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任

任小梅 (Xiaomei Ren)

Shanghai Institute of Organic Chemistry

37H-index
168Paper Count
4.8KCitation Count
Published Papers 86
Publication Date
Design, synthesis and biological evaluation of a series of new, potent FLT3 PROTAC degraders with rigid linkers
err2026-09-19
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PREAI
errLicheng Zhou; Yinglong Chen; Jiahe Li; Yayuan Yang; Wenyan Liu; Yingfan Liu; Bohai Fan; Yang Zhou; Jinwei Zhang; Xiaomei Ren; Ke Ding; Weixue Huang; Zhen Wang; Fengtao Zhou
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The conformational–condensate code of GRB2: State switching, spatial organization, and therapeutic windows
err2026-08-24
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errOAAI
errJinwei Zhang; Jie Wang; Weixue Huang; Fengtao Zhou; Zhen Wang; Xiaomei Ren; Boris S. Shenkman; Ke Ding
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A regulator of amino acid catabolism controls Acinetobacter baumannii gut colonization
err2026-08-14
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errOAAI
errJohn H. Geary; Xiaomei Ren; Dziedzom A. Bansah; Ngoc T. T. Pham; Iván C. Acosta; Jim M. Camilleri; Bryan M. Kigongo; Jonathan D. Winkelman; Francis Alonzo; Matthew T. Henke; Lauren D. Palmer
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Discovery of a Potent; Selective and In Vivo Active Aurora A PROTAC Degrader from a Promiscuous Kinase Inhibitor
err2026-05-29
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PREAI
errYulin Mao; Meiying Zhang; Hao Tang; Jiaguo Li; Jie Wang; Fengtao Zhou; Jinwei Zhang; Weixue Huang; Xiaomei Ren; Ke Ding; Zhen Wang
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Inhibiting STING1 promotes recovery of cardiac function and structure after diabetic myocardial infarction by facilitating angiogenesis
err2026-05-12
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PREAI
errXinyue Wang; Yue Cai; Jia Xu; Guangyao Zang; Xiaomei Ren; Wenwen Sun; Lihua Li; Zheng Tao; Zhongqun Wang
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Amino acid competition shapes Acinetobacter baumannii gut carriage
err2025-08-04
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errOAAI
errXiaomei Ren; R. Mason Clark; Dziedzom A. Bansah; Elizabeth N. Varner; Connor R. Tiffany; Kanchan Jaswal; John H. Geary; Olivia A. Todd; Jonathan D. Winkelman; Elliot S. Friedman; Riley N. Jarrett; Babette S. Zemel; Gary D. Wu; Joseph P. Zackular; William H. DePas; Judith Behnsen; Lauren D. Palmer
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Ultrasound combined with microbubble enhanced renoprotective effects of NLRP3 inflammasome inhibitor MCC950 in CKD model
err2025-08-02
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errOAAI
errWen Wen†; Bin Tu†; Xiaomei Ren†; Yangli Liu; Rufang Jiang; Xiaofeng Wu; Jian Liu
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The design and synthesis of selective and potent selenium-containing KRASG12D inhibitors
err2025-07-24
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PREAI
errLiping Zhou; Yayuan Yang; Bingzhong Chen; Jie Wang; Ping Zhang; Yang Zhou; Jinwei Zhang; Xiaomei Ren; Zhen Wang; Weixue Huang; Zhimin Zhang; Xin Zhang; Shingpan Chan; Fengtao Zhou
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Discovery of YJZ5118: A Potent and Highly Selective Irreversible CDK12/13 Inhibitor with Synergistic Effects in Combination with Akt Inhibition
err2025-03-13
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PREAI
errYang, Jianzhang; Chang, Yu; Zhou, Kaijie; Huang, Weixue; Tien, Jean Ching-Yi; Zhang, Pujuan; Liu, Wenyan; Zhou, Licheng; Zhou, Yang; Ren, Xiaomei; Mannan, Rahul; Mahapatra, Somnath; Zhang, Yuping; Hamadeh, Rudana; Ervine, Grafton; Wang, Zhen; Wang, George Xiaoju; Chinnaiyan, Arul M.; Ding, Ke
