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M

Michael M. Hann

medicines research centre

28H-index
91Paper Count
5.9KCitation Count
Published Papers 21
Publication Date
Orthogonal IMiD-Degron Pairs Induce Selective Protein Degradation in Cells
err2025-11-02
err0
errOAAI
errPatrick J. Brennan; Rebecca E. Saunders; Mary Spanou; Sarah E. Singleton; Marta Serafini; Liang Sun; Guillaume P. Heger; Agnieszka Konopacka; Ryan D. Beveridge; C. Cameron Taylor; Peter DePaola IV; Laurie Gordon; Shenaz B. Bunally; Aurore Saudemont; Andrew B. Benowitz; Carlos Martinez-Fleites; Danielle L. Schmitt; Robert Damoiseaux; Markus A. Queisser; Heeseon An; Charlotte M. Deane; Michael M. Hann; Lewis L. Brayshaw; Stuart J. Conway
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A Career doing STUFF
err2025-02-01
err0
PREAI
errHann, Michael M.
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Reactive fragments targeting carboxylate residues employing direct to biology, high-throughput chemistry
err2023-01-01
err8
errOAAI
errThomas, Ross P. P.; Grant, Emma K. K.; Dickinson, Eleanor R. R.; Zappacosta, Francesca; Edwards, Lee J. J.; Hann, Michael M. M.; House, David; Tomkinson, Nicholas C. O.; Bush, Jacob T. T.
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The PROTACtable genome
err2021-07-20
err143
PREAI
errSchneider, Melanie; Radoux, Chris J.; Hercules, Andrew; Ochoa, David; Dunham, Ian; Zalmas, Lykourgos-Panagiotis; Hessler, Gerhard; Ruf, Sven; Shanmugasundaram, Veerabahu; Hann, Michael M.; Thomas, Pam J.; Queisser, Markus A.; Benowitz, Andrew B.; Brown, Kris; Leach, Andrew R.
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A direct-to-biology high-throughput chemistry approach to reactive fragment screening
err2021-01-01
err27
errOAAI
errThomas, Ross P.; Heap, Rachel E.; Zappacosta, Francesca; Grant, Emma K.; Pogany, Peter; Besley, Stephen; Fallon, David J.; Hann, Michael M.; House, David; Tomkinson, Nicholas C. O.; Bush, Jacob T.
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A Photoaffinity-Based Fragment-Screening Platform for Efficient Identification of Protein Ligands
err2020-09-07
err44
errOAAI
errGrant, Emma K.; Fallon, David J.; Hann, Michael M.; Fantom, Ken G. M.; Quinn, Chad; Zappacosta, Francesca; Annan, Roland S.; Chung, Chun-wa; Bamborough, Paul; Dixon, David P.; Stacey, Peter; House, David; Patel, Vipulkumar K.; Tomkinson, Nicholas C. O.; Bush, Jacob T.
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Coupling the core of the anticancer drug etoposide to an oligonucleotide induces topoisomerase II-mediated cleavage at specific DNA sequences
err2018-02-13
err24
errOAAI
errLara, Lorena Infante; Fenner, Sabine; Ratcliffe, Steven; Isidro-Llobet, Albert; Hann, Michael; Bax, Ben; Osheroff, Neil
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Modulators of 14-3-3 Protein-Protein Interactions
err2017-10-02
err210
errOAAI
errStevers, Loes M.; Sijbesma, Eline; Botta, Maurizio; MacKintosh, Carol; Obsil, Tomas; Landrieu, Isabelle; Cau, Ylenia; Wilson, Andrew J.; Karawajczyk, Anna; Eickhoff, Jan; Davis, Jeremy; Hann, Michael; O'Mahony, Gavin; Doveston, Richard G.; Brunsveld, Luc; Ottmann, Christian
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What is the future for fragment-based drug discovery?
err2017-08-10
err6
PREAI
errKeseru, Gyorgy M.; Hann, Michael M.
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Prediction of intracellular exposure bridges the gap between target- and cell-based drug discovery
err2017-07-12
err74
errOAAI
errMateus, Andre; Gordon, Laurie J.; Wayne, Gareth J.; Almqvist, Helena; Axelsson, Hanna; Seashore-Ludlow, Brinton; Treyer, Andrea; Matsson, Par; Lundback, Thomas; West, Andy; Hann, Michael M.; Artursson, Per
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Stabilization of protein-protein interactions in drug discovery
err2017-07-11
err142
errOAAI
errAndrei, Sebastian A.; Sijbesma, Eline; Hann, Michael; Davis, Jeremy; O'Mahony, Gavin; Perry, Matthew W. D.; Karawajczyk, Anna; Eickhoff, Jan; Brunsveld, Luc; Doveston, Richard G.; Milroy, Lech-Gustav; Ottmann, Christian
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Design Principles for Fragment Libraries: Maximizing the Value of Learnings from Pharma Fragment-Based Drug Discovery (FBDD) Programs for Use in Academia
err2016-05-16
err178
PREAI
errKeseru, Gyoergy M.; Erlanson, Daniel A.; Ferenczy, Gyoergy G.; Hann, Michael M.; Murray, Christopher W.; Pickett, Stephen D.
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Structural basis of DNA gyrase inhibition by antibacterial QPT-1, anticancer drug etoposide and moxifloxacin
err2015-12-07
err123
errOAAI
errChan, Pan F.; Srikannathasan, Velupillai; Huang, Jianzhong; Cui, Haifeng; Fosberry, Andrew P.; Gu, Minghua; Hann, Michael M.; Hibbs, Martin; Homes, Paul; Ingraham, Karen; Pizzollo, Jason; Shen, Carol; Shillings, Anthony J.; Spitzfaden, Claus E.; Tanner, Robert; Theobald, Andrew J.; Stavenger, Robert A.; Bax, Benjamin D.; Gwynn, Michael N.
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Intracellular drug concentration and disposition - The missing link?
errMETHODS
IF4.3
err2014-07-01
err39
PREAI
errHann, Michael M.; Simpson, Graham L.
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Mycobacterium tuberculosis DNA gyrase ATPase domain structures suggest a dissociative mechanism that explains how ATP hydrolysis is coupled to domain motion
err2013-11-08
err42
PREAI
errAgrawal, Alka; Roue, Melanie; Spitzfaden, Claus; Petrella, Stephanie; Aubry, Alexandra; Hann, Michael; Bax, Benjamin; Mayer, Claudine
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