhara, Hiroyuki
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Pharmacokinetics and protein binding of cholesterol-conjugated heteroduplex oligonucleotide
err2025-04-01
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errOAAI
errYoshioka, Yukitake; Yamamoto, Syunsuke; Kusamori, Kosuke; Nakayama, Miyu; Fujita, Hisashi; Goto, Akihiko; Iwasaki, Shinji; Nagata, Tetsuya; Itakura, Shoko; Kusuhara, Hiroyuki; Yokota, Takanori; Hirabayashi, Hideki
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Development of an OATP1-humanized transchromosomic mouse model for prediction of hepatic drug uptake in humans
err2025-02-01
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PREAI
errKoishikawa, Tomoki; Kazuki, Kanako; Ohnishi, Rina; Okita, Koki; Mizuno, Tadahaya; Abe, Satoshi; Nanchi, Isamu; Masago, Yusaku; Yamazaki, Kyotaro; Ohzeki, Jun-ichiro; Kusuhara, Hiroyuki; Kazuki, Yasuhiro
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Development of the serotonin release assay with enterochromaffin cell-rich human intestinal organoids for the risk evaluation of drug-induced emesis
err2024-12-17
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PREAI
errHashimoto, Yoshiki; Maeda, Kazuya; Shimomura, Osamu; Miyazaki, Yoshihiro; Hashimoto, Shinji; Oda, Tatsuya; Kusuhara, Hiroyuki
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Development of a novel gut microphysiological system that facilitates assessment of drug absorption kinetics in gut
err2024-12-02
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errOAAI
errImaoka, Tomoki; Onuki-Nagasaki, Reiko; Kimura, Hiroshi; Tai, Kempei; Ishii, Mitsuharu; Nozue, Ayaka; Kaisaki, Ikuko; Hoshi, Misa; Watanabe, Kengo; Maeda, Kazuya; Kamizono, Takashi; Yoshioka, Takahiro; Fujimoto, Takashi; Satoh, Taku; Nakamura, Hiroko; Ando, Osamu; Kusuhara, Hiroyuki; Ito, Yuzuru
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SLC35G1 is a highly chloride-sensitive transporter responsible for the basolateral membrane transport in intestinal citrate absorption
err2024-11-07
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errOAAI
errMimura, Yoshihisa; Yasujima, Tomoya; Inoue, Katsuhisa; Akino, Shogo; Namba, Chitaka; Kusuhara, Hiroyuki; Sekiguchi, Yutaro; Ohta, Kinya; Yamashiro, Takahiro; Yuasa, Hiroaki
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Effects of Cimetidine and Dolutegravir on the Endogenous Drug-Drug Interaction Biomarkers for Organic Cation Transporter 2 and Multidrug and Toxin Extrusion Protein 1 in Healthy Volunteers
err2024-11-05
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errOAAI
errKoishikawa, Tomoki; Fujiwara, Kaku; Taskar, Kunal; Zamek-Gliszczynski, Maciej J.; Yoshida, Kenta; Chu, Xiaoyan; Hirabayashi, Hideki; Mao, Jialin; Rockich, Kevin; Takashima, Tadayuki; Yamaura, Yoshiyuki; Lai, Yurong; Tomoda, Yukana; Kito, Tomoko; Maeda, Kazuya; Furihata, Kenichi; Sugiyama, Yuichi; Kusuhara, Hiroyuki
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Utility of Biomarker-Informed Drug Interaction Evaluation in Drug Development and Regulatory Decision Making
err2024-09-09
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errOAAI
errIshiguro, Akihiro; Kusuhara, Hiroyuki; Kimoto, Emi; Miyoshi, So; Mizuno, Katsuhiko; Hoshino, Motohiro; Suzuki, Hiroshi
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Rapid in vivo evaluation system for cholestasis-related genes in mice with humanized bile acid profiles
err2024-04-01
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errOAAI
errWakasa, Kihiro; Tamura, Ryutaro; Osaka, Shuhei; Takei, Hajime; Asai, Akihiro; Nittono, Hiroshi; Kusuhara, Hiroyuki; Hayashi, Hisamitsu
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