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Discovery of the first potent ROR1 degrader for the treatment of non-small cell lung cancer
err2025-03-01
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PREAI
errLi, Jinlin; Li, Lin; Hou, Caiyun; Tian, Zhaodi; Zhou, Yang; Zhang, Jinwei; Ren, Xiaomei; Wang, Zhen; Huang, Weixue; Ding, Ke; Zhou, Fengtao
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Discovery of the first selective and potent PROTAC degrader for the pseudokinase TRIB2
err2025-01-01
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PREAI
errWen, Chaowei; Gajjala, Prathibha R.; Liu, Yihan; Chen, Bingzhong; Bal, Mehtab S.; Sutaria, Payal; Qiao, Yuanyuan; Zheng, Yang; Zhou, Yang; Zhang, Jinwei; Huang, Weixue; Ren, Xiaomei; Wang, Zhen; Ding, Ke; Chinnaiyan, Arul M.; Zhou, Fengtao
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Structure-Based Design of Head-to-Tail Macrocyclic PROTACs
errJACS AU
IF8.7
err2024-11-21
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errOAAI
errLi, Chungen; Chen, Yihan; Huang, Weixue; Qiu, Yudi; Huang, Shengjie; Zhou, Yang; Zhou, Fengtao; Xu, Jian; Ren, Xiaomei; Zhang, Jinwei; Wang, Zhen; Ding, Ming; Ding, Ke
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Discovery of ZLC491 as a Potent, Selective, and Orally Bioavailable CDK12/13 PROTAC Degrader
err2024-10-10
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errOAAI
errZhou, Licheng; Zhou, Kaijie; Chang, Yu; Yang, Jianzhang; Fan, Bohai; Su, Yuhan; Li, Zilu; Mannan, Rahul; Mahapatra, Somnath; Ding, Ming; Zhou, Fengtao; Huang, Weixue; Ren, Xiaomei; Xu, Jian; Wang, George Xiaoju; Zhang, Jinwei; Wang, Zhen; Chinnaiyan, Arul M.; Ding, Ke
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RGT-264 a highly potent, selective and orally bioavailable HPK1 (MAP4K1) inhibitor augments immune activation and anti-tumor immunity
err2024-10-01
err0
PREAI
errXiao, F.; Liu, H.; Wu, L.; Feng, S.; Liu, Y.; Xiao, H.; Li, H.; Huang, W.; Ren, X.; Ren, B.; Yao, L.; Lin, J.; Zhong, W.; Xie, Z.
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Analytical and clinical evaluation of a novel real-time PCR-based detection kit for Mpox virus
err2024-08-05
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errOAAI
errBunse, Till; Ziel, Anne; Hagen, Philipp; Rigopoulos, George; Yasar, Umit; Inan, Hakan; Koese, Gurbet; Eigner, Ulrich; Kaiser, Rolf; Bardeck, Nils; Koeffer, Jasmin; Kolb, Melissa; Ren, Xiaomei; Tan, Deyong; Dai, Lizhong; Protzer, Ulrike; Wettengel, Jochen M.
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Mechanisms of acquired resistance to HER2-Positive breast cancer therapies induced by HER3: A comprehensive review
err2024-08-01
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errOAAI
errGeng, Wujun; Thomas, Holly; Chen, Zhiyuan; Yan, Zhixiu; Zhang, Pujuan; Zhang, Meiying; Huang, Weixue; Ren, Xiaomei; Wang, Zhen; Ding, Ke; Zhang, Jinwei
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Amine response smartphone-based portable and intelligent polyvinyl alcohol films for real-time detection of shrimp freshness
err2024-08-01
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PREAI
errLuo, Man; Liu, Ji; Zhang, Yating; Wang, Tao; Ren, Xiaomei; Gui, Lijuan; Zhao, Junyuan; Zhang, Xuwei; Tang, Yunqing; Zeng, Ziting; Hou, Fengzhen; Zhong, Qifeng; Yuan, Zhenwei; Xu, Hui
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Discovery of LLC355 as an Autophagy-Tethering Compound for the Degradation of Discoidin Domain Receptor 1
err2024-05-10
err0
PREAI
errLiu, Lianchao; Zhao, Lijie; Yang, Lujun; Chai, Minxue; Liu, Zhengyong; Ma, Nan; Wang, Yongxing; Wu, Qinxue; Guo, Jing; Zhou, Fengtao; Huang, Weixue; Ren, Xiaomei; Wang, Jian; Ding, Ming; Wang, Zhen; Ding, Ke
